Drugs / Isoproterenol
last change Jun 2026 re-read 2 minutes ago

Isoproterenol

Small molecule

Developed for
anorexia nervosa · acute respiratory distress syndrome · cardiac arrest · lipoma · urolithiasis
Investigated by
Laureate Institute for Brain Research, Inc. · University of Missouri-Columbia · American Heart Association · Brain & Behavior Research Foundation · Fredericia Hosptial · Fudan University
+25 more · Guangdong Provincial People's Hospital · Hadassah Medical Organization · Lipothera · NYU Langone Health · National Cancer Institute (NCI) · National Heart, Lung, and Blood Institute (NHLBI) · National Institute of Mental Health (NIMH) · Ningbo No. 1 Hospital · Odense University Hospital · Peking Union Medical College Hospital · Pennington Biomedical Research Center · Renmin Hospital of Wuhan University · Second Affiliated Hospital, School of Medicine, Zhejiang University · Taizhou Hospital of Zhejiang Province affiliated to Wenzhou Medical University · The First Affiliated Hospital of Zhengzhou University · The Second Affiliated Hospital of Harbin Medical University · Union Hospital, Tongji Medical College, Huazhong University of Science and Technology · University of Alberta · University of Arizona · University of Oklahoma · University of Southern Denmark · University of Texas Southwestern Medical Center · University of Wisconsin, Madison · Vanderbilt University Medical Center · West China Hospital

Regulatory milestones approvals, filings & regulatory actions · 3 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansions (2) US (FDA) ISUPREL 1986-10-08 – 1999-05-04 fda.gov
Approved US (FDA) ISUPREL 1948-02-19 fda.gov

Trials 15 · a red edge is where a trial was stopped

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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 03 trials
Phase 0 NCT06520982 Sep 2024 → Jun 2027 expected sympathetic nervous system disorder University of Missouri-Columbia Recruiting No outcome recorded
Phase 0 NCT05219799 Mar 2023 → Jun 2026 overdue isoproterenol-mediated vasodilatation, obesity disorder University of Missouri-Columbia Recruiting No outcome recorded
Phase 0 NCT06643221 Jan 2018 → May 2031 expected leukemia, lymphoma University of Arizona Recruiting No outcome recorded
Phase 11 trial
Phase 1 NCT02833207 Apr 2012 → Nov 2021 obesity disorder University of Wisconsin, Madison Terminated No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT00624416 Oct 2007 → Mar 2009 lipoma Pennington Biomedical Research Center Completed No outcome recorded
Phase 21 trial
Phase 2 NCT00323843 Jun 2006 → Feb 2007 urolithiasis Fredericia Hosptial Unknown No outcome recorded
Phase 43 trials
Phase 4 NCT06473116 Mar 2025 → Jul 2029 expected cardiac arrest University of Southern Denmark Not yet recruiting No outcome recorded
Phase 4 NCT05997732 Oct 2023 → Dec 2027 expected University of Alberta Recruiting No outcome recorded
Phase 4 NCT05658692 Oct 2022 → Oct 2023 acute respiratory distress syndrome Second Affiliated Hospital, School of Medicine, Zhejiang University Unknown No outcome recorded
Phase not applicable6 trials
NCT03019081 Jan 2017 → Aug 2021 anorexia nervosa Laureate Institute for Brain Research, Inc. Unknown No outcome recorded
NCT02725060 Feb 2016 → Oct 2026 expected cardiac rhythm disease, postural orthostatic tachycardia syndrome, primary dysautonomia Vanderbilt University Medical Center Enrolling by invitation No outcome recorded
NCT02615119 Oct 2015 → Jun 2023 anorexia nervosa, brain injury, generalized anxiety disorder, major depressive disorder +1 Laureate Institute for Brain Research, Inc. Completed No outcome recorded
NCT02524145 Jun 2015 → Nov 2017 heart failure University of Texas Southwestern Medical Center Completed No outcome recorded
NCT01377636 Aug 2009 → Sep 2011 NYU Langone Health Completed No outcome recorded
NCT00226551 Aug 1999 → ? coronary artery disorder Hadassah Medical Organization Completed No outcome recorded
Also used as a comparator or background therapy in 8 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT00748059 Background Dec 1996 → Dec 2020 autonomic nervous system disorder, disorder of catecholamine synthesis, orthostatic hypotension Vanderbilt University Medical Center Completed No outcome recorded
Phase 21 trial
Phase 2 NCT03032965 Background Oct 2011 → Jul 2015 paroxysmal atrial fibrillation University of Michigan Completed No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT00428428 Comparator Feb → Nov 2007 benign urinary system neoplasm, urolithiasis Fredericia Hosptial Completed No outcome recorded
Phase not applicable5 trials
NCT06082388 Comparator Nov 2023 → Sep 2025 cardiac rhythm disease Medical University of Lodz Unknown No outcome recorded
NCT04950881 Background Jul 2021 → Dec 2022 Daping Hospital and the Research Institute of Surgery of the Third Military Medical University Unknown No outcome recorded
NCT04274413 Background Feb 2021 CFTR-related disorder, cystic fibrosis The Hospital for Sick Children Withdrawn No outcome recorded
NCT02726620 Background Jan → Dec 2017 hypotensive disorder Vanderbilt University Medical Center Completed No outcome recorded
NCT02310789 Background Jul 2015 → Aug 2016 cystic fibrosis Richard Barry Moss Completed No outcome recorded

Evidence & citations 61 cited values

Every value below carries the sentence it was read from. 25 sources stand behind the page.

FieldValueCited text
Known as Isoproterenol “Lastly, beta-adrenergic sweating will be stimulated by injecting a combination of the following drugs: atropine, isoproterenol, and aminophylline (β-cocktail).” NCT04274413
20

“Agonists include: ATP, Bradykinin (BK), Isoproterenol (ISO), and Acetylcholine (Ach), will be infused 3 times each (order randomized).” NCT02833207

“atropine (0.01-0.02mg/kg) or isoproterenol (1-2 μg/per time)is given intravenously to increase the heart rate.” NCT04950881

“Cocktail composed of atropine (280µM), isoproterenol (160µM), and aminophylline (20 mM).” NCT02310789

isoproterenolNCT05658692

NCT02726620

NCT05997732

NCT00624416

NCT00323843

NCT02725060

NCT00428428

NCT03032965

NCT02524145

NCT02615119

NCT01377636

NCT00226551

NCT00748059

NCT06520982

NCT03019081

NCT05219799

NCT06643221

Known as Aerolone ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Aerotrol ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Aleudrin ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Aludrin ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Aludrine ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Asiprenol ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Asmalar ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Assiprenol ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Bellasthman ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Dl-isoprenaline hydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Euspiran ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Imuprel ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isomenyl ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isomist ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isonorin ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isoprenalina ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isoprenaline ClinicalTrials.gov intervention name — accepted as the source's own label NCT06082388
1

NCT06473116

Known as Isoprenaline hydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isoprenaline hydrochloride, dl- ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isoprenaline sulfate ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isoprenaline sulfate dihydrate ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isoprenaline sulphate ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isoprenalini sulfas ChEMBL registry synonym — accepted as the source's own label CHEMBL434
Known as Isopropydrin ChEMBL registry synonym — accepted as the source's own label CHEMBL434