Drugs / BI 1467335
last change Nov 2023 re-read 2 minutes ago

BI 1467335

targets AOC3, MAOB via inhibition

Developed for
diabetic retinopathy · NAFLD1
Investigated by
Boehringer Ingelheim

Trials 10 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 18 trials
Phase 1 NCT03979820 Jul 2019 → Apr 2020 Boehringer Ingelheim Terminated No outcome recorded
Phase 1 NCT03927209 Jun → Nov 2019 Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT03483506 Apr → Jun 2018 Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT03382509 Jan → Apr 2018 Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT03302091 Oct 2017 → Aug 2018 impaired renal function disease Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT03159455 Jun → Dec 2017 Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT02999191 Jan → Mar 2017 Boehringer Ingelheim Completed No outcome recorded
Phase 1 NCT02733627 Jul 2016 → Jul 2017 Boehringer Ingelheim Completed No outcome recorded
Phase 22 trials
Phase 2 NCT03238963 Sep 2017 → May 2020 diabetic retinopathy Boehringer Ingelheim Completed No outcome recorded
Phase 2 NCT03166735 Jun 2017 → Jun 2019 NAFLD1 Boehringer Ingelheim Completed No outcome recorded

Evidence & citations 4 cited values

Every value below carries the sentence it was read from. 11 sources stand behind the page.

FieldValueCited text
Known as BI 1467335 ClinicalTrials.gov intervention name — accepted as the source's own label NCT03159455
9

NCT02733627

NCT03979820

NCT03238963

NCT03382509

NCT03927209

NCT03166735

NCT03483506

NCT02999191

NCT03302091

Action Inhibit “These changes indicated that BI 1467335 dose-dependently inhibited AOC3 activity” PMID 37932258 Nov 2023
Route Oral “following oral administration” NCT02733627
Target AOC3 “an amine oxidase copper-containing 3 (AOC3) inhibitor” PMID 37932258 Nov 2023