Drugs / Icotinib
last change Jul 2026 re-read 2 minutes ago

Icotinib

Small molecule targets EGFR via inhibition

Developed for
non-small cell lung carcinoma · metastatic malignant neoplasm in the brain · lung cancer · adenocarcinoma · lung adenocarcinoma · psoriasis · cancer of unknown primary site · malignant pancreatic neoplasm
+16 more · nasopharyngeal carcinoma · acoustic neuroma · adenosquamous lung carcinoma · breast cancer · bronchial neoplasm · carcinoma of esophagus · esophageal cancer · esophageal squamous cell carcinoma · gastroesophageal junction adenocarcinoma · lung carcinoma · lung large cell carcinoma · lung neoplasm · metastatic malignant neoplasm · neoplastic disease or syndrome · NF2-related schwannomatosis · squamous cell lung carcinoma
Investigated by
Betta Pharmaceuticals Co., Ltd. · Sun Yat-sen University · Tianjin Medical University Cancer Institute and Hospital · Nanfang Hospital, Southern Medical University · Chia Tai Tianqing Pharmaceutical Group Co., Ltd. · Chinese Academy of Medical Sciences
+48 more · Guangdong Association of Clinical Trials · Tigermed Consulting Co., Ltd · Zhejiang Cancer Hospital · Zhejiang University · 307 Hospital of PLA · 309th Hospital of Chinese People's Liberation Army · Affiliated Hospital of Jiangnan University · Anhui Medical University · Beijing Haidian Hospital · Beta Pharma, Inc. · Changzhou No.2 People's Hospital · Chinese PLA General Hospital · Daping Hospital and the Research Institute of Surgery of the Third Military Medical University · First People's Hospital of Hangzhou · Fuda Cancer Hospital, Guangzhou · Fujian Cancer Hospital · Fuzhou General Hospital · Guangdong Provincial People's Hospital · Hangzhou Cancer Hospital · Hebei Medical University Fourth Hospital · Henan Cancer Hospital · Henan Provincial People's Hospital · Jiangsu Simcere Pharmaceutical Co., Ltd. · Jiangyin People's Hospital · Li Peng · Liaoning Cancer Hospital & Institute · LuBing · Nanchang University · Nantong University · Peking University Cancer Hospital & Institute · Peking University People's Hospital · People's Hospital of Guangxi Zhuang Autonomous Region · Qilu Hospital of Shandong University · Quintiles, Inc. · Roswell Park Cancer Institute · Second Affiliated Hospital of Nanchang University · Second Affiliated Hospital of Soochow University · Shandong Cancer Hospital and Institute · Shanghai Chest Hospital · Sichuan Cancer Hospital and Research Institute · Taizhou Hospital · The First Affiliated Hospital of Guangzhou Medical University · The First Affiliated Hospital of Soochow University · The First Affiliated Hospital of Xiamen University · The First People's Hospital of Changzhou · Wu Nan · Yuhong Li · Zaiwen Fan

Trials 84 · started per year

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2009201020112012201320142015201620172018201920202021202220232024202520262027
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT07458919 Mar 2026 → Oct 2030 expected lung cancer Fuzhou General Hospital Not yet recruiting No outcome recorded
Phase 16 trials
Phase 1 NCT02801435 Sep 2016 → Jun 2017 psoriasis Betta Pharmaceuticals Co., Ltd. Completed No outcome recorded
Phase 1 NCT02574091 Nov 2015 → Feb 2017 psoriasis Betta Pharmaceuticals Co., Ltd. Completed No outcome recorded
Phase 1 NCT02278458 Oct 2014 → