Drugs / decernotinib
last change Apr 2016 re-read 2 minutes ago

decernotinib

also known as VX-509 · Adelatinib · VRT-831509

Small molecule targets JAK3 via inhibition

Developed for
rheumatoid arthritis
Investigated by
Vertex Pharmaceuticals Incorporated

Trials 6 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT01886209 Jun → Aug 2013 Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 1 NCT00789126 Oct 2008 → ? Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 23 trials
Phase 2 NCT01754935 Jan 2013 → Jan 2014 rheumatoid arthritis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 2 NCT01590459 Apr 2012 → Jul 2014 rheumatoid arthritis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 2 NCT01052194 Feb 2010 → Jul 2011 rheumatoid arthritis Vertex Pharmaceuticals Incorporated Completed No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT01830985 Apr 2013 → Jul 2014 rheumatoid arthritis Vertex Pharmaceuticals Incorporated Completed No outcome recorded

Press releases naming this drug 4 releases

DateIssuerRelease
2013-10-18 Vertex Pharmaceuticals Incorporated Oral Selective JAK3 Inhibitor VX-509 Showed Statistically Significant Improvements in Signs and Symptoms of Rheumatoid Arthritis After 12 Weeks of Treatment in Phase 2b Study vrtx.com
2011-11-05 Vertex Pharmaceuticals Incorporated Phase 2 Data for Selective Oral JAK3 Inhibitor VX-509 Show Significant Improvements in Signs and Symptoms of Rheumatoid Arthritis vrtx.com
2011-10-24 Vertex Pharmaceuticals Incorporated Vertex Announces Presentation of New Data for Oral JAK3 Inhibitor VX-509 at Annual Meeting of the American College of Rheumatology vrtx.com
2011-09-06 Vertex Pharmaceuticals Incorporated Phase 2a Study of Selective Oral JAK3 Inhibitor VX-509 Showed Significant Improvements in Signs and Symptoms of Rheumatoid Arthritis vrtx.com

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 8 sources stand behind the page.

FieldValueCited text
Known as decernotinib “Efficacy of VX-509 (decernotinib) in combination with a disease-modifying antirheumatic drug in patients with rheumatoid arthritis: clinical and MRI findings.” PMID 27084959 Apr 2016
Known as Adelatinib ChEMBL registry synonym — accepted as the source's own label CHEMBL3039513
Known as VRT-831509 ChEMBL registry synonym — accepted as the source's own label CHEMBL3039513
Known as VX-509 ClinicalTrials.gov intervention name — accepted as the source's own label NCT01886209
5

NCT00789126

NCT01052194

NCT01590459

NCT01754935

NCT01830985

Action Inhibit “VX-509, a JAK3 inhibitor” NCT01052194
Modality Small molecule CHEMBL3039513
Route Oral “50 mg oral tablet” NCT01590459
Target JAK3 “VX-509, a JAK3 inhibitor” NCT01052194