Drugs / lesogaberan
last change Dec 2017 re-read 2 minutes ago

lesogaberan

also known as AZD3355

Small molecule targets GABBR1, GABBR2 via activation

Developed for
gastroesophageal reflux disease
Investigated by
AstraZeneca · Ministry of Science and Technology, Taiwan · National Taiwan University Hospital

Trials 10 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 14 trials
Phase 1 NCT00863161 Mar 2009 → Feb 2010 gastroesophageal reflux disease AstraZeneca Completed No outcome recorded
Phase 1 NCT00757419 Sep → Dec 2008 gastroesophageal reflux disease AstraZeneca Completed No outcome recorded
Phase 1 NCT00688402 Apr → Jun 2008 gastroesophageal reflux disease AstraZeneca Completed No outcome recorded
Phase 1 NCT00684190 Mar → Jun 2008 gastroesophageal reflux disease AstraZeneca Completed No outcome recorded
Phase 26 trials
Phase 2 NCT02818309 Jan 2015 → Nov 2017 gastroesophageal reflux disease National Taiwan University Hospital Unknown No outcome recorded
Phase 2 NCT01043185 Dec 2009 → May 2010 gastroesophageal reflux disease AstraZeneca Completed No outcome recorded
Phase 2 NCT01005251 Oct 2009 → Jul 2010 dyspepsia, gastroesophageal reflux disease AstraZeneca Completed No outcome recorded
Phase 2 NCT00703534 May 2008 → Jan 2009 dyspepsia, gastroesophageal reflux disease AstraZeneca Completed No outcome recorded
Phase 2 NCT00743444 Feb 2007 → Feb 2008 gastroesophageal reflux disease AstraZeneca Completed No outcome recorded
Phase 2 NCT00394472 Nov 2006 → Jun 2007 gastroesophageal reflux disease AstraZeneca Completed No outcome recorded

Evidence & citations 7 cited values

Every value below carries the sentence it was read from. 14 sources stand behind the page.

FieldValueCited text
Known as lesogaberan “The γ-aminobutyric acid type B-receptor agonist lesogaberan (AZD3355) has been developed for use in patients with gastroesophageal reflux disease (GERD) symptoms despite proton...” PMID 25407279 Nov 2014
2

NCT01005251

NCT02818309

Known as AZD3355 “Lesogaberan (AZD3355) is a novel γ-aminobutyric acid B-type receptor agonist designed to treat gastro-oesophageal reflux disease (GERD) by inhibiting transient lower...” PMID 22730470 Jun 2012
8

NCT00743444

NCT01043185

NCT00863161

NCT00688402

NCT00394472

NCT00703534

NCT00684190

NCT00757419

Action Activate “a novel gamma-aminobutyric acid type B receptor agonist” PMID 20451523 May 2010
2

“GABA-B receptor 1 agonist” CHEMBL448343

“GABA-B receptor 2 agonist” CHEMBL448343

Modality Small molecule CHEMBL448343
Route Oral “150 mg bid, oral, 7 days” NCT00684190
Target GABBR1 “GABA-B receptor 1 agonist” CHEMBL448343
Target GABBR2 “GABA-B receptor 2 agonist” CHEMBL448343