Drugs / Aminolevulinic Acid
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Aminolevulinic Acid

Diagnostic / imaging agent targets HMOX1 via activation

Developed for
actinic keratosis · glioblastoma · brain neoplasm · acne · glioma · malignant glioma · adult glioblastoma · brain cancer
+50 more · precancerous condition · skin carcinoma · anaplastic astrocytoma · anaplastic oligodendroglioma · astrocytoma (excluding glioblastoma) · basal cell carcinoma · giant cell glioblastoma · gliosarcoma · lichen planus, oral · neurofibromatosis type 1 · oral mucosa leukoplakia · primary brain neoplasm · skin cancer · skin squamous cell carcinoma · soft tissue sarcoma · actinic cheilitis · aortic valve disorder · breast cancer · chronic graft versus host disease · colon carcinoma · colorectal carcinoma · coronary artery disorder · Crohn disease · desmoid tumor caused by somatic mutation · epithelial skin neoplasm · erythroplakia · head and neck cancer · lentigo · leukemia · leukoplakia · lymphoma · malaria · mitral valve disorder · mycosis fungoides · neoplasm · nevoid basal cell carcinoma syndrome · oral cavity cancer · oral cavity squamous cell carcinoma · primary cutaneous T-cell lymphoma · radiation-induced disorder · rosacea · skin basal cell carcinoma · skin neoplasm · skin squamous cell carcinoma in situ · tinea unguium · ulcerative colitis · vulvar lichen sclerosus · seborrheic dermatitis · superficial multifocal basal cell carcinoma · type 2 diabetes mellitus
Investigated by
National Cancer Institute (NCI) · DUSA Pharmaceuticals, Inc. · Biofrontera Bioscience GmbH · photonamic GmbH & Co. KG · Roswell Park Cancer Institute · Biofrontera Inc.
+108 more · Joint Authority for Päijät-Häme Social and Health Care · NX Development Corp · Alpheus Medical, Inc. · David W. Roberts · Massachusetts General Hospital · National Institute of Neurological Disorders and Stroke (NINDS) · Sun Pharmaceutical Industries, Inc. · Tampere University · University of California, Davis · University of Münster · medac GmbH · Advocate Hospital System · Dartmouth-Hitchcock Medical Center · Hospices Civils de Lyon · Mayo Clinic · Oslo University Hospital · Shanghai Fudan-Zhangjiang Bio-Pharmaceutical Co., Ltd. · St. Joseph's Hospital and Medical Center, Phoenix · Tel-Aviv Sourasky Medical Center · The Center for Clinical and Cosmetic Research · University of California, Irvine · Abramson Cancer Center at Penn Medicine · Aligarh Muslim University · Andrew Sloan, MD · Barretos Cancer Hospital · Brigham and Women's Hospital · Carl Zeiss Meditec AG · Constantinos Hadjipanayis · Costas Hadjipanayis · Deutsche Krebshilfe e.V., Bonn (Germany) · Donald Basel · Edward Maytin, MD, PhD · Edward Nelson · Emerald Clinical Inc. · Endeavor Health · Fondazione I.R.C.C.S. Istituto Neurologico Carlo Besta · Fox Chase Cancer Center · French National Institute of Health and Medical Research · Fundación Instituto Valenciano de Oncología · George Washington University · Goldman, Butterwick, Fitzpatrick and Groff · Graceway Pharmaceuticals, LLC · Harry T Whelan, MD · Hemerion Therapeutics · Henry Ford Health System · Huslab, Finland · Icahn School of Medicine at Mount Sinai · Jawaharlal Nehru Medical College · Karkinos Healthcare Hospitals Ernakulam, Kerala, India · Laser and Skin Surgery Center of New York · Lee's Pharmaceutical Limited · Legacy Health System · LifePhotonic GmbH · Matthew R Quigley · Medical Dermatology Specialists · Medical University of Bialystok · Merete Haedersdal · Michael Vogelbaum, MD, PhD · MultiCare Health System Research Institute · NX PharmaGen · Nathalie Zeitouni · National Center for Advancing Translational Sciences (NCATS) · Neopharma Japan Co., Ltd. · Neuroscience Research Foundation · Nobelpharma · Northwestern University · Norwegian University of Science and Technology · Parexel · Princess Al-Johara Al-Ibrahim Cancer Research Center · Psoriasis Treatment Center of Central New Jersey · Päijänne Tavastia Central Hospital · Rhode Island Hospital · Rothman Institute Orthopaedics · Royal Cornwall Hospitals Trust · all 114 on the full record

Regulatory milestones approvals, filings & regulatory actions · 5 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansion US (FDA) AMELUZ 2024-10-04 fda.gov
Label expansions (2) US (FDA) LEVULAN 2010-03-12 – 2018-03-06 fda.gov
Approved EU (EMA) Gliolan 2007-09-07 europa.eu
Approved US (FDA) LEVULAN 1999-12-03 fda.gov

