Drugs / Almonertinib
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Almonertinib

Small molecule targets EGFR via inhibition

Developed for
non-small cell lung carcinoma · lung cancer · metastatic malignant neoplasm in the brain · cancer · neoplastic meningitis · adenosquamous lung carcinoma · CDK4 linked melanoma · lung adenocarcinoma
+2 more · lung carcinoma · malignant leptomeningeal tumor
Investigated by
Jiangsu Hansoh Pharmaceutical Co., Ltd. · Sun Yat-sen University · Tianjin Medical University Cancer Institute and Hospital · Cancer Institute and Hospital, Chinese Academy of Medical Sciences · EQRx International, Inc. · First People's Hospital of Hangzhou
+38 more · Hansoh BioMedical R&D Company · Jiangsu HengRui Medicine Co., Ltd. · Second Affiliated Hospital of Nanchang University · Shanghai Chest Hospital · Shanghai Pulmonary Hospital, Shanghai, China · Suzhou Suncadia Biopharmaceuticals Co., Ltd. · The First Affiliated Hospital of Guangzhou Medical University · Baohui Han · Chia Tai Tianqing Pharmaceutical Group Nanjing Shunxin Pharmaceutical Co., Ltd. · China-Japan Friendship Hospital · Chinese Academy of Medical Sciences · Chongqing University Cancer Hospital · EQRx, Inc. · Fudan University · Fujian Cancer Hospital · GeneCast Biotechnology Co., Ltd. · Guangdong Association of Clinical Trials · Guangdong Provincial People's Hospital · Guangzhou Institute of Respiratory Disease · Hangzhou Cancer Hospital · Henan Cancer Hospital · Kunming Medical University · Laibin People's Hospital · Li-kun Chen · Nanfang Hospital, Southern Medical University · Peking Union Medical College Hospital · Peking University People's Hospital · Qianfoshan Hospital · Shanghai Cancer Hospital, China · Shanghai Zhongshan Hospital · Sichuan University · Taipei Medical University · Taipei Medical University Hospital · The First Affiliated Hospital of Xiamen University · The First Affiliated Hospital with Nanjing Medical University · West China Hospital · Yuan Chen · Zhejiang Cancer Hospital

Regulatory milestones approvals, filings & regulatory actions · 1 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved EU (EMA) Aumseqa 2026-02-12 europa.eu

Trials 62 · started per year

today
EU approved 2026
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9
17
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2018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 19 trials
Phase 1 NCT07645222 Jun 2026 → Oct 2028 expected lung cancer Hansoh BioMedical R&D Company Recruiting No outcome recorded
Phase 1 NCT06926413 Feb → Oct 2025 overdue non-small cell lung carcinoma Jiangsu Hansoh Pharmaceutical Co., Ltd. Recruiting No outcome recorded
Phase 1 NCT07130916 Dec 2024 → Aug 2025 overdue non-small cell lung carcinoma Jiangsu Hansoh Pharmaceutical Co., Ltd. Recruiting No outcome recorded
Phase 1 NCT06585059 Sep 2024 → Dec 2025 overdue non-small cell lung carcinoma Chia Tai Tianqing Pharmaceutical Group Nanjing Shunxin Pharmaceutical Co., Ltd. Not yet recruiting No outcome recorded
Phase 1 NCT05199610 Mar 2022 → Apr 2023 EQRx International, Inc. Completed No outcome recorded
Phase 1 NCT05430386 Jan 2022 → Dec 2023 non-small cell lung carcinoma Jiangsu Hansoh Pharmaceutical Co., Ltd. Unknown No outcome recorded
Phase 1 NCT05826483 Jan 2022 → Dec 2024 lung cancer Guangzhou Institute of Respiratory Disease Unknown No outcome recorded
Phase 1 NCT05048134 Oct 2021 → Feb 2023 cancer Jiangsu HengRui Medicine Co., Ltd. Terminated No outcome recorded
Phase 1 NCT04969965 Jun → Oct 2021 non-small cell lung carcinoma EQRx, Inc. Completed No outcome recorded
Phase 1/24 trials
Phase 1/2 NCT06947811 Jun 2025 → Mar 2027 expected CDK4 linked melanoma Sun Yat-sen University Recruiting No outcome recorded
Phase 1/2 NCT06092268 Oct 2023 → Dec 2025 cancer Suzhou Suncadia Biopharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 1/2 NCT05503888 Oct 2022 → Jul 2027 expected non-small cell lung carcinoma Suzhou Suncadia Biopharmaceuticals Co., Ltd. Not yet recruiting No outcome recorded
Phase 1/2 NCT02981108 May 2017 → Jan 2019 non-small cell lung carcinoma Jiangsu Hansoh Pharmaceutical Co., Ltd. Unknown No outcome recorded
Phase 231 trials
Phase 2 NCT07624487 Jun 2026 → Dec 2028 expected lung adenocarcinoma Taipei Medical University Hospital Recruiting No outcome recorded
Phase 2 NCT07637448 May 2026 → Mar 2029 expected non-small cell lung carcinoma Nanfang Hospital, Southern Medical University Recruiting No outcome recorded
Phase 2 NCT06951464 Jun 2025 → May 2027 expected non-small cell lung carcinoma Sichuan University Recruiting No outcome recorded
Phase 2 NCT06924398 Apr → Dec 2025 overdue non-small cell lung carcinoma Sun Yat-sen University Recruiting No outcome recorded
Phase 2 NCT06752408 Dec 2024 → Jan 2027 expected non-small cell lung carcinoma Peking Union Medical College Hospital Not yet recruiting No outcome recorded
Phase 2 NCT06227897 Jun 2024 → Apr 2026 lung cancer Sun Yat-sen University Withdrawn No outcome recorded
Phase 2 NCT06463171 Jun 2024 → Jun 2026 non-small cell lung carcinoma Shanghai Pulmonary Hospital, Shanghai, China Unknown No outcome recorded
Phase 2 NCT06300424 Apr 2024 → Jan 2026 overdue non-small cell lung carcinoma Guangdong Provincial People's Hospital Active not recruiting No outcome recorded
Phase 2 NCT06185400 Feb 2024 → Jul 2025 overdue non-small cell lung carcinoma Cancer Institute and Hospital, Chinese Academy of Medical Sciences Not yet recruiting No outcome recorded
Phase 2 NCT05946460 Aug 2023 → Jul 2025 lung cancer The First Affiliated Hospital of Guangzhou Medical University Unknown No outcome recorded
Phase 2/32 trials
Phase 2/3 NCT06417008 May 2024 → Jun 2026 overdue non-small cell lung carcinoma Hansoh BioMedical R&D Company Recruiting No outcome recorded
Phase 2/3 NCT05994339 Sep 2023 → Aug 2025 lung carcinoma Laibin People's Hospital Unknown No outcome recorded
Phase 312 trials
Phase 3 NCT06110663 Dec 2023 → Dec 2024 non-small cell lung carcinoma Jiangsu Hansoh Pharmaceutical Co., Ltd. Unknown No outcome recorded
Phase 3 NCT06043973 Sep 2023 → Sep 2026 expected non-small cell lung carcinoma Qianfoshan Hospital Recruiting No outcome recorded
Phase 3 NCT05800223 Jan 2023 → Dec 2027 expected non-small cell lung carcinoma Shanghai Cancer Hospital, China Recruiting No outcome recorded
Phase 3 NCT05493501 Dec 2022 → Aug 2023 non-small cell lung carcinoma EQRx International, Inc. Terminated No outcome recorded
Phase 3 NCT04841811 Jun 2022 → Dec 2026 expected lung cancer Guangdong Association of Clinical Trials Active not recruiting No outcome recorded
Phase 3 NCT04923906 Aug 2021 → Jun 2024 overdue non-small cell lung carcinoma Jiangsu Hansoh Pharmaceutical Co., Ltd. Active not recruiting No outcome recorded
Phase 3 NCT04762459 Aug 2021 → May 2026 overdue non-small cell lung carcinoma Chinese Academy of Medical Sciences Enrolling by invitation No outcome recorded
Phase 3 NCT04951648 Jul 2021 → Oct 2023 non-small cell lung carcinoma Jiangsu Hansoh Pharmaceutical Co., Ltd. Unknown No outcome recorded
Phase 3 NCT04870190 Jun 2021 → Jun 2024 non-small cell lung carcinoma Shanghai Chest Hospital Unknown No outcome recorded
Phase 3 NCT04687241 Apr 2021 → Jul 2024 overdue non-small cell lung carcinoma Jiangsu Hansoh Pharmaceutical Co., Ltd. Active not recruiting No outcome recorded
Phase not applicable4 trials
NCT07398599 Feb 2026 → Dec 2027 expected malignant leptomeningeal tumor, non-small cell lung carcinoma Second Affiliated Hospital of Nanchang University Recruiting No outcome recorded
NCT06102928 Oct 2023 → Oct 2026 expected non-small cell lung carcinoma Kunming Medical University Recruiting No outcome recorded
NCT04944069 Jul 2021 → Mar 2024 neoplastic meningitis, non-small cell lung carcinoma Second Affiliated Hospital of Nanchang University Unknown No outcome recorded
NCT04778800 Mar 2021 → Feb 2023 metastatic malignant neoplasm in the brain, neoplastic meningitis, non-small cell lung carcinoma Henan Cancer Hospital Unknown No outcome recorded
Also used as a comparator or background therapy in 10 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT05223595 Background Apr 2021 → Sep 2023 non-small cell lung carcinoma Changchun GeneScience Pharmaceutical Co., Ltd. Unknown No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT06474455 Background Jul 2024 → Jun 2029 expected cancer Shanghai Hengrui Pharmaceutical Co., Ltd. Recruiting No outcome recorded
Phase 23 trials
Phase 2 NCT06452433 Background Jun 2024 → Dec 2027 expected non-small cell lung carcinoma Cancer Institute and Hospital, Chinese Academy of Medical Sciences Not yet recruiting No outcome recorded
Phase 2 NCT04755738 Background Jan 2022 → Mar 2023 non-small cell lung carcinoma Qianfoshan Hospital Unknown No outcome recorded
Phase 2 NCT04519983 Background Jan 2022 → Dec 2023 lung carcinoma Shanghai Cancer Hospital, China Unknown No outcome recorded
Phase 34 trials
Phase 3 NCT07183189 Comparator Oct 2025 → Nov 2032 expected non-small cell lung carcinoma Suzhou Suncadia Biopharmaceuticals Co., Ltd. Recruiting No outcome recorded
Phase 3 NCT05768490 Background Mar 2023 → Dec 2028 expected metastatic malignant neoplasm in the brain Sun Yat-sen University Recruiting No outcome recorded
Phase 3 NCT04500717 Comparator Oct 2020 → Oct 2022 non-small cell lung carcinoma Cancer Institute and Hospital, Chinese Academy of Medical Sciences Unknown No outcome recorded
Phase 3 NCT04500704 Comparator Oct 2020 → Dec 2021 non-small cell lung carcinoma Cancer Institute and Hospital, Chinese Academy of Medical Sciences Unknown No outcome recorded
Phase 41 trial
Phase 4 NCT04401059 Comparator Nov 2020 → Sep 2025 adenocarcinoma, non-small cell lung carcinoma Tian Xie Unknown No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 74 sources stand behind the page.

FieldValueCited text
Known as almonertinib Almonertinib (HS-10296) is a novel, third-generation EGFR tyrosine kinase inhibitor (EGFR TKI) that targets both EGFR-sensitizing and T790M resistance mutations.” PMID 32916310 Sep 2020
52

“Aumolertinib (formerly almonertinib; HS-10296) is a novel third-generation epidermal growth factor receptor tyrosine kinase inhibitor approved in China.” PMID 35580297 May 2022

“Gentuximab: 8mg/kg or 12mg/kg intravenous (IV) infusion administered on Day 1 and 15 of each cycle; Almonertinib: 110 mg orally once daily.” NCT05223595

“Gefitinib(Iressa,YiRuiKe), Erlotinib(Tarceva), Icotinib(Kaimeina), Osimertinib(Tagrisso), Almonertinib, Furmonertinib, etc.” NCT04401059

“Dose escalation: HS-10241 and Almonertinib will be administered in combination.” NCT05430386

“Intervention: Oral almonertinib (110 mg/day) for three months” NCT06924398

“2. Almonertinib: 110mg, orally once a day” NCT04978753

almonertinib 220mg once daily” NCT07398599

NCT06110663

NCT04951635

NCT06951464

NCT04951648

NCT04808752

NCT04785742

NCT05662813

NCT04643847

NCT04755738

NCT04500704

NCT04952168

NCT04905550

NCT04500717

NCT04354961

NCT06043973

NCT06947811

NCT06185400

NCT04762459

NCT04553887

NCT04778800

NCT06463171

NCT06474455

NCT04423185

NCT04636593

NCT05048134

NCT04646824

NCT06300424

NCT05800223

NCT04944069

NCT04870190

NCT04687241

NCT04882345

NCT04785729

NCT04592666

NCT05994339

NCT06452433

NCT05768490

NCT04841811

NCT05503888

NCT04685070

NCT04455594

NCT05534113

NCT05826483

NCT06585059

NCT06092268

Known as Almonertinib Mesilate Almonertinib Mesilate Tablets.” NCT06474455
Known as aumolertinib Aumolertinib (formerly almonertinib; HS-10296) is a novel third-generation epidermal growth factor receptor tyrosine kinase inhibitor approved in China.” PMID 35580297 May 2022
19

“All patients receive first-line oral therapy with standard-dose third-generation EGFR-TKIs (osimertinib, aumolertinib, or furmonertinib).” NCT07637448

“INTERVENTIONS: Patients received aumolertinib, 165 mg, orally once daily until disease progression or unacceptable toxic effects.” PMID 40569623 Aug 2025

NCT04519983

NCT05493501

NCT05778149

NCT07130916

NCT06102928

NCT06227897

NCT05946460

NCT06417008

NCT04923906

NCT07645222

NCT05199610

NCT06752408

NCT07624487

NCT04922138

NCT07183189

NCT06926413

NCT04969965

Known as aumolertinib mesylate Aumolertinib mesylate tablets are administered 110 mg orally once a day” NCT06102928
Known as HS-10296 “This is a phase II, single-arm, open-label study to evaluate the efficacy and safety of the third generation tyrosine kinase inhibitors (TKIs) Almonertinib (HS-10296) as...” NCT04685070
3

“Almonertinib (HS-10296) is a novel, third-generation EGFR tyrosine kinase inhibitor (EGFR TKI) that targets both EGFR-sensitizing and T790M resistance mutations.” PMID 32916310 Sep 2020

“Aumolertinib (formerly almonertinib; HS-10296) is a novel third-generation epidermal growth factor receptor tyrosine kinase inhibitor approved in China.” PMID 35580297 May 2022

NCT03904823

Action Inhibit “tyrosine kinase inhibitor (EGFR TKI)” PMID 32916310 Sep 2020
Modality Small molecule “novel, third-generation EGFR tyrosine kinase inhibitor (EGFR TKI)” PMID 32916310 Sep 2020
Route Oral “Eligible patients were enrolled and randomly assigned in a 1:1 ratio to orally receive either aumolertinib or gefitinib in a double-blinded fashion.” PMID 39016053 Jul 2024
Target EGFR “targets both EGFR-sensitizing and T790M resistance mutations” PMID 32916310 Sep 2020