Drugs / icosapent ethyl
last change Aug 2026 re-read 2 minutes ago

icosapent ethyl

Small molecule

Developed for
hypertriglyceridemia · cardiovascular disorder · atherosclerosis · coronary artery disorder · metabolic dysfunction-associated steatohepatitis · type 2 diabetes mellitus · Alzheimer disease · aortic valve stenosis
+13 more · colon carcinoma · colorectal cancer · COVID-19 · female breast carcinoma · heart failure · hyperlipidemia · inflammatory breast carcinoma · inflammatory disease · intracranial vasospasm · lip disorder · metastasis from malignant tumor of colon · NAFLD1 · respiratory tract infectious disorder
Investigated by
Amarin Pharma Inc. · Mochida Pharmaceutical Company, Ltd. · Canadian Medical and Surgical Knowledge Translation Research Group · HLS Therapeutics, Inc · National Cancer Institute (NCI) · Academic Medical Center - University of Amsterdam
+23 more · Amarin Corporation · Brigham and Women's Hospital · Gilead Sciences · Hospital San Juan de la Cruz · Iwate Medical University · Kobe University · M.D. Anderson Cancer Center · Mark A Hull, PhD FRCP · Marubeni Pharmaceuticals (Suzhou) Co., Ltd. · Massachusetts General Hospital · Nakamura Memorial Hospital · National Institutes of Health (NIH) · Ootemachi Hospital · Ottawa Heart Institute Research Corporation · Tohoku University · Unity Health Toronto · University of Louisville · University of Pennsylvania · University of Wisconsin, Madison · VA Office of Research and Development · Western University, Canada · Yamaguchi University Hospital · Yorkshire Cancer Research

Regulatory milestones approvals, filings & regulatory actions · 3 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved EU (EMA) Vazkepa 2021-03-26 europa.eu
Label expansion US (FDA) VASCEPA 2019-12-13 fda.gov
Approved US (FDA) VASCEPA 2012-07-26 fda.gov