Trials 118 · started per year

today
US approved 1999
EU approved 2007
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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 04 trials
Phase 0 NCT07038278 Apr 2026 → Nov 2027 expected soft tissue sarcoma University of Colorado, Denver Not yet recruiting No outcome recorded
Phase 0 NCT07076472 Aug 2025 → Dec 2026 expected glioblastoma Mayo Clinic Recruiting No outcome recorded
Phase 0 NCT03281811 Nov 2017 → Feb 2020 mycosis fungoides Mayo Clinic Completed No outcome recorded
Phase 0 NCT00663910 Mar 2008 → Oct 2009 skin carcinoma The Cleveland Clinic Terminated No outcome recorded
Phase 121 trials
Phase 1 NCT07053852 Jun → Dec 2025 actinic keratosis, radiation-induced disorder Sherrif Ibrahim Completed No outcome recorded
Phase 1 NCT06665724 Jan 2025 → Feb 2026 anaplastic astrocytoma, anaplastic oligodendroglioma, glioblastoma University of Münster Completed No outcome recorded
Phase 1 NCT06623201 Oct 2024 → Dec 2026 expected basal cell carcinoma Nathalie Zeitouni Recruiting No outcome recorded
Phase 1 NCT06252727 Jul 2024 → Feb 2026 soft tissue sarcoma University of California, Davis Withdrawn No outcome recorded
Phase 1 NCT06039709 Jan 2024 → Dec 2026 expected glioblastoma Shayan Moosa, MD Recruiting No outcome recorded
Phase 1 NCT05362409 Jun 2022 → Dec 2024 malignant glioma Alpheus Medical, Inc. Completed No outcome recorded
Phase 1 NCT05060237 Dec 2021 → Apr 2023 actinic keratosis, keratosis Biofrontera Bioscience GmbH Completed No outcome recorded
Phase 1 NCT04044898 Jan → Jul 2021 acne Shanghai Fudan-Zhangjiang Bio-Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT04381806 Jul 2020 → Feb 2027 neoplasm Fox Chase Cancer Center Suspended No outcome recorded
Phase 1 NCT04319159 Mar → Sep 2020 actinic keratosis Biofrontera Bioscience GmbH Completed No outcome recorded
Phase 1/213 trials
Phase 1/2 NCT06307548 Jul 2024 → Jun 2027 expected colorectal carcinoma Roswell Park Cancer Institute Recruiting No outcome recorded
Phase 1/2 NCT05736406 Feb 2024 → Mar 2026 overdue glioblastoma Hemerion Therapeutics Active not recruiting No outcome recorded
Phase 1/2 NCT05590689 Nov 2022 → Jan 2028 expected glioblastoma University of Münster Recruiting No outcome recorded
Phase 1/2 NCT04164849 Nov 2019 → Oct 2023 Crohn disease University Hospital, Akershus Completed No outcome recorded
Phase 1/2 NCT03109353 Sep 2017 → Dec 2022 chronic graft versus host disease, primary cutaneous T-cell lymphoma St. Olavs Hospital Completed No outcome recorded
Phase 1/2 NCT03110159 Aug 2017 → Feb 2024 actinic keratosis, hyperpigmentation of the skin, skin carcinoma Medical Dermatology Specialists Completed No outcome recorded
Phase 1/2 NCT03638622 Mar 2017 → Oct 2020 oral cavity cancer Massachusetts General Hospital Completed No outcome recorded
Phase 1/2 NCT02367547 Mar 2015 → Sep 2018 basal cell carcinoma Joint Authority for Päijät-Häme Social and Health Care Unknown No outcome recorded
Phase 1/2 NCT02050243 Feb 2014 → Feb 2016 central nervous system cancer Tel-Aviv Sourasky Medical Center Unknown No outcome recorded
Phase 1/2 NCT01522677 Aug 2012 → May 2014 colon carcinoma Edward Nelson Withdrawn No outcome recorded
Phase 238 trials
Phase 2 NCT06876038 Sep 2026 → May 2028 expected lichen planus, oral, oral cavity squamous cell carcinoma, oral mucosa leukoplakia University of Massachusetts, Boston Not yet recruiting No outcome recorded
Phase 2 NCT07657975 Sep 2026 → Sep 2028 expected epilepsy Hospices Civils de Lyon Not yet recruiting No outcome recorded
Phase 2 NCT06907485 Aug 2026 → Feb 2028 expected brain neoplasm Costas Hadjipanayis Not yet recruiting No outcome recorded
Phase 2 NCT06948552 Apr 2026 → Dec 2027 expected renal pelvis/ureter urothelial carcinoma Henry Ford Health System Recruiting No outcome recorded
Phase 2 NCT07225621 Jan 2026 → Dec 2027 expected glioblastoma Alpheus Medical, Inc. Recruiting No outcome recorded
Phase 2 NCT06678867 Mar 2025 → Jun 2026 overdue brain neoplasm University College, London Not yet recruiting No outcome recorded
Phase 2 NCT06577311 Aug 2024 → Aug 2025 overdue skin squamous cell carcinoma The Center for Clinical and Cosmetic Research Recruiting No outcome recorded
Phase 2 NCT06159842 Aug 2023 → Sep 2024 skin squamous cell carcinoma in situ The Center for Clinical and Cosmetic Research Completed No outcome recorded
Phase 2 NCT04845919 Feb 2023 → Oct 2024 glioblastoma Fondazione I.R.C.C.S. Istituto Neurologico Carlo Besta Completed No outcome recorded
Phase 2 NCT05080764 Dec 2021 → Aug 2025 acne Biofrontera Inc. Completed No outcome recorded
Phase 317 trials
Phase 3 NCT07144852 Nov 2025 → Jan 2027 expected actinic keratosis Sun Pharmaceutical Industries, Inc. Recruiting No outcome recorded
Phase 3 NCT07144345 Nov 2025 → Jan 2027 expected actinic keratosis Sun Pharmaceutical Industries, Inc. Recruiting No outcome recorded
Phase 3 NCT06160492 Apr 2025 → Feb 2026 overdue Lee's Pharmaceutical Limited Recruiting No outcome recorded
Phase 3 NCT06417281 Jun 2024 → Aug 2025 malignant glioma, porphyria due to ALA dehydratase deficiency Shanghai Fudan-Zhangjiang Bio-Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 3 NCT05804370 May 2024 → Sep 2028 expected ovarian cancer NX Development Corp Recruiting No outcome recorded
Phase 3 NCT05662202 Dec 2022 → Sep 2025 actinic keratosis Biofrontera Inc. Completed No outcome recorded
Phase 3 NCT04815083 Apr 2021 → Oct 2024 breast cancer SBI ALApharma Canada, Inc. Terminated No outcome recorded
Phase 3 NCT04305470 Oct 2020 → Nov 2022 meningioma NX Development Corp Completed No outcome recorded
Phase 3 NCT04636242 Aug 2019 → Aug 2021 Rothman Institute Orthopaedics Unknown No outcome recorded
Phase 3 NCT03573401 Sep 2018 → Mar 2024 overdue skin basal cell carcinoma Biofrontera Inc. Active not recruiting No outcome recorded
Phase 412 trials
Phase 4 NCT06745999 May 2023 → May 2025 actinic keratosis Psoriasis Treatment Center of Central New Jersey Unknown No outcome recorded
Phase 4 NCT05359419 May 2022 → Aug 2023 skin neoplasm Goldman, Butterwick, Fitzpatrick and Groff Unknown No outcome recorded
Phase 4 NCT03963102 Oct 2019 → Mar 2024 actinic keratosis Royal Cornwall Hospitals Trust Terminated No outcome recorded
Phase 4 NCT04221126 Apr → Aug 2019 Merete Haedersdal Completed No outcome recorded
Phase 4 NCT02685592 Feb 2016 → Mar 2018 lentigo Joint Authority for Päijät-Häme Social and Health Care Completed No outcome recorded
Phase 4 NCT02647151 Dec 2015 → Mar 2016 actinic keratosis Fundación Instituto Valenciano de Oncología Unknown No outcome recorded
Phase 4 NCT02464709 Jun 2015 → Oct 2017 actinic keratosis Joint Authority for Päijät-Häme Social and Health Care Completed No outcome recorded
Phase 4 NCT03327831 Apr 2015 → Feb 2017 actinic keratosis University of California, Irvine Completed No outcome recorded
Phase 4 NCT02409732 Apr 2015 → Jul 2017 actinic cheilitis Dartmouth-Hitchcock Medical Center Completed No outcome recorded
Phase 4 NCT02075671 Apr 2014 → Aug 2019 rosacea George Washington University Completed No outcome recorded
Phase not applicable13 trials
NCT05228483 Nov 2021 → Nov 2023 vulvar lichen sclerosus Xijing Hospital Unknown No outcome recorded
NCT07536737 Sep 2021 → Jan 2023 lichen planus, oral Medical University of Bialystok Completed No outcome recorded
NCT02867722 Dec 2020 → Dec 2021 actinic keratosis, skin cancer Brigham and Women's Hospital Withdrawn No outcome recorded
NCT04631250 Nov 2018 → Jul 2020 acne Tel-Aviv Sourasky Medical Center Completed No outcome recorded
NCT03048240 May 2017 → Apr 2021 glioblastoma University Hospital, Lille Completed No outcome recorded
NCT03066843 Mar 2017 → Aug 2023 actinic keratosis Northwestern University Completed No outcome recorded
NCT03025724 Jan 2017 → Jan 2020 skin squamous cell carcinoma Rhode Island Hospital Unknown No outcome recorded
NCT02157623 Feb → Sep 2016 nevoid basal cell carcinoma syndrome Edward Maytin, MD, PhD Completed No outcome recorded
NCT02594644 Nov 2014 → Jun 2016 actinic keratosis University of California, Davis Completed No outcome recorded
NCT02119338 Feb 2014 → Jun 2017 glioma St. Joseph's Hospital and Medical Center, Phoenix Unknown No outcome recorded
Also used as a comparator or background therapy in 19 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT03114111 Comparator Jan 2017 → Dec 2019 seborrheic dermatitis University of California, Davis Completed No outcome recorded
Phase 12 trials
Phase 1 NCT02698293 Background Dec 2019 → Jan 2023 anus disorder, in situ carcinoma Abramson Cancer Center at Penn Medicine Withdrawn No outcome recorded
Phase 1 NCT03322293 Background Dec 2017 → Dec 2018 actinic keratosis University of California, San Francisco Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT02755142 Comparator Feb 2000 → Jun 2001 brain neoplasm medac GmbH Completed No outcome recorded
Phase 24 trials
Phase 2 NCT04391062 Background Sep 2021 → Mar 2024 glioblastoma University Hospital, Lille Completed No outcome recorded
Phase 2 NCT01556009 Comparator Apr 2012 → Dec 2015 nevoid basal cell carcinoma syndrome UCSF Benioff Children's Hospital Oakland Completed No outcome recorded
Phase 2 NCT00865878 Comparator May 2009 → Sep 2011 actinic keratosis DUSA Pharmaceuticals, Inc. Terminated No outcome recorded
Phase 2 NCT00706433 Comparator Mar 2007 → Jul 2008 acne DUSA Pharmaceuticals, Inc. Completed No outcome recorded
Phase 34 trials
Phase 3 NCT02144077 Comparator Jan 2014 → Nov 2015 basal cell carcinoma Biofrontera Bioscience GmbH Completed No outcome recorded
Phase 3 NCT01966120 Comparator Oct 2013 → Sep 2014 actinic keratosis Biofrontera Bioscience GmbH Completed No outcome recorded
Phase 3 NCT02799069 Comparator Apr 2008 → Aug 2009 actinic keratosis Biofrontera Bioscience GmbH Completed No outcome recorded
Phase 3 NCT02799082 Comparator Dec 2007 → Oct 2008 actinic keratosis Biofrontera Bioscience GmbH Completed No outcome recorded
Phase 42 trials
Phase 4 NCT02622594 Comparator Oct 2015 → Apr 2017 actinic keratosis Dermatology, Laser & Vein Specialists of the Carolinas Completed No outcome recorded
Phase 4 NCT01491711 Comparator Aug 2013 → Apr 2015 superficial multifocal basal cell carcinoma Maastricht University Medical Center Unknown No outcome recorded
Phase not applicable5 trials
NCT05488860 Background Jul 2022 → Jun 2024 keloid, plantar wart Xiangya Hospital of Central South University Unknown No outcome recorded
NCT02644187 Background Dec 2015 → Mar 2017 actinic keratosis Vastra Gotaland Region Completed No outcome recorded
NCT02379572 Comparator Jun 2015 → Jun 2020 glioblastoma University Hospital Tuebingen Completed No outcome recorded
NCT02481141 Comparator Jul 2014 → Jul 2015 type 2 diabetes mellitus SBI Pharmaceuticals Co, Ltd. Completed No outcome recorded
NCT00814918 Background Feb 2009 → Feb 2013 acne University of Chicago Withdrawn No outcome recorded

Evidence & citations 37 cited values

Every value below carries the sentence it was read from. 146 sources stand behind the page.

FieldValueCited text
Known as aminolevulinic acid Aminolevulinic acid 20% solution with blue light photodynamic therapy (ALA-PDT) has previously been shown to be superior to vehicle plus PDT (VEH-PDT) for treatment of AKs of...” PMID 38125671 Dec 2023
50

Aminolevulinic Acid (ALA) preparation and administration: The FDA-approved Aminolevulinic Acid (ALA) from Dusa Pharmaceuticals, Inc., Wilmington, Massachusetts (MA) will be...” NCT03638622

“PDT treatment consists of applying a gel containing aminolevulinic acid hydrochloride (licensed for clinical use as Ameluz®) to the abnormal area.” NCT03963102

“A Pharmacokinetics and Safety Study of Aminolevulinic Acid Hydrochloride Topical Powder in Subjects With Moderate to Severe Facial Acne Vulgaris.” NCT04044898

“A Proof of Principle Study of Aminolevulinic Acid (ALA) - Induced Fluorescence Detection in Resectable Non-Small Cell Lung Cancer” NCT01611584

“Photodynamic therapy with aminolevulinic acid (ALA) 20% topical solution is also an approved treatment for actinic keratoses.” NCT01203878

“The purpose of this study is to improve the current ECP technology using aminolevulinic acid (ALA) and UV light.” NCT03109353

“previous severe adverse reaction to topical 20% aminolevulinic acid (Kerastick)” NCT03025724

