Drugs / Trimetazidine
last change Jul 2026 re-read 2 minutes ago

Trimetazidine

Small molecule

Developed for
coronary artery disorder · hepatocellular carcinoma · pulmonary arterial hypertension · type 2 diabetes mellitus · acute kidney injury · acute respiratory distress syndrome · amyotrophic lateral sclerosis · cardiomyopathy
+16 more · cardiovascular disorder · coronary microvascular disorder · COVID-19 · diabetes mellitus · diabetic kidney disease · diastolic heart failure · intermediate coronary syndrome · metabolic dysfunction-associated steatotic liver disease · paroxysmal atrial fibrillation · platelet disorder, undefined · poisoning · chemotherapy-induced neuropathy · heart failure · hypertrophic cardiomyopathy · ischemic stroke · wild type ATTR amyloidosis
Investigated by
Anyang Tumor Hospital · First Affiliated Hospital of Xinjiang Medical University · First People's Hospital of Shangqiu · Luoyang Central Hospital · Nanyang Central Hospital · The First Affiliated Hospital of Zhengzhou University
+31 more · Third People's Hospital of Jiaozuo · Ain Shams University · Beni-Suef University · Cairo University · China National Center for Cardiovascular Diseases · Chinese PLA General Hospital · Clinical Hospital Center Zemun · FightMND · Fondo Nacional de Desarrollo Científico y Tecnológico, Chile · IRCCS San Raffaele · InCor Heart Institute · Indonesia University · Julius Clinical · King's College London · Martin Pharmaceuticals · Ministry of Health, Brazil · National Research Center for Preventive Medicine · October 6 University · Peking University Third Hospital · Pingmei Shenma Medical Group General Hospital · Pontificia Universidad Catolica de Chile · Shanghai 10th People's Hospital · Shenma Medical Group General Hospital · Shiyan City Renmin Hospital · Sun Yat-sen University · The University of Queensland · The University of The West Indies · Tongji Hospital · UMC Utrecht · University of Sao Paulo General Hospital · Yonsei University

Trials 23 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT03737448 Nov 2018 → Jun 2021 liver disorder Martin Pharmaceuticals Suspended No outcome recorded
Phase 27 trials
Phase 2 NCT06140953 Dec 2023 → Jun 2024 metabolic dysfunction-associated steatotic liver disease October 6 University Completed No outcome recorded
Phase 2 NCT05556005 Sep 2022 → Sep 2023 cardiomyopathy, type 2 diabetes mellitus Ain Shams University Unknown No outcome recorded
Phase 2 NCT05147194 Jan 2022 → Dec 2023 diabetic kidney disease Tongji Hospital Unknown No outcome recorded
Phase 2 NCT04788745 Jun 2021 → May 2023 amyotrophic lateral sclerosis The University of Queensland Completed No outcome recorded
Phase 2 NCT04760821 Dec 2020 → Apr 2021 COVID-19, acute respiratory distress syndrome Ministry of Health, Brazil Unknown No outcome recorded
Phase 2 NCT03603249 Jul 2018 → Apr 2019 platelet disorder, undefined The University of The West Indies Completed No outcome recorded
Phase 2 NCT02102672 Mar 2014 → Dec 2016 pulmonary arterial hypertension Pontificia Universidad Catolica de Chile Unknown No outcome recorded
Phase 2/32 trials
Phase 2/3 NCT04939857 Jun 2021 → Jul 2022 poisoning Peking University Third Hospital Unknown No outcome recorded
Phase 2/3 NCT03273387 Sep 2017 → Nov 2018 pulmonary arterial hypertension Indonesia University Completed No outcome recorded
Phase 34 trials
Phase 3 NCT04980716 Jun 2021 → Jan 2026 overdue non-small cell lung carcinoma Sun Yat-sen University Recruiting No outcome recorded
Phase 3 NCT03715582 Oct 2018 → Oct 2020 diabetes mellitus, intermediate coronary syndrome University of Sao Paulo General Hospital Unknown No outcome recorded
Phase 3 NCT03274427 Jul 2017 → Jul 2021 hepatocellular carcinoma The First Affiliated Hospital of Zhengzhou University Unknown No outcome recorded
Phase 3 NCT03278444 Jul 2017 → Jul 2021 hepatocellular carcinoma The First Affiliated Hospital of Zhengzhou University Unknown No outcome recorded
Phase 44 trials
Phase 4 NCT05540184 Sep 2022 → Sep 2025 acute kidney injury Beni-Suef University Unknown No outcome recorded
Phase 4 NCT03887013 Mar 2019 → Oct 2020 coronary artery disorder, diastolic heart failure China National Center for Cardiovascular Diseases Unknown No outcome recorded
Phase 4 NCT02107144 Apr 2014 → Mar 2023 coronary artery disorder Clinical Hospital Center Zemun Completed No outcome recorded
Phase 4 NCT00282360 Feb 1999 → Oct 2003 coronary artery disorder, type 2 diabetes mellitus IRCCS San Raffaele Completed No outcome recorded
Phase not applicable5 trials
NCT07074834 Feb 2021 → Sep 2022 coronary artery disorder Shiyan City Renmin Hospital Completed No outcome recorded
NCT03504202 Mar 2019 → Apr 2020 coronary microvascular disorder Shanghai 10th People's Hospital Unknown No outcome recorded
NCT02826616 Jul 2016 → Aug 2017 cardiovascular disorder Chinese PLA General Hospital Unknown No outcome recorded
NCT04511520 Jul 2013 → Dec 2016 paroxysmal atrial fibrillation National Research Center for Preventive Medicine Completed No outcome recorded
NCT01857921 Dec 2010 → Apr 2018 coronary artery disorder Yonsei University Completed No outcome recorded
Also used as a comparator or background therapy in 9 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT03333499 Comparator Nov 2017 → Dec 2018 heart failure Dalian University Unknown No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT06459193 Comparator Jun 2024 → Jan 2025 chemotherapy-induced neuropathy Minia University Completed No outcome recorded
Phase 21 trial
Phase 2 NCT01696370 Comparator Apr 2012 → Apr 2014 hypertrophic cardiomyopathy University College, London Unknown No outcome recorded
Phase 31 trial
Phase 3 NCT06656442 Comparator Sep 2024 → Feb 2025 ischemic stroke Ain Shams University Completed No outcome recorded
Phase 44 trials
Phase 4 NCT05633563 Comparator Oct 2021 → Jun 2023 mitochondrial disease, wild type ATTR amyloidosis Steen Hvitfeldt Poulsen Completed No outcome recorded
Phase 4 NCT04661709 Background Mar 2021 → Mar 2023 intermediate coronary syndrome Guang'anmen Hospital of China Academy of Chinese Medical Sciences Unknown No outcome recorded
Phase 4 NCT03809273 Comparator Aug 2019 → Dec 2020 Shenyang Northern Hospital Completed No outcome recorded
Phase 4 NCT03072082 Background Jun 2017 → Dec 2018 coronary artery disorder Jun Li Unknown No outcome recorded
Phase not applicable1 trial
NCT04702906 Comparator Feb → Jun 2021 poisoning Tanta University Unknown No outcome recorded

Evidence & citations 17 cited values

Every value below carries the sentence it was read from. 35 sources stand behind the page.

FieldValueCited text
Known as Trimetazidine “4. Drugs to improve myocardial metabolism: trimetazidine hydrochloride 35 mg bid” NCT04980716
30

NCT03603249

NCT05540184

NCT06140953

NCT03072082

NCT04760821

NCT03504202

NCT05556005

NCT03274427

NCT06656442

NCT01696370

NCT02826616

NCT03737448

NCT04788745

NCT03715582

NCT03333499

NCT01857921

NCT04511520

NCT04939857

NCT00282360

NCT03273387

NCT04661709

NCT02102672

NCT05633563

NCT02107144

NCT07074834

NCT06459193

NCT04702906

NCT03809273

NCT05147194

NCT03887013

Known as Dilatan ChEMBL registry synonym — accepted as the source's own label CHEMBL203266
Known as metacardia “trimetazidine hydrochloride "metacardia" ® (20 mg three times daily produced by Global NAPI Pharmaceuticals-Egypt)” NCT04702906
Known as NSC-759317 ChEMBL registry synonym — accepted as the source's own label CHEMBL203266
Known as TMZ “Patients, who are trimetazidine (TMZ) naïve, will be randomly assigned to receive trimetazidine plus previous medications (TMZ group) 48h before scheduled PCI” NCT02107144
2

“This prospective study aimed to determine whether trimetazidine (TMZ) alters the pharmacodynamic (PD) effects of clopidogrel.” PMID 31292901 Jul 2019

“Vastarel® (Trimetazidine, TMZ) is an already known drug for the treatment of chest pain.” NCT05633563

Known as Trimetazidina ChEMBL registry synonym — accepted as the source's own label CHEMBL203266
Known as Trimetazidine di-hcl ChEMBL registry synonym — accepted as the source's own label CHEMBL203266
Known as Trimetazidine dihydrochloride “The trimetazidine group will receive conventional standard treatment plus Trimetazidine dihydrochloride "metacardia" ® (20 mg three times daily produced by Pharco-Egypt) will...” NCT04702906
Known as Trimetazidine hcl ChEMBL registry synonym — accepted as the source's own label CHEMBL203266
Known as trimetazidine hydrochloride trimetazidine hydrochloride "metacardia" ® (20 mg three times daily produced by Global NAPI Pharmaceuticals-Egypt)” NCT04702906
2

Trimetazidine hydrochloride may play an anti-tumor role by inhibiting fatty acid oxidation.” NCT03274427

NCT03278444

Known as Trimethazidine dihydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL203266
Known as Vastarel Vastarel® (Trimetazidine, TMZ) is an already known drug for the treatment of chest pain.” NCT05633563
Known as Vastarel MR 35 mg “When the patient is randomized to the trimetazidine pill group, he / she will initiate the medication at 70 mg oral dose (2 tablets of Vastarel ® MR 35 mg single dose) 2 hours...” NCT03715582
Known as Vastarel mr ChEMBL registry synonym — accepted as the source's own label CHEMBL203266
Action Inhibit “free fatty acid inhibition with Trimetazidine” NCT00282360
Modality Small molecule “Trimetazidine is a piperazine derivative.” NCT05147194
Route Oral oral therapy with trimetazidine” PMID 30725091 Mar 2019