Drugs / VS-7375
last change Jul 2026 re-read 2 minutes ago

VS-7375

Small molecule targets KRAS via inhibition

Developed for
colorectal cancer · non-small cell lung carcinoma · pancreatic ductal adenocarcinoma
Investigated by
Verastem, Inc.

Trials 4 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 1/21 trial
Phase 1/2 NCT07020221 Jun 2025 → Dec 2028 expected colorectal cancer, non-small cell lung carcinoma, pancreatic ductal adenocarcinoma Verastem, Inc. Recruiting No outcome recorded
Phase 23 trials
Phase 2 NCT07659795 Jul 2026 → Jun 2027 expected colorectal cancer Verastem, Inc. Recruiting No outcome recorded
Phase 2 NCT07644559 Jun 2026 → Jun 2027 expected pancreatic ductal adenocarcinoma Verastem, Inc. Recruiting No outcome recorded
Phase 2 NCT07659782 Jun 2026 → Jun 2027 expected non-small cell lung carcinoma Verastem, Inc. Not yet recruiting No outcome recorded

Evidence & citations 5 cited values

Every value below carries the sentence it was read from. 4 sources stand behind the page.

FieldValueCited text
Known as VS-7375 ClinicalTrials.gov intervention name — accepted as the source's own label NCT07644559
3

NCT07659782

NCT07020221

NCT07659795

Action Inhibit “VS-7375 is a highly selective oral, non-covalent, small molecule KRAS G12D (ON/OFF) inhibitor.” NCT07020221
Modality Small molecule “VS-7375 is a highly selective oral, non-covalent, small molecule KRAS G12D (ON/OFF) inhibitor.” NCT07020221
Route Oral “VS-7375 is a highly selective oral, non-covalent, small molecule KRAS G12D (ON/OFF) inhibitor.” NCT07020221
Target KRAS “VS-7375 is a highly selective oral, non-covalent, small molecule KRAS G12D (ON/OFF) inhibitor.” NCT07020221