“10% aminolevulinic acid gel (Ameluz®, BF-200 ALA)” NCT05662202

NCT07076472

NCT02101931

NCT02728388

NCT01689935

NCT06307548

NCT00978081

NCT00706433

NCT01458587

NCT02075671

NCT02464709

NCT00671710

NCT07144852

NCT03322293

NCT01148966

NCT00054171

NCT00865878

NCT02137785

NCT00663910

NCT05359419

NCT00002963

NCT00747903

NCT00752323

NCT06252727

NCT01351519

NCT01575275

NCT02594644

NCT02622594

NCT00002975

NCT01812837

NCT02647151

NCT06159842

NCT06577311

NCT06623201

NCT02367547

NCT00571558

NCT07144345

NCT00524485

NCT02628236

NCT01556009

NCT02239679

NCT03327831

NCT00961090

Known as .delta.-aminolevulinic acid ChEMBL registry synonym — accepted as the source's own label CHEMBL601
Known as .delta.-aminolevulinic acid hydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL601
Known as 5 ala hcl (trivial name) ChEMBL registry synonym — accepted as the source's own label CHEMBL601
Known as 5-ALA “This is a prospective, single-arm feasibility study investigating the use of 5-aminolevulinic acid (5-ALA, Gleolan) to enhance intraoperative tumor visualization in patients...” NCT06948552
37

“The patient will receive 5-ALA ( 5-aminolevulinic acid hydrochloride),GLIOLAN drinkable 6h before surgery + lighting of the tumor bed by a red light source (laser with...” NCT04391062

“patient will be instructed to apply 5-aminolevulinic acid HCL topical solution to their shoulder prior to their surgery. 16 minutes before skin incision a blue light will be...” NCT04636242

“Only one phase III prospective randomized study, published in 2006, has assessed the performance of 5-aminolevulinic acid (5-ALA) fluorescence-guided surgery (FGS) for...” PMID 37856381 Oct 2023

“Here, we present a safety and feasibility trial after treating GBM intraoperatively by photodynamic therapy (PDT) after 5-aminolevulinic acid (5-ALA) administration and maximal...” PMID 33743128 Mar 2021

“5-aminolevulinic acid (5-ALA) is a photosensitizing agent which can induce photochemical reactions in tissues in response to an appropriate wavelength of light (red light 630-635nm).” NCT05228483

“This study is intended to investigate the utility, safety and efficacy of 5-aminolevulinic acid (5-ALA) induced brain tumor fluorescence during malignant brain tumor resection.” NCT00977795

“A multifaceted treatment approach can include nutritional supplements with antioxidant properties such as 5-aminolevulinic acid (5-ALA) with sodium ferrous citrate (SFC).” PMID 27738640 Sep 2016

“BACKGROUND: 5-aminolevulinic acid (5-ALA; GleolanTM, NX Development Corps., Lexington, USA) is approved for fluorescence-guided resections of suspected malignant gliomas.” PMID 36009108 Aug 2022

“Topical application of BF-200 ALA containing 7.8% 5-ALA (5-aminolevulinic acid) red light photodynamic therapy (PDT) utilizing BF-RhodoLED® after 1h incubation.” NCT05080764

“5-aminolevulinic acid (5-ALA) has been shown to be valuable in intraoperative marking of various cancers.” NCT02050243

“All patients will receive 5-aminolevulinic acid (5-ALA) in combination with blue light photopheresis.” NCT04164849

“using oral 5-aminolevulinic Acid (5-ALA) which results in fluorescence of the malignant cells” NCT01128218

“PD P 506 A is a dermal patch of 4 cm² in size loaded with 2 mg 5-ALA (as 5-ALA HCl) per cm².” NCT02355899

“PD P 506 A is a dermal patch of 4 cm² in size loaded with 2 mg 5-ALA (as 5-ALA HCl) per cm²” NCT03606122

“Topical application of BF-200 ALA containing 7.8% 5-ALA (5-aminolevulinic acid).” NCT05662202

“Topical application of BF-200 ALA containing 7.8% 5-ALA (5-aminolevulinic acid).” NCT03573401

“single oral dose of 5-aminolevulinic acid (5-ALA) oral solution powder” NCT06417281

“5-AMINOLEVULINIC ACID (5-ALA), is a non fluorescent prodrug.” NCT01898416

“5-aminolevulinic acid (5-ALA) (also known as Gliolan)” NCT01502605

“containing 7.8% 5-ALA (5-aminolevulinic acid)” NCT04319159

“5-Aminolevulinic Acid hydrochloride (5-ALA)” NCT07027670

“5-aminolevulinic acid (5-ALA)” NCT00241670

NCT04381806

NCT06039709

NCT06678867

NCT02119338

NCT05488860

NCT07038278

NCT01522677

NCT01459393

NCT07225621

NCT01445691

NCT02379572

NCT07657975

NCT00814528

NCT02050243

NCT00814918

Known as 5-ALA HCL “We report updated, exploratory analyses of OS, PFS, and health-related quality of life (HRQOL) for patients receiving intraoperative photodynamic therapy (PDT) with...” PMID 38753093 May 2024
3

5-ALA HCl (5-amino-levulenic acid) for oral solution (20 mg/kg) p.o. 6-8 hours prior to LIDU SDT” NCT07225621

“or orally administered aminolevulinic acid hydrochloride (5-ALA HCL)” NCT07076472

“5-aminolevulinic acid hydrochloride (5-ALA HCl, Gliolan®)” NCT06665724

Known as 5-ALA, 5-aminolevulic acid hydrochloride 5-ALA, 5-aminolevulic acid hydrochlorideNCT01167322
Known as 5-amino-levulenic acid “5-ALA HCl (5-amino-levulenic acid) for oral solution (20 mg/kg) p.o. 6-8 hours prior to LIDU SDT” NCT07225621
Known as 5-aminolaevulinic acid “Following topical application of 5-aminolaevulinic acid, the substance is metabolized to protoporphyrin IX, a photoactive compound which accumulates intracellularly in the...” NCT02647151
Known as 5-aminolevulinic acid “This is a prospective, randomized controlled trial to evaluation the ability of 5-aminolevulinic acid HCL topical solution photodynamic therapy to decrease the colonization of...” NCT04636242
54

“The aim of this study is to test the effectiveness and safety of the medicine Ameluz® (5-aminolevulinic acid) in comparison to methyl-aminolevulinate (MAL), used with...” NCT02144077

“The drug, 5-aminolevulinic acid (ALA), which leads to intracellular accumulation of fluorescent porphyrins in gliomas will be used under investigation for identification and...” NCT01116661

“Only one phase III prospective randomized study, published in 2006, has assessed the performance of 5-aminolevulinic acid (5-ALA) fluorescence-guided surgery (FGS) for...” PMID 37856381 Oct 2023

“Here, we present a safety and feasibility trial after treating GBM intraoperatively by photodynamic therapy (PDT) after 5-aminolevulinic acid (5-ALA) administration and maximal...” PMID 33743128 Mar 2021

“BACKGROUND: 5-aminolevulinic acid (5-ALA; GleolanTM, NX Development Corps., Lexington, USA) is approved for fluorescence-guided resections of suspected malignant gliomas.” PMID 36009108 Aug 2022

“A multifaceted treatment approach can include nutritional supplements with antioxidant properties such as 5-aminolevulinic acid (5-ALA) with sodium ferrous citrate (SFC).” PMID 27738640 Sep 2016

“Topical application of BF-200 ALA containing 7.8% 5-ALA (5-aminolevulinic acid) red light photodynamic therapy (PDT) utilizing BF-RhodoLED® after 1h incubation.” NCT05080764

5-aminolevulinic acid (5-ALA) fluorescence-guided resection of high-grade gliomas (HGG) increases the extent of resection (EOR) and progression-free survival.” PMID 36656388 Jan 2023

“The aim of this study is to assess the pharmacokinetics (PK) of the parent drug 5-aminolevulinic acid (ALA) and its active metabolite protoporphyrin IX (PpIX)” NCT04319159

“This study aims to determine the safety and utility of using 5-Aminolevulinic Acid (ALA) in removing malignant brain tumors during surgery.” NCT01403311

“For 5-ALA guided glioma resections patients have to drink 100ml of a solution with 5-Aminolevulinic acid 4-6 hours before surgery.” NCT02379572

5-aminolevulinic acid hydrochloride (Gliolan), orally, 40 mg/kg administered approximately 4-6 hours before light administration.” NCT02698293

5-aminolevulinic acid (5-ALA) associated with 20% dimethyl sulfoxide (DMSO) and 3% ethylene diamine acid (EDTA) emulsion” NCT01459393

“ALA (5-aminolevulinic acid) will be applied to subjects' skin for either zero time incubation or one hour incubation” NCT03066843

“orally-administered 5-aminolevulinic acid (ALA) given as a radiosensitizer prior to low-dose radiation therapy (RT)” NCT04381806

“A 5% 5-aminolevulinic acid (ALA) mucoadhesive formulation is applied topically to oral lichen planus lesions.” NCT07536737

5-aminolevulinic acid (5-ALA) has been shown to be valuable in intraoperative marking of various cancers.” NCT02050243

5-aminolevulinic acid hydrochloride (5-ALA HCl) administration + brain cavity illumination” NCT05736406

“Topical application of BF-200 ALA gel containing 78 mg/g 5-aminolevulinic acid (ALA).” NCT02799069

“Topical application of BF-200 ALA containing 7.8% 5-ALA (5-aminolevulinic acid).” NCT03573401

“Topical application of BF-200 ALA containing 7.8% 5-ALA (5-aminolevulinic acid).” NCT05662202

5-aminolevulinic acid \[5-ALA\] administered orally 20 mg/kg every 4 weeks” NCT05362409

“BF-200 ALA (containing the active ingredient 5 - aminolevulinic acid- ALA)” NCT02799030

“single oral dose of 5-aminolevulinic acid (5-ALA) oral solution powder” NCT06417281

“Levulan (5-aminolevulinic acid) photodynamic therapy - Dose level 1” NCT01682811

“naturally occurring amino acid, 5-aminolevulinic acid (5-ALA)” NCT01128218

“Flourescein = Fluorescite; ALA = 5-Aminolevulinic AcidNCT02691923

5-aminolevulinic acid compounded in a cream” NCT04221126

NCT00571974

NCT04164849

NCT06948552

NCT01898416

NCT02644187

NCT00241670

NCT07027670

NCT06665724

NCT05228483

NCT04738162

NCT04631250

NCT04469699

NCT00870779

NCT07536737

NCT06417281

NCT03897491

NCT06160492

NCT04020653

NCT06876038

NCT02191488

NCT01491711

NCT00977795

NCT01502280

NCT01502605

NCT03109353

NCT04845919

Known as 5-aminolevulinic acid HCL “This is a prospective, randomized controlled trial to evaluation the ability of 5-aminolevulinic acid HCL topical solution photodynamic therapy to decrease the colonization of...” NCT04636242
Known as 5-Aminolevulinic Acid hydrochloride “The patient will receive 5-ALA ( 5-aminolevulinic acid hydrochloride),GLIOLAN drinkable 6h before surgery + lighting of the tumor bed by a red light source (laser with...” NCT04391062
6

“We report updated, exploratory analyses of OS, PFS, and health-related quality of life (HRQOL) for patients receiving intraoperative photodynamic therapy (PDT) with...” PMID 38753093 May 2024

“NPC-07 (5-aminolevulinic acid hydrochloride) induced tissue fluorescence” NCT01167322

5-aminolevulinic acid hydrochloride (5-ALA HCl, Gliolan®)” NCT06665724

5-Aminolevulinic acid Hydrochloride (Gliolan®)” NCT06948552

5-Aminolevulinic Acid hydrochloride (5-ALA)” NCT07027670

NCT05101798

Known as 5-aminolevulinic acid nanoemulsion ClinicalTrials.gov intervention name — accepted as the source's own label NCT02685592
Known as 5-aminolévulinique acid ClinicalTrials.gov intervention name — accepted as the source's own label NCT01811121
Known as ALA “The drug, 5-aminolevulinic acid (ALA), which leads to intracellular accumulation of fluorescent porphyrins in gliomas will be used under investigation for identification and...” NCT01116661
25

“The objective of this study was to detect 5-aminolevulinic acid (ALA)-induced tumor fluorescence from glioma below the surface of the surgical field by using red-light illumination.” PMID 28777025 Aug 2017

“Individual lesions on patients within each stratum are randomized to receive either a 4-5 or 18-24 hour application of aminolevulinic acid (ALA).” NCT00002975

“This study aims to determine the safety and utility of using 5-Aminolevulinic Acid (ALA) in removing malignant brain tumors during surgery.” NCT01403311

“The nanoemulsion-based 10% aminolevulinic acid (ALA) hydrochloride gel BF-200 ALA optimizes epidermal penetration of its active ingredient” PMID 34633154 Oct 2021

“A Proof of Principle Study of Aminolevulinic Acid (ALA) - Induced Fluorescence Detection in Resectable Non-Small Cell Lung Cancer” NCT01611584

“topically applied aminolevulinic acid (ALA) into the lesions of patients with primary basal cell and squamous cell carcinomas.” NCT00002963

“Photodynamic therapy with aminolevulinic acid (ALA) 20% topical solution is also an approved treatment for actinic keratoses.” NCT01203878

“PDT involves the topical application of aminolevulinic acid (ALA), or one of its derivatives, as a photosensitizing agent.” NCT03322293

“Aminolevulinic acid (ALA) is a naturally occurring metabolite in the synthesis of pathway of cellular heme production.” NCT04636242

“20% aminolevulinic acid HCL (ALA) applied topically for 90 +/- 30 minutes prior to treatment with 10 j/cm2 blue light.” NCT00865878

“orally-administered 5-aminolevulinic acid (ALA) given as a radiosensitizer prior to low-dose radiation therapy (RT)” NCT04381806

“The purpose of this study is to improve the current ECP technology using aminolevulinic acid (ALA) and UV light.” NCT03109353

“A 5% 5-aminolevulinic acid (ALA) mucoadhesive formulation is applied topically to oral lichen planus lesions.” NCT07536737

“Photodynamic therapy (PDT) uses a drug called ALA (aminolevulinic acid), which is marketed as Levulan®.” NCT01689935

“Topical application of BF-200 ALA gel containing 78 mg/g 5-aminolevulinic acid (ALA).” NCT02799069

“Aminolevulinic Acid 20% Topical Solution (Levulan® Kerastick® Applicators) (ALA)” NCT06159842

“Patients receive topical ALA topical (aminolevulinic acid) 2 hours before PDT.” NCT00524485

“BF-200 ALA (containing the active ingredient 5 - aminolevulinic acid- ALA)” NCT02799030

“aminolevulinic acid HCL (ALA)” NCT06623201

“Aminolevulinic Acid PDT (ALA)” NCT01458587

“Aminolevulinic Acid (ALA)” NCT02137785

“Aminolevulinic Acid (ALA)” NCT02628236

“Aminolevulinic Acid (ALA)” NCT02622594

NCT02691923

NCT03066843

Known as ALA HCl “Reformulated Levulan Kerastick containing aminolevulinic acid hydrochloride (ALA HCl), 20%” NCT07144345
Known as Alabel ChEMBL registry synonym — accepted as the source's own label CHEMBL601
Known as Alaglio ChEMBL registry synonym — accepted as the source's own label CHEMBL601
Known as Ameluz “PDT treatment consists of applying a gel containing aminolevulinic acid hydrochloride (licensed for clinical use as Ameluz®) to the abnormal area.” NCT03963102
8

“A 0,25mm-thick layer of BF-200 ALA (aminolevulinic acid, Ameluz®) light sensitizer gel is applied on one randomized treatment side of face.” NCT02464709

“using 5-aminolevulinic acid nanoemulsion (BF-200 ALA, Ameluz®) as a light sensitizing cream” NCT02685592

AMELUZ® (aminolevulinic acid hydrochloride) gel, 10%” NCT05359419

“10% aminolevulinic acid gel (Ameluz®, BF-200 ALA)” NCT05662202

“BF-200 ALA 10% gel (Ameluz®)” NCT04319159

“BF-200 ALA (Ameluz®)” NCT05060237

NCT06745999

NCT07053852

Known as Aminolevulinic acid (ALA) Aminolevulinic acid (ALA)NCT03638622
2

NCT02281136

NCT03114111

Known as aminolevulinic acid HCL “A Pharmacokinetic Study of Levulan Kerastick (Aminolevulinic Acid HCl) for Topical Solution, 20% Under Maximal Use Conditions” NCT02628236
5

“20% aminolevulinic acid HCL (ALA) applied topically for 90 +/- 30 minutes prior to treatment with 10 j/cm2 blue light.” NCT00865878

“Drug intervention: Aminolevulinic acid HCl (ALA) topical solution 20%” NCT03322293

“LEVULAN® KERASTICK® (aminolevulinic acid HCl) topical solution, 20%” NCT05359419

aminolevulinic acid HCL (ALA)” NCT06623201

NCT02867722

Known as aminolevulinic acid HCL (ALA) “Levulan® Kerastick® containing 20% aminolevulinic acid HCL (ALA, active study drug)” NCT00706433
Known as aminolevulinic acid hydrochloride “Participants will have their facial Cutaneous Squamous Cell Carcinoma in situ (SCCis) prepped then treated with Aminolevulinic acid hydrochloride 10% topical gel (Ameluz ®),...” NCT06577311
8

AMINOLEVULINIC ACID HYDROCHLORIDE (ALA) gel 78mg/g. Intervention: Just one application of the product in the actinic keratosis lesions before the photodynamic therapy” NCT02647151

“Reformulated Levulan Kerastick containing aminolevulinic acid hydrochloride (ALA HCl), 20%” NCT07144345

“AMELUZ® (aminolevulinic acid hydrochloride) gel, 10%” NCT05359419

“Drug: aminolevulinic acid hydrochlorideNCT00571558

NCT04815083

NCT02409732

NCT03281811

NCT06907485

Known as BF-200 ALA “A 0,25mm-thick layer of BF-200 ALA (aminolevulinic acid, Ameluz®) light sensitizer gel is applied on one randomized treatment side of face.” NCT02464709
8

“The nanoemulsion-based 10% aminolevulinic acid (ALA) hydrochloride gel BF-200 ALA optimizes epidermal penetration of its active ingredient” PMID 34633154 Oct 2021

“using 5-aminolevulinic acid nanoemulsion (BF-200 ALA, Ameluz®) as a light sensitizing cream” NCT02685592

“10% aminolevulinic acid gel (Ameluz®, BF-200 ALA)” NCT05662202

“Drug: BF200-ALA/5-aminolevulinic acid” NCT02644187

NCT01966120

NCT05060237

NCT02799082

NCT01893203

Known as Gleolan “This is a prospective, single-arm feasibility study investigating the use of 5-aminolevulinic acid (5-ALA, Gleolan) to enhance intraoperative tumor visualization in patients...” NCT06948552
3

“The combination of 5-ALA (Gleolan) and LIFU is collectively known as sonodynamic therapy (SDT).” NCT06039709

NCT04305470

NCT05804370