drugset / Trial / NCT06385925

A Study of TSN1611 Treating Patients With Advanced Solid Tumors Harboring KRAS G12D Mutation

NCT06385925

Phase 1/2 Recruiting 440 enrolled Tyligand Pharmaceuticals (Suzhou) Limited
Non-randomizedSequentialOpen-labelTreatment

Summary

The study is a first-in-human (FIH), open-label, multi-center phase 1/2 study of TSN1611 in subjects with KRAS G12D mutant advanced solid tumors. This study will consist of a phase 1 dose escalation part and phase 2 dose expansion part. This study will evaluate the efficacy of TSN1611 at RP2D(s) through ORR using RECIST version 1.1, and determine and confirm the MTD/RP2D for TSN1611 in combination with cetuximab, in combination with cetuximab and mFOLFOX6, in combination with gemcitabine and albumin-bound paclitaxel in subjects with selected solid tumors.

Timeline

Start
2024-04-29
Primary completion
2026-10-30
Completion
2027-04-30

Drugs

EvaluationDrugModalityDoseRoute
Background Paclitaxel Small molecule Oral
Background Cetuximab Monoclonal antibody 500 mg/m2 Intravenous
Background Gemcitabine Small molecule 1000 mg/m2 Intravenous
Background Leucovorin Small molecule
Background Oxaliplatin Small molecule
Background Paclitaxel Small molecule 125 mg/m2 Intravenous
Background fluorouracil Small molecule

Indications