Drugs / Tiragolumab
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Tiragolumab

also known as Tira · MTIG-7192A · RG-6058 · RO-7092284

Monoclonal antibody targets TIGIT via inhibition

Developed for
non-small cell lung carcinoma · cancer · colorectal cancer · high grade malignant neoplasm · melanoma · small cell lung carcinoma · esophageal squamous cell carcinoma · gastroesophageal junction adenocarcinoma
+38 more · head and neck cancer · head and neck squamous cell carcinoma · hepatocellular carcinoma · renal cell carcinoma · triple-negative breast carcinoma · urinary bladder cancer · urothelial carcinoma · anal canal squamous cell carcinoma · atypical teratoid rhabdoid tumor · breast cancer · cancer of unknown primary site · cervical cancer · cutaneous melanoma · digestive system carcinoma · endometrial cancer · epithelioid sarcoma · esophageal adenocarcinoma · esophageal cancer · follicular lymphoma · gastric cancer · gastroesophageal adenocarcinoma · gastroesophageal cancer · head and neck neoplasm · IDH-wildtype glioblastoma · kidney medullary carcinoma · liver cancer · lung cancer · metastatic malignant neoplasm · metastatic neoplasm · non-Hodgkin lymphoma · oral cavity squamous cell carcinoma · pancreatic adenocarcinoma · plasma cell myeloma · poorly differentiated chordoma · rectal cancer · refractory malignant neoplasm · squamous cell carcinoma · squamous cell lung carcinoma
Investigated by
Hoffmann-La Roche · Genentech, Inc. · M.D. Anderson Cancer Center · National Cancer Institute (NCI) · Alliance Foundation Trials, LLC. · Adagene Inc
+33 more · Alain Algazi · American Head and Neck Society · BioLineRx, Ltd. · Centre Georges Francois Leclerc · Chugai Pharmaceutical · Eli Lilly and Company · Foundation Medicine · Georgetown University · Gilead Sciences, Inc., GlaxoSmithKline plc, Seattle Genetics and Astellas · Grupo Espanol Multidisciplinario del Cancer Digestivo · Gustave Roussy, Cancer Campus, Grand Paris · Halozyme Therapeutics · Immune-Onc Therapeutics · Institut Curie · Institut für Klinische Krebsforschung IKF GmbH at Krankenhaus Nordwest · Liza Villaruz, MD · Mayo Clinic · National Taiwan University Hospital · NiKang Therapeutics, Inc. · Omico · Pfizer · Roche Global Development · Roche Pharma AG · SCRI Development Innovations, LLC · Strategic Alliance · Tempest Therapeutics · The George Institute for Global Health, Australia · The Netherlands Cancer Institute · Thoraxklinik-Heidelberg gGmbH · University Medical Center Groningen · University of Colorado, Denver · Washington University School of Medicine · Yonsei University

Trials 65 · started per year

today
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2017201820192020202120222023202420252026
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 16 trials
Phase 1 NCT06760481 Apr 2025 → Sep 2028 expected high grade malignant neoplasm M.D. Anderson Cancer Center Active not recruiting No outcome recorded
Phase 1 NCT05259319 Dec 2022 → Dec 2024 head and neck cancer, non-small cell lung carcinoma, renal cell carcinoma, urinary bladder cancer Centre Georges Francois Leclerc Unknown No outcome recorded
Phase 1 NCT04929223 Oct 2021 → Aug 2030 expected colorectal cancer Hoffmann-La Roche Recruiting No outcome recorded
Phase 1 NCT04584112 Sep 2020 → Mar 2023 triple-negative breast carcinoma Hoffmann-La Roche Completed No outcome recorded
Phase 1 NCT04045028 Jul 2019 → Mar 2023 non-Hodgkin lymphoma, plasma cell myeloma Genentech, Inc. Terminated No outcome recorded
Phase 1 NCT02794571 May 2016 → Nov 2024 metastatic neoplasm Genentech, Inc. Completed No outcome recorded
Phase 1/214 trials
Phase 1/2 NCT05908786 Dec 2023 → Aug 2025 hepatocellular carcinoma Hoffmann-La Roche Completed No outcome recorded
Phase 1/2 NCT05743504 Sep 2023 → May 2025 esophageal squamous cell carcinoma National Taiwan University Hospital Unknown No outcome recorded
Phase 1/2 NCT05459129 Apr 2023 → Aug 2024 head and neck squamous cell carcinoma Hoffmann-La Roche Completed No outcome recorded
Phase 1/2 NCT05394337 Feb 2023 → Dec 2028 expected metastatic malignant neoplasm M.D. Anderson Cancer Center Recruiting No outcome recorded
Phase 1/2 NCT05286801 Nov 2022 → Mar 2030 expected atypical teratoid rhabdoid tumor, epithelioid sarcoma, high grade malignant neoplasm, kidney medullary carcinoma +1 National Cancer Institute (NCI) Active not recruiting No outcome recorded
Phase 1/2 NCT05315713 May 2022 → Jul 2023 follicular lymphoma Hoffmann-La Roche Terminated No outcome recorded
Phase 1/2 NCT05251948 Mar 2022 → Sep 2025 gastroesophageal cancer Hoffmann-La Roche Terminated No outcome recorded
Phase 1/2 NCT05116202 Feb 2022 → Sep 2023 melanoma Hoffmann-La Roche Completed No outcome recorded
Phase 1/2 NCT04486352 Oct 2021 → Oct 2026 expected endometrial cancer Alliance Foundation Trials, LLC. Recruiting No outcome recorded
Phase 1/2 NCT04524871 Nov 2020 → Jul 2027 expected liver cancer Hoffmann-La Roche Recruiting No outcome recorded
Phase 235 trials
Phase 2 NCT06603818 Aug 2025 colorectal cancer National Cancer Institute (NCI) Withdrawn No outcome recorded
Phase 2 NCT07038915 Jul 2025 squamous cell lung carcinoma M.D. Anderson Cancer Center Withdrawn No outcome recorded
Phase 2 NCT06328036 Apr → Jul 2025 IDH-wildtype glioblastoma National Cancer Institute (NCI) Withdrawn No outcome recorded
Phase 2 NCT06754501 Apr 2025 → Jul 2027 expected cancer M.D. Anderson Cancer Center Active not recruiting No outcome recorded
Phase 2 NCT06784947 Mar → Sep 2025 overdue colorectal cancer University of Colorado, Denver Active not recruiting No outcome recorded
Phase 2 NCT06713798 Jan → Sep 2025 lung cancer Gustave Roussy, Cancer Campus, Grand Paris Withdrawn No outcome recorded
Phase 2 NCT06331598 Nov 2024 → Oct 2028 cancer Hoffmann-La Roche Withdrawn No outcome recorded
Phase 2 NCT06342037 Jun 2024 → Apr 2026 overdue breast cancer The Netherlands Cancer Institute Recruiting No outcome recorded
Phase 2 NCT06175390 Mar 2024 → Aug 2026 overdue triple-negative breast carcinoma Institut Curie Active not recruiting No outcome recorded
Phase 2 NCT06003621 Dec 2023 → May 2026 overdue cancer Omico Recruiting No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT04619797 Dec 2020 → Apr 2024 non-small cell lung carcinoma Hoffmann-La Roche Completed No outcome recorded
Phase 39 trials
Phase 3 NCT06267001 Mar 2024 → Dec 2025 non-small cell lung carcinoma Hoffmann-La Roche Terminated No outcome recorded
Phase 3 NCT05904886 Sep 2023 → May 2025 overdue hepatocellular carcinoma Hoffmann-La Roche Active not recruiting No outcome recorded
Phase 3 NCT05862285 Jun 2023 → Mar 2033 expected cancer Hoffmann-La Roche Recruiting No outcome recorded
Phase 3 NCT04665856 Dec 2020 → Aug 2023 overdue small cell lung carcinoma Hoffmann-La Roche Active not recruiting No outcome recorded
Phase 3 NCT04540211 Oct 2020 → Feb 2023 esophageal cancer Hoffmann-La Roche Completed No outcome recorded
Phase 3 NCT04543617 Sep 2020 → Mar 2027 expected esophageal squamous cell carcinoma Hoffmann-La Roche Active not recruiting No outcome recorded
Phase 3 NCT04513925 Aug 2020 → May 2025 non-small cell lung carcinoma Hoffmann-La Roche Completed No outcome recorded
Phase 3 NCT04294810 Mar 2020 → Dec 2025 non-small cell lung carcinoma Hoffmann-La Roche Completed No outcome recorded
Phase 3 NCT04256421 Feb 2020 → Sep 2022 small cell lung carcinoma Hoffmann-La Roche Completed No outcome recorded

Press releases naming this drug 3 releases

DateIssuerRelease
2021-12-10 Roche Global Development New data from the phase II CITYSCAPE trial show encouraging results with Roche’s novel anti-TIGIT tiragolumab plus Tecentriq roche.com
2021-01-05 Roche Global Development Roche’s novel anti-TIGIT tiragolumab granted FDA Breakthrough Therapy Designation in combination with Tecentriq for PD-L1-high non-small cell lung cancer roche.com
2020-05-14 Roche Global Development Roche to present first clinical data on novel anti-TIGIT cancer immunotherapy tiragolumab at ASCO roche.com

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 68 sources stand behind the page.

FieldValueCited text
Known as Tiragolumab “All patients receive atezolizumab (1200mg) plus tiragolumab (600 mg) for 2 cycles (Q3W) in concomitance with the 6 weeks of standard scheduled chemoradiotherapy” NCT05661188
64

“four cycles of 1200 mg of atezolizumab (Tecentriq®, Roche) and 600 mg of Tiragolumab (Roche) every 3 weeks” NCT06175390

NCT04294810

NCT04958811

NCT05009069

NCT05394337

NCT04929223

NCT04832854

NCT05459129

NCT06603818

NCT05060003

NCT06784947

NCT04300647

NCT05259319

NCT05116202

NCT05681039

NCT06331598

NCT05315713

NCT04933227

NCT04256421

NCT03784326

NCT03563716

NCT06760481

NCT04584112

NCT04543617

NCT05746481

NCT05908786

NCT06003621

NCT03337698

NCT05862285

NCT05286801

NCT05798663

NCT04665843

NCT05661578

NCT07038915

NCT05805501

NCT06342037

NCT03977467

NCT05743504

NCT04524871

NCT04665856

NCT03193190

NCT05483400

NCT03554083

NCT05034055

NCT06328036

NCT03869190

NCT04632992

NCT06754501

NCT04308785

NCT06713798

NCT06267001

NCT04540211

NCT03708224

NCT04513925

NCT05251948

NCT05645692

NCT05825625

NCT05904886

NCT04486352

NCT05715281

NCT03281369

NCT04045028

NCT02794571

NCT04619797

Known as MTIG-7192A ChEMBL registry synonym — accepted as the source's own label CHEMBL4298050
Known as RG-6058 ChEMBL registry synonym — accepted as the source's own label CHEMBL4298050
Known as RO-7092284 ChEMBL registry synonym — accepted as the source's own label CHEMBL4298050
Known as Tira “Participants will receive atezolizumab and Tiragolumab (Tira) until unacceptable toxicity or loss of clinical benefit, as determined by the investigator after an integrated...” NCT03869190
1

“This study evaluated the safety and efficacy of atezolizumab (Atezo) with or without tiragolumab (Tira) after nCRT in patients with LARC.” PMID 41529226 Jan 2026

Action Inhibit “that blocks the binding of TIGIT to CD155” PMID 38105505 Jan 2024
Modality Monoclonal antibody “Tiragolumab is a first-in-class, fully human IgG1/kappa anti-TIGIT monoclonal antibodyPMID 38105505 Jan 2024
Route Intravenous “Tiragolumab will be given via IV infusion” NCT02794571
Target TIGIT “Tiragolumab is a first-in-class, fully human IgG1/kappa anti-TIGIT monoclonal antibody that blocks the binding of TIGIT to CD155” PMID 38105505 Jan 2024