Drugs / CB-839

Trials 23 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 110 trials
Phase 1 NCT03944902 Sep 2021 → Jan 2022 ovarian cancer University of Alabama at Birmingham Terminated No outcome recorded
Phase 1 NCT04250545 Oct 2020 → Nov 2025 overdue metastatic malignant neoplasm in the brain, neoplastic meningitis, non-small cell lung carcinoma National Cancer Institute (NCI) Active not recruiting No outcome recorded
Phase 1 NCT04607512 Oct → Dec 2020 Calithera Biosciences, Inc Completed No outcome recorded
Phase 1 NCT04540965 Sep → Dec 2020 Calithera Biosciences, Inc Completed No outcome recorded
Phase 1 NCT03798678 Jul 2019 → Nov 2023 overdue plasma cell myeloma National Cancer Institute (NCI) Active not recruiting No outcome recorded
Phase 1 NCT03528642 May 2019 → Sep 2026 expected astrocytoma, IDH-mutant, grade 2, astrocytoma, IDH-mutant, grade 3 National Cancer Institute (NCI) Active not recruiting No outcome recorded
Phase 1 NCT02944435 Oct → Nov 2016 Calithera Biosciences, Inc Completed No outcome recorded
Phase 1 NCT02071927 Mar 2014 → Oct 2016 acute lymphoblastic leukemia, acute myeloid leukemia Calithera Biosciences, Inc Completed No outcome recorded
Phase 1 NCT02071888 Feb 2014 → Apr 2016 T-cell non-Hodgkin lymphoma, Waldenstrom macroglobulinemia, plasma cell myeloma Calithera Biosciences, Inc Completed No outcome recorded
Phase 1 NCT02071862 Feb 2014 → Mar 2019 gastrointestinal stromal tumor, mesothelioma, non-small cell lung carcinoma, renal cell carcinoma +1 Calithera Biosciences, Inc Completed No outcome recorded
Phase 1/27 trials
Phase 1/2 NCT07223528 Aug 2026 → Sep 2028 expected pulmonary hypertension Chan, Stephen, MD, PhD Not yet recruiting No outcome recorded
Phase 1/2 NCT03831932 Mar 2020 → Jun 2024 overdue non-small cell lung carcinoma National Cancer Institute (NCI) Active not recruiting No outcome recorded
Phase 1/2 NCT03875313 May 2019 → Jul 2020 clear cell renal carcinoma, colorectal cancer, triple-negative breast carcinoma Calithera Biosciences, Inc Terminated No outcome recorded
Phase 1/2 NCT03047993 Nov 2017 → Mar 2023 acute myeloid leukemia with multilineage dysplasia, chronic myelomonocytic leukemia, myelodysplastic syndrome M.D. Anderson Cancer Center Completed No outcome recorded
Phase 1/2 NCT03263429 Aug 2017 → Aug 2023 colorectal cancer Vanderbilt-Ingram Cancer Center Completed No outcome recorded
Phase 1/2 NCT02861300 Sep 2016 → Jan 2023 colon carcinoma, rectal cancer David Bajor, MD Completed No outcome recorded
Phase 1/2 NCT02771626 Aug 2016 → Apr 2020 clear cell renal carcinoma, melanoma, non-small cell lung carcinoma Calithera Biosciences, Inc Terminated No outcome recorded
Phase 26 trials
Phase 2 NCT05521997 Jul 2026 → Oct 2032 expected cervical carcinoma Washington University School of Medicine Not yet recruiting No outcome recorded
Phase 2 NCT04824937 Jul → Dec 2021 metastatic prostate carcinoma Massachusetts General Hospital Unknown No outcome recorded
Phase 2 NCT04265534 Jul 2020 → Nov 2021 non-small cell lung carcinoma Calithera Biosciences, Inc Terminated No outcome recorded
Phase 2 NCT03872427 Dec 2019 → Oct 2023 overdue malignant peripheral nerve sheath tumor, metastatic malignant neoplasm National Cancer Institute (NCI) Active not recruiting No outcome recorded
Phase 2 NCT03428217 Apr 2018 → Aug 2020 clear cell renal carcinoma Calithera Biosciences, Inc Completed No outcome recorded
Phase 2 NCT03057600 May 2017 → Nov 2019 triple-negative breast carcinoma Calithera Biosciences, Inc Completed No outcome recorded
Also used as a comparator or background therapy in 1 trial
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 2 NCT03163667 Comparator Sep 2017 → Apr 2019 clear cell renal carcinoma Calithera Biosciences, Inc Completed No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 25 sources stand behind the page.

FieldValueCited text
Known as CB-839 “A Phase 1b Trial of Telaglenastat (CB-839) HCI in Combination With Radiation Therapy and Temozolomide in Patients With IDH-Mutated Diffuse Astrocytoma and Anaplastic Astrocytoma” NCT03528642
14

“Eligible participants will be taking 800 mg Telaglenastat (CB-839) by mouth with food twice a day for a total of 12 weeks.” NCT07223528

“Participants will receive a fixed dose of Niraparib and CB-839, 800mg.” NCT03944902

NCT02771626

NCT02071862

NCT02944435

NCT03875313

NCT03163667

NCT03047993

NCT03263429

NCT02071888

NCT03057600

NCT02861300

NCT02071927

NCT03428217

Known as telaglenastat telaglenastat (CB-839), a selective glutaminase inhibitor, combined with azacytidine (AZA)” PMID 39300320 Sep 2024
9

NCT07223528

NCT03798678

NCT04607512

NCT04265534

NCT03528642

NCT05521997

NCT03872427

NCT04824937

NCT04540965

Known as Telaglenastat Hydrochloride “Testing Whether Cancers With Specific Mutations Respond Better to Glutaminase Inhibitor, Telaglenastat Hydrochloride, Anti-Cancer Treatment, BeGIN Study” NCT03872427
3

“Drug: Telaglenastat HydrochlorideNCT03528642

NCT03831932

NCT04250545

Action Inhibit “CB-839, a potent and selective inhibitor of the first enzyme in glutamine utilization, glutaminase” NCT02071862
Route Oral “CB-839 administered as oral capsules two (BID) or three times daily (TID)” NCT02071862