Trials 21 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT03885661 Jan 2016 → Aug 2018 hyperlipidemia, hypertriglyceridemia, lip disorder University of Pennsylvania Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT05198843 Nov 2022 → Dec 2023 female breast carcinoma, inflammatory breast carcinoma National Cancer Institute (NCI) Terminated No outcome recorded
Phase 1/2 NCT04216251 Dec 2020 → Sep 2022 colorectal adenoma, colorectal cancer Massachusetts General Hospital Completed No outcome recorded
Phase 25 trials
Phase 2 NCT06466278 Jun 2023 → Jul 2026 overdue aortic valve stenosis Academic Medical Center - University of Amsterdam Active not recruiting No outcome recorded
Phase 2 NCT04412018 Jun → Nov 2020 COVID-19, inflammatory disease Canadian Medical and Surgical Knowledge Translation Research Group Completed No outcome recorded
Phase 2 NCT02940223 Mar 2017 → Nov 2020 metastatic malignant neoplasm M.D. Anderson Cancer Center Terminated No outcome recorded
Phase 2 NCT02781584 Jun 2016 → Dec 2020 NAFLD1, metabolic dysfunction-associated steatohepatitis Gilead Sciences Completed No outcome recorded
Phase 2 NCT01154985 Jun 2010 → Oct 2012 metabolic dysfunction-associated steatohepatitis Mochida Pharmaceutical Company, Ltd. Completed No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT02719327 Jun 2017 → Sep 2023 Alzheimer disease VA Office of Research and Development Completed No outcome recorded
Phase 38 trials
Phase 3 NCT06710080 Apr → Dec 2026 expected atherosclerosis, pneumonia Ottawa Heart Institute Research Corporation Recruiting No outcome recorded
Phase 3 NCT04239950 May 2020 → Jul 2023 hypertriglyceridemia Mochida Pharmaceutical Company, Ltd. Completed No outcome recorded
Phase 3 NCT03428477 May 2018 → Nov 2025 overdue colon carcinoma, metastasis from malignant tumor of colon Mark A Hull, PhD FRCP Active not recruiting No outcome recorded
Phase 3 NCT02708771 Mar 2016 → Jun 2018 heart failure Hospital San Juan de la Cruz Completed No outcome recorded
Phase 3 NCT02422446 Apr 2015 → Mar 2017 coronary artery disorder, type 2 diabetes mellitus Brigham and Women's Hospital Terminated No outcome recorded
Phase 3 NCT01492361 Nov 2011 → May 2018 cardiovascular disorder Amarin Pharma Inc. Completed No outcome recorded
Phase 3 NCT01047501 Dec 2009 → Feb 2011 hypertriglyceridemia Amarin Pharma Inc. Completed No outcome recorded
Phase 3 NCT01047683 Dec 2009 → Oct 2010 hypertriglyceridemia Amarin Pharma Inc. Completed No outcome recorded
Phase 44 trials
Phase 4 NCT06280976 Mar 2024 → Jan 2025 atherosclerosis, coronary artery disorder, myocardial infarction University of Louisville Withdrawn No outcome recorded
Phase 4 NCT04562467 Sep 2020 → May 2023 cardiovascular disorder, hypertriglyceridemia, type 2 diabetes mellitus Canadian Medical and Surgical Knowledge Translation Research Group Completed No outcome recorded
Phase 4 NCT00839449 Dec 2004 → Jun 2008 intracranial vasospasm, subarachnoid hemorrhage Yamaguchi University Hospital Completed No outcome recorded
Phase 4 NCT00231738 Nov 1996 → Nov 2004 cardiovascular disorder Kobe University Completed No outcome recorded
Also used as a comparator or background therapy in 8 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT02113163 Comparator Mar → Jun 2014 hypertriglyceridemia, type 2 diabetes mellitus Thetis Pharmaceuticals LLC Completed No outcome recorded
Phase 1 NCT02859129 Comparator Sep → Nov 2013 hypertriglyceridemia AstraZeneca Completed No outcome recorded
Phase 22 trials
Phase 2 NCT04177680 Comparator Jun → Nov 2020 hypertriglyceridemia Matinas BioPharma Nanotechnologies, Inc. Completed No outcome recorded
Phase 2 NCT03661047 Comparator Nov 2019 → Nov 2021 colon carcinoma Massachusetts General Hospital Withdrawn No outcome recorded
Phase 32 trials
Phase 3 NCT07680829 Background Aug 2026 → Jun 2030 expected Zhejiang Doer Biologics Co., Ltd. Not yet recruiting No outcome recorded
Phase 3 NCT04460651 Comparator Aug 2020 → Aug 2021 COVID-19 Estudios Clínicos Latino América Completed No outcome recorded
Phase 42 trials
Phase 4 NCT04505098 Comparator Aug 2020 → Dec 2022 COVID-19, atherosclerosis, respiratory tract infectious disorder Kaiser Permanente Terminated No outcome recorded
Phase 4 NCT02926027 Comparator Mar 2017 → May 2020 hypertriglyceridemia Lundquist Institute for Biomedical Innovation at Harbor-UCLA Medical Center Completed No outcome recorded

Press releases naming this drug 1 release

DateIssuerRelease
2023-03-01 CSL Behring CSL Seqirus and Amarin sign licensing agreement to commercialise Vazkepa (icosapent ethyl) in Australia and New Zealand csl.com

Evidence & citations 20 cited values

Every value below carries the sentence it was read from. 35 sources stand behind the page.

FieldValueCited text
Known as icosapent ethyl “AMR101 (icosapent ethyl \[ethyl-EPA\]) is a highly purified ethyl ester of eicosapentaenoic acid (EPA) developed by Amarin Pharma Inc. for the treatment of cardiovascular...” NCT01492361
18

“We evaluated the safety and efficacy of icosapent ethyl (Vascepa) and fenofibrate to mitigate triglyceride elevations in patients with NASH treated with CILO and FIR.” PMID 34999207 Jan 2022

Icosapent ethyl is an omega-3 fatty acid and in a class of medications called antilipemic or lipid-regulating agents.” NCT05198843

Icosapent ethyl (IPE; formerly AMR101) is a high-purity prescription form of eicosapentaenoic acid ethyl ester.” PMID 23312052 Jul 2012

“AMR101 is commercially available in the US as VASCEPA (icosapent ethyl).” NCT03661047

“AMR101 is commercially available in the US as VASCEPA (icosapent ethyl)” NCT04216251

icosapent ethyl or Vascepa” NCT02113163

NCT07680829

NCT02719327

NCT02422446

NCT04460651

NCT04505098

NCT04177680

NCT06710080

NCT06466278

NCT04412018

NCT03885661

NCT03428477

NCT04562467

Known as AMR101 “Icosapent ethyl (IPE; formerly AMR101) is a high-purity prescription form of eicosapentaenoic acid ethyl ester.” PMID 23312052 Jul 2012
4

NCT01492361

NCT03661047

NCT04216251

NCT01047501

Known as Eicosapentaenoic acid ethyl ester “Each capsule contains: 460 mg eicosapentaenoic acid ethyl ester and 380 mg docosahexaenoic acid ethyl ester.” NCT02708771
2

NCT00839449

NCT00231738

Known as EPA-E “This is a controlled study to determine the effectiveness and safety of ethyl icosapentate (EPA-E) in the treatment of adult patients with non-alcoholic steatohepatitis (NASH).” NCT01154985
Known as Epadel ChEMBL registry synonym — accepted as the source's own label CHEMBL2095209
Known as EPADEL Capsule 300 TM “Eicosapentaenoic acid ethyl ester(EPADEL Capsule 300 TM)” NCT00231738
Known as EPADEL S900 TM (EPA ethyl ester, purity >98%) EPADEL S900 TM (EPA ethyl ester, purity >98%)NCT00839449
Known as Ethyl icosapent ChEMBL registry synonym — accepted as the source's own label CHEMBL2095209
Known as ethyl icosapentate “This is a controlled study to determine the effectiveness and safety of ethyl icosapentate (EPA-E) in the treatment of adult patients with non-alcoholic steatohepatitis (NASH).” NCT01154985
3

“AMR101 (ethyl icosapentate) 4 capsules/day for 12 weeks” NCT01047501

NCT04239950

NCT02940223

Known as ethyl-EPA “AMR101 (icosapent ethyl \[ethyl-EPA\]) is a highly purified ethyl ester of eicosapentaenoic acid (EPA) developed by Amarin Pharma Inc. for the treatment of cardiovascular...” NCT01492361
Known as Icosapent ethyl ester ChEMBL registry synonym — accepted as the source's own label CHEMBL2095209
Known as IPE “The EPA for Metastasis Trial 2 trial is a randomised, double-blind, placebo-controlled, phase 3 trial of 4 g EPA ethyl ester (icosapent ethyl (IPE; Vascepa)) daily in patients...” PMID 38030258 Nov 2023
4

“Icosapent ethyl (IPE; formerly AMR101) is a high-purity prescription form of eicosapentaenoic acid ethyl ester.” PMID 23312052 Jul 2012

“Icosapent ethyl (IPE), an omega-3 fatty acid, demonstrates both pro-resolving and cardioprotective properties.” PMID 41781043 Mar 2026

“purified form of the omega-3 fatty acid eicosapentaenoic acid (EPA) called icosapent ethyl (IPE)” NCT02719327

“Icosapent ethyl (IPE) is a safe, well-tolerated oral therapy” NCT04460651

Known as MND-21 MND-21, a highly purified form of ethyl icosapentate” PMID 41500861 Dec 2025
Known as NSC-759597 ChEMBL registry synonym — accepted as the source's own label CHEMBL2095209
Known as Timnodonic acid ethyl ester ChEMBL registry synonym — accepted as the source's own label CHEMBL2095209
Known as Vascepa “We evaluated the safety and efficacy of icosapent ethyl (Vascepa) and fenofibrate to mitigate triglyceride elevations in patients with NASH treated with CILO and FIR.” PMID 34999207 Jan 2022
9

“pre-treatment with icosapent ethyl (IPE), also known as Vascepa®, compared to usual standard of care” NCT04505098

“AMR101 is commercially available in the US as VASCEPA (icosapent ethyl).” NCT03661047

“Icosapent Ethyl 1000 MG Oral Capsule [Vascepa]” NCT06710080

“Icosapent Ethyl 1000 MG [Vascepa]” NCT03885661

“icosapent ethyl or VascepaNCT02113163

VascepaNCT04412018

NCT02859129

NCT06280976

NCT02926027

Known as VASCEPA (icosapent ethyl) “VASCEPA® (icosapent ethyl)” NCT01047683
Known as Vazkepa ChEMBL registry synonym — accepted as the source's own label CHEMBL2095209
Modality Small molecule “Ethyl-eicosapentanoic acid (EPA-E) is a synthetic polyunsaturated fatty acid that reduces hypertriglyceridemia.” PMID 24818764 May 2014
Route Oral “Patients in the group A are orally administered eicosapentaenoic acid ethyl ester.” NCT00839449