Drugs / Rifapentine
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Rifapentine

Small molecule

Developed for
tuberculosis · latent tuberculosis infection · pulmonary tuberculosis · female genital tuberculosis · lymph node tuberculosis · Mycobacterium avium complex disease · respiratory tract infectious disorder · silicotuberculosis
+1 more · tuberculosis, spinal
Investigated by
Centers for Disease Control and Prevention · Johns Hopkins University · National Institute of Allergy and Infectious Diseases (NIAID) · Huashan Hospital · Sanofi · US Department of Veterans Affairs
+111 more · The Aurum Institute NPC · University of Cape Town · Advancing Clinical Therapeutics Globally for HIV/AIDS and Other Infections · McGill University Health Centre/Research Institute of the McGill University Health Centre · Merck Sharp & Dohme LLC · National Institutes of Health Clinical Center (CC) · National Taiwan University Hospital · University of Stellenbosch · ViiV Healthcare · Yale University · APIN Public Health Initiatives · Aarhus University Hospital · Affiliated Wenling Hospital of Wenzhou Medical University · All India Institute of Medical Sciences · All India Institute of Medical Sciences, Bhubaneswar · Anderson Clinical Research · Aurum Institute · Beijing Ditan Hospital · Beijing YouAn Hospital · Bellvitge Biomedical Research Institute · Bhumibol Adulyadej Hospital · Brigham and Women's Hospital · Buddhachinnaraj Hospital · Canadian Institutes of Health Research (CIHR) · Centers for Disease Control, Taiwan · Centre for the AIDS Programme of Research in South Africa · Chang Gung Memorial Hospital · Chengdu Public Health Clinical Center · Chest Hospital of Guangxi Zhuang Autonomous Region · Chiangrai Prachanukroh Hospital · Chongqing Public Health Medical Center · Chris Hani Baragwanath Academic Hospital · Dr. Nyanda Elias Ntinginya · Elizabeth Glaser Pediatric AIDS Foundation · Eunice Kennedy Shriver National Institute of Child Health and Human Development (NICHD) · Faculty of Medicine Universitas Padjadjaran · Federal University of Rio de Janeiro · First Affiliated Hospital of Zhejiang University · Fred Hutchinson Cancer Center · Freundeskreis Für Internationale Tuberkulosehilfe e.V · Gilead Sciences · Global Alliance for TB Drug Development · Government Vellore Medical College, Vellore · Government of Canada · Government of Nunavut · Guangzhou eighth People's Hospital ,Guangzhou Medilcal University · Guiyang Public Health Clinical Center · HatYai Hospital · Hoechst Marion Roussel · Institute of Child Health, Chennai · Instituto de Salud Carlos III · Kaohsiung Veterans General Hospital. · Kilimanjaro Christian Medical University College (KCMUCo), Tanzania · King Chulalongkorn Memorial Hospital · King's College London · Klang Hospital · London School of Hygiene and Tropical Medicine · Madurai Medical College · Maharat Nakhon Ratchasima Hospital · Makerere University · Meng Chao Hepatobiliary Hospital of Fujian Medical University · Miguel Santin · National Institute of Mental Health (NIMH) · National Institute of Tuberculosis and Respiratory Diseases, New Delhi · National Institute on Drug Abuse (NIDA) · National Taiwan University · National University Hospital, Singapore · Otago University, New Zealand · Ottawa Hospital Research Institute · Peking Union Medical College Hospital · Police General Hospital · Pontificia Universidad Catolica de Chile · Pranangklao Hospital · Queen Sawang Vadhana Memorial Hospital · all 117 on the full record

Regulatory milestones approvals, filings & regulatory actions · 4 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansions (3) US (FDA) PRIFTIN 2000-10-20 – 2014-11-25 fda.gov
Approved US (FDA) PRIFTIN 1998-06-22 fda.gov

Trials 63 · started per year

today
US approved 1998
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1995199619971998199920002001200220032004200520062007200820092010201120122013201420152016201720182019202020212022202320242025202620272028
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 111 trials
Phase 1 NCT07069582 Apr → Oct 2026 expected tuberculosis McGill University Health Centre/Research Institute of the McGill University Health Centre Not yet recruiting No outcome recorded
Phase 1 NCT06281834 Nov 2024 → Feb 2027 expected latent tuberculosis infection Brigham and Women's Hospital Recruiting No outcome recorded
Phase 1 NCT03886701 Apr → May 2019 HIV infectious disease, isoniazid toxicity, latent tuberculosis infection Walter K. Kraft Completed No outcome recorded
Phase 1 NCT03510468 Jun 2018 → Nov 2022 National Institutes of Health Clinical Center (CC) Completed No outcome recorded
Phase 1 NCT02771249 Jun 2016 → Aug 2021 latent tuberculosis infection National Institutes of Health Clinical Center (CC) Completed No outcome recorded
Phase 1 NCT01690403 Dec 2012 → Mar 2014 tuberculosis Sanofi Completed No outcome recorded
Phase 1 NCT01574638 Jun 2012 → Jun 2013 tuberculosis National Institute of Allergy and Infectious Diseases (NIAID) Completed No outcome recorded
Phase 1 NCT01162486 Apr 2010 → Feb 2011 pulmonary tuberculosis Johns Hopkins University Completed No outcome recorded
Phase 1 NCT02216331 Mar → May 2010 tuberculosis Global Alliance for TB Drug Development Completed No outcome recorded
Phase 1 NCT00809718 Feb 2009 → May 2011 The University of Texas Health Science Center at San Antonio Completed No outcome recorded
Phase 1/26 trials
Phase 1/2 NCT07124559 Jul 2026 → Jan 2028 expected tuberculosis National Institute of Allergy and Infectious Diseases (NIAID) Not yet recruiting No outcome recorded
Phase 1/2 NCT05122026 Jan 2024 → Oct 2025 overdue pregnancy disorder, tuberculosis The Aurum Institute NPC Active not recruiting No outcome recorded
Phase 1/2 NCT05122767 May 2023 → Jul 2025 overdue HIV infectious disease, tuberculosis The Aurum Institute NPC Active not recruiting No outcome recorded
Phase 1/2 NCT03730181 Oct 2019 → Dec 2024 latent tuberculosis infection Centers for Disease Control and Prevention Completed No outcome recorded
Phase 1/2 NCT03435146 Jan 2018 → Dec 2022 HIV infectious disease, respiratory tract infectious disorder The Aurum Institute NPC Completed No outcome recorded
Phase 1/2 NCT02651259 Mar 2017 → Apr 2019 tuberculosis National Institute of Allergy and Infectious Diseases (NIAID) Completed No outcome recorded
Phase 29 trials
Phase 2 NCT07595042 Jul 2026 → Jun 2029 expected tuberculosis National Institute of Allergy and Infectious Diseases (NIAID) Not yet recruiting No outcome recorded
Phase 2 NCT06917495 Apr 2025 → Dec 2027 expected tuberculosis, spinal Shandong University Not yet recruiting No outcome recorded
Phase 2 NCT04311502 Nov 2021 → Jun 2024 HIV infectious disease, tuberculosis National Institute of Allergy and Infectious Diseases (NIAID) Terminated No outcome recorded
Phase 2 NCT04272242 Feb → Dec 2021 HIV infectious disease, latent tuberculosis infection National Institute of Allergy and Infectious Diseases (NIAID) Terminated No outcome recorded
Phase 2 NCT00814671 Apr 2010 → Jun 2013 tuberculosis Johns Hopkins University Completed No outcome recorded
Phase 2 NCT00728507 Nov 2009 → Apr 2013 tuberculosis Johns Hopkins University Terminated No outcome recorded
Phase 2 NCT00694629 Dec 2008 → Jun 2013 pulmonary tuberculosis Centers for Disease Control and Prevention Completed No outcome recorded
Phase 2 NCT00023426 Jul 1999 → Feb 2003 tuberculosis Centers for Disease Control and Prevention Completed No outcome recorded
Phase 2 NCT00002192 HIV infectious disease, Mycobacterium avium complex disease Anderson Clinical Research Completed No outcome recorded
Phase 2/35 trials
Phase 2/3 NCT06568484 May 2026 → Jul 2027 expected latent tuberculosis infection Johns Hopkins University Recruiting No outcome recorded
Phase 2/3 NCT06498414 Jun 2025 → Apr 2027 expected latent tuberculosis infection McGill University Health Centre/Research Institute of the McGill University Health Centre Recruiting No outcome recorded
Phase 2/3 NCT03474029 Aug 2019 → Dec 2029 expected latent tuberculosis infection Centers for Disease Control and Prevention Recruiting No outcome recorded
Phase 2/3 NCT03474198 Mar 2018 → Jan 2022 pulmonary tuberculosis University College, London Completed No outcome recorded
Phase 2/3 NCT02735590 Sep 2016 → Dec 2019 tuberculosis University of Cape Town Unknown No outcome recorded
Phase 318 trials
Phase 3 NCT06191692 Aug 2025 → Dec 2026 expected latent tuberculosis infection Freundeskreis Für Internationale Tuberkulosehilfe e.V Not yet recruiting No outcome recorded
Phase 3 NCT06253715 Jan 2025 → Sep 2027 expected lymph node tuberculosis, pulmonary tuberculosis Johns Hopkins University Recruiting No outcome recorded
Phase 3 NCT05330884 Jul 2024 → Jun 2027 tuberculosis Tuberculosis Research Centre, India Suspended No outcome recorded
Phase 3 NCT06022146 Sep 2023 → Sep 2026 expected latent tuberculosis infection Huashan Hospital Recruiting No outcome recorded
Phase 3 NCT05454345 Oct 2022 → Jun 2025 pulmonary tuberculosis First Affiliated Hospital of Zhejiang University Unknown No outcome recorded
Phase 3 NCT04600167 Jun 2022 → Dec 2025 diabetes mellitus, tuberculosis Dr. Nyanda Elias Ntinginya Unknown No outcome recorded
Phase 3 NCT04528277 Sep 2020 → Sep 2021 female genital tuberculosis, female infertility, latent tuberculosis infection Huashan Hospital Unknown No outcome recorded
Phase 3 NCT04856644 Jan 2020 → Dec 2023 overdue pulmonary tuberculosis Kaohsiung Veterans General Hospital. Active not recruiting No outcome recorded
Phase 3 NCT04094012 Sep 2019 → Oct 2023 latent tuberculosis infection National Taiwan University Hospital Completed No outcome recorded
Phase 3 NCT03785106 Aug 2019 → Mar 2038 expected The HIV Netherlands Australia Thailand Research Collaboration Active not recruiting No outcome recorded
Phase 48 trials
Phase 4 NCT06153069 Nov 2025 → Nov 2027 expected tuberculosis Huashan Hospital Recruiting No outcome recorded
Phase 4 NCT05021731 Apr 2024 → Apr 2025 kidney failure, latent tuberculosis infection Miguel Santin Unknown No outcome recorded
Phase 4 NCT05118490 Jul 2023 → Jul 2025 overdue AIDS-related disorder, tuberculosis The Aurum Institute NPC Active not recruiting No outcome recorded
Phase 4 NCT05411744 Jul 2022 → Jan 2026 overdue end stage renal failure, latent tuberculosis infection Rutgers, The State University of New Jersey Active not recruiting No outcome recorded
Phase 4 NCT04703075 Mar 2022 → Jun 2024 tuberculosis Johns Hopkins University Completed No outcome recorded
Phase 4 NCT04551573 May → Oct 2021 HIV infectious disease, tuberculosis Yale University Withdrawn No outcome recorded
Phase 4 NCT03266991 Oct 2017 → Feb 2023 Aarhus University Hospital Terminated No outcome recorded
Phase 4 NCT02689089 Nov 2016 → Aug 2019 tuberculosis Ottawa Hospital Research Institute Completed No outcome recorded
Phase not applicable6 trials
NCT07608172 May 2026 → Jun 2028 expected pulmonary tuberculosis Shanghai Public Health Clinical Center Not yet recruiting No outcome recorded
NCT07086820 Oct 2025 → May 2028 expected latent tuberculosis infection Pontificia Universidad Catolica de Chile Recruiting No outcome recorded
NCT03900858 Dec 2018 → Jan 2022 silicotuberculosis Huashan Hospital Unknown No outcome recorded
NCT03089983 Aug 2017 → Apr 2024 HIV infectious disease, hepatitis, opiate dependence, tuberculosis Yale University Completed No outcome recorded
NCT00164450 Sep 2005 → Aug 2008 tuberculosis Centers for Disease Control and Prevention Completed No outcome recorded
NCT00023387 Mar 2000 → May 2001 tuberculosis Centers for Disease Control and Prevention Completed No outcome recorded
Also used as a comparator or background therapy in 5 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT02099240 Comparator Mar 2014 → Nov 2018 osteomyelitis University of Louisville Terminated No outcome recorded
Phase 21 trial
Phase 2 NCT05630872 Background Feb 2024 → May 2025 tuberculosis National Institute of Allergy and Infectious Diseases (NIAID) Completed No outcome recorded
Phase 32 trials
Phase 3 NCT02980016 Comparator Nov 2016 → Oct 2019 HIV infectious disease, tuberculosis The Aurum Institute NPC Completed No outcome recorded
Phase 3 NCT00057122 Comparator Sep 2002 → Nov 2008 HIV infectious disease, tuberculosis National Institute of Allergy and Infectious Diseases (NIAID) Completed No outcome recorded
Phase 41 trial
Phase 4 NCT06874725 Comparator Apr 2018 → Apr 2024 overdue latent tuberculosis infection Taichung Veterans General Hospital Active not recruiting No outcome recorded

Evidence & citations 16 cited values

Every value below carries the sentence it was read from. 69 sources stand behind the page.

FieldValueCited text
Known as Rifapentine “A recent multi-centered, multi-national randomized control non inferiority trial with approximately 4,000 patients per arm demonstrated that Rifapentine and INH (3HP) given...” NCT02689089
67

“Once-weekly isoniazid and rifapentine for 3 months is a treatment option in persons with human immunodeficiency virus and latent tuberculosis infection.” PMID 29415190 Jul 2018

“8 weeks of daily isoniazid, rifapentine, moxifloxacin and pyrazinamide, followed by 9 weeks of daily isoniazid, rifapentine and moxifloxacin.” NCT07608172

“Oral chemoprophylaxis will be standard of care - either 6 months of Isoniazid or 3 months of weekly Isoniazid and RifapentineNCT05330884

“weekly oral Rifapentine 15 mg/kg (up to 900mg) plus Isoniazid 15 mg/kg (up to 900mg) for 12 doses” NCT02430259

“daily rifapentine (R) and moxifloxacin (M) plus isoniazid (H) and pyrazinamide (P)” NCT05630872

“high-dose rifapentine (P), isoniazid (H), pyrazinamide (Z), and moxifloxacin (M)” NCT06153069

Rifapentine (RPT) 900 mg once-weekly x 12 doses (3 months)” NCT00023452

“once-weekly rifapentine (RPT) and isoniazid (INH) (3HP)” NCT05122767

RifapentineNCT02099240

NCT03730181

NCT05411744

NCT02735590

NCT04272242

NCT02208427

NCT03089983

NCT06281834

NCT00694629

NCT00057122

NCT06874725

NCT05122026

NCT02410772

NCT03266991

NCT04551573

NCT07086820

NCT07595042

NCT03510468

NCT00460759

NCT03474198

NCT03785106

NCT03886701

NCT05118490

NCT06917495

NCT03474029

NCT00023426

NCT00002192

NCT07069582

NCT00023387

NCT06022146

NCT00023335

NCT04856644

NCT00814671

NCT06253715

NCT04094012

NCT06191692

NCT06568484

NCT01582711

NCT05454345

NCT04703075

NCT01574638

NCT00164450

NCT01690403

NCT06498414

NCT04600167

NCT01404312

NCT03435146

NCT00728507

NCT04528277

NCT02651259

NCT04311502

NCT05021731

NCT02980016

NCT07124559

NCT00809718

NCT02563327

NCT01162486

NCT02216331

NCT03900858

Known as ANTIBIOTIC DL-473IT ChEMBL registry synonym — accepted as the source's own label CHEMBL1660
Known as DL-473 ChEMBL registry synonym — accepted as the source's own label CHEMBL1660
Known as KTC-1 ChEMBL registry synonym — accepted as the source's own label CHEMBL1660
Known as M000473 “rifapentine (M000473)” NCT01690403
Known as MDL 473 ChEMBL registry synonym — accepted as the source's own label CHEMBL1660
Known as Prifitin ChEMBL registry synonym — accepted as the source's own label CHEMBL1660
Known as Priftin ChEMBL registry synonym — accepted as the source's own label CHEMBL1660
Known as Priftin - Rifapentine Priftin - RifapentineNCT00809718
1

“Priftin (rifapentine)” NCT02980016

Known as R-77-3 ChEMBL registry synonym — accepted as the source's own label CHEMBL1660
Known as Rifapentin ChEMBL registry synonym — accepted as the source's own label CHEMBL1660
Known as Rifapentina ChEMBL registry synonym — accepted as the source's own label CHEMBL1660
Known as Rifapentine RPT Rifapentine RPTNCT03900858
Known as RPT “The investigators hypothesize that short-course (4-week) daily isoniazid/rifapentine (INH/RPT) (1HP) is not inferior to standard -course (12 weeks) INH/RPT weekly regimen (3HP)...” NCT03785106
11

“600 mg of Rifapentine (RPT) given once daily (o.d., omni die) for 6 weeks (6wP).” NCT03474029

“steady-state dolutegravir (DTG) and rifapentine (RPT) concentrations” NCT06281834

“escalating doses of rifapentine (RPT) administered daily by oral” NCT01162486

“once-weekly rifapentine (RPT) and isoniazid (INH) (3HP)” NCT05122767

“rifapentine (RPT, 900 mg)” NCT04600167

“Drug: Rifapentine (RPT)” NCT06917495

“Rifapentine (RPT)” NCT04272242

“Rifapentine (RPT)” NCT01574638

“Rifapentine (RPT)” NCT02651259

“Rifapentine (RPT)” NCT03886701

“Rifapentine (RPT)” NCT01404312

Modality Small molecule CHEMBL1660
Route Oral “Rifapentine plus Isoniazid taken orally, weekly, by direct observation for 12 weeks” NCT00164450