Drugs / ispronicline
last change May 2014 re-read 2 minutes ago

ispronicline

also known as AZD3480 · Isproniclina · TC-01734 · TC-1734

Small molecule

Developed for
Alzheimer disease · attention deficit-hyperactivity disorder · cognitive disorder · schizophrenia
Investigated by
AstraZeneca · Targacept Inc.

Trials 12 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 17 trials
Phase 1 NCT00713765 Dec 2008 Alzheimer disease AstraZeneca Terminated No outcome recorded
Phase 1 NCT00777361 Oct 2008 → Oct 2009 Alzheimer disease AstraZeneca Terminated No outcome recorded
Phase 1 NCT00689559 Mar 2008 → Apr 2009 Alzheimer disease AstraZeneca Completed No outcome recorded
Phase 1 NCT00686179 Jan → Aug 2008 AstraZeneca Completed No outcome recorded
Phase 1 NCT00686413 Jan → Aug 2008 AstraZeneca Completed No outcome recorded
Phase 1 NCT00692510 Nov 2007 → Sep 2008 Alzheimer disease AstraZeneca Completed No outcome recorded
Phase 1 NCT00689637 Sep 2007 → Feb 2009 Alzheimer disease AstraZeneca Completed No outcome recorded
Phase 25 trials
Phase 2 NCT01466088 Oct 2011 → May 2014 Alzheimer disease Targacept Inc. Completed No outcome recorded
Phase 2 NCT00683462 May 2008 → Jul 2009 attention deficit-hyperactivity disorder AstraZeneca Completed No outcome recorded
Phase 2 NCT00528905 Aug 2007 → Oct 2008 schizophrenia AstraZeneca Completed No outcome recorded
Phase 2 NCT00501111 Jul 2007 → Aug 2008 Alzheimer disease AstraZeneca Completed No outcome recorded
Phase 2 NCT00109564 Jan → Oct 2005 cognitive disorder Targacept Inc. Completed No outcome recorded

Evidence & citations 8 cited values

Every value below carries the sentence it was read from. 15 sources stand behind the page.

FieldValueCited text
Known as ispronicline ClinicalTrials.gov intervention name — accepted as the source's own label NCT00109564
Known as AZD3480 “The objective of this study was to assess the safety, tolerability and efficacy of TC-1734 (AZD3480), a selective α4β2 nicotinic agonist, in the treatment of age-associated...” PMID 20542923 Jun 2010
11

NCT00777361

NCT00713765

NCT00686413

NCT00689637

NCT00528905

NCT00689559

NCT00692510

NCT00686179

NCT00501111

NCT00683462

NCT01466088

Known as Isproniclina ChEMBL registry synonym — accepted as the source's own label CHEMBL188462
Known as TC-01734 ChEMBL registry synonym — accepted as the source's own label CHEMBL188462
Known as TC-1734 “This was a within-subjects, randomized, placebo-controlled double-blind trial of the nicotinic agonist AZD3480 (also termed TC-1734) at doses of 5 mg and 50 mg and placebo in...” PMID 23856296 Jul 2013
Action Activate “a selective α4β2 nicotinic agonist” PMID 20542923 Jun 2010
Modality Small molecule CHEMBL188462
Route Oral “Subjects were randomly assigned to receive orally 25 mg (n = 59), 50 mg (n = 68) TC-1734 (AZD3480) or placebo” PMID 20542923 Jun 2010