Drugs / SHR4640
last change Feb 2026 re-read 2 minutes ago

SHR4640

also known as Ruzinurad

Small molecule targets SLC22A12 via inhibition

Developed for
gout
Investigated by
Jiangsu HengRui Medicine Co., Ltd. · Atridia Pty Ltd.

Trials 19 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 113 trials
Phase 1 NCT06196580 Jan → Feb 2024 gout Jiangsu HengRui Medicine Co., Ltd. Completed No outcome recorded
Phase 1 NCT05954169 Aug 2023 → Jul 2024 Jiangsu HengRui Medicine Co., Ltd. Completed No outcome recorded
Phase 1 NCT04850638 Jun → Sep 2021 Jiangsu HengRui Medicine Co., Ltd. Completed No outcome recorded
Phase 1 NCT04620408 Dec 2020 → Jan 2021 Jiangsu HengRui Medicine Co., Ltd. Unknown No outcome recorded
Phase 1 NCT04586803 Oct → Nov 2020 gout Jiangsu HengRui Medicine Co., Ltd. Unknown No outcome recorded
Phase 1 NCT04305392 Aug 2020 → Dec 2022 Jiangsu HengRui Medicine Co., Ltd. Unknown No outcome recorded
Phase 1 NCT04260373 Mar → Apr 2020 Jiangsu HengRui Medicine Co., Ltd. Completed No outcome recorded
Phase 1 NCT04157959 Oct 2019 → Jun 2020 Jiangsu HengRui Medicine Co., Ltd. Unknown No outcome recorded
Phase 1 NCT03211403 Jul 2017 → Feb 2018 gout Atridia Pty Ltd. Completed No outcome recorded
Phase 1 NCT03131583 Feb 2017 → Jan 2018 gout Jiangsu HengRui Medicine Co., Ltd. Completed No outcome recorded
Phase 24 trials
Phase 2 NCT07362355 Feb 2026 → Jul 2027 expected gout Jiangsu HengRui Medicine Co., Ltd. Recruiting No outcome recorded
Phase 2 NCT05513976 Sep 2022 → May 2023 gout Jiangsu HengRui Medicine Co., Ltd. Unknown No outcome recorded
Phase 2 NCT04180982 Dec 2019 → Jul 2020 Jiangsu HengRui Medicine Co., Ltd. Unknown No outcome recorded
Phase 2 NCT03185793 Jul 2017 → Jul 2018 Jiangsu HengRui Medicine Co., Ltd. Completed No outcome recorded
Phase 32 trials
Phase 3 NCT04956432 Jun 2021 → Dec 2023 gout Jiangsu HengRui Medicine Co., Ltd. Completed No outcome recorded
Phase 3 NCT04052932 Jul 2019 → Jul 2021 gout Jiangsu HengRui Medicine Co., Ltd. Completed No outcome recorded

Evidence & citations 6 cited values

Every value below carries the sentence it was read from. 21 sources stand behind the page.

FieldValueCited text
Known as SHR4640 ClinicalTrials.gov intervention name — accepted as the source's own label NCT04620408
18

NCT04157959

NCT04586803

NCT05954169

NCT03211403

NCT04260373

NCT02890966

NCT07362355

NCT05513976

NCT04850638

NCT06196580

NCT04956432

NCT04052932

NCT04180982

NCT03185793

NCT04305392

NCT03015948

NCT02815839

NCT03131583

Known as Ruzinurad ChEMBL registry synonym — accepted as the source's own label CHEMBL3746329
Action Inhibit “a highly selective urate transporter 1 inhibitor” PMID 33693494 Nov 2021
1

“Solute carrier family 22 member 12 inhibitor” CHEMBL3746329

Modality Small molecule CHEMBL3746329
Route Oral oral administration” NCT02890966
Target SLC22A12 “Solute carrier family 22 member 12 inhibitor” CHEMBL3746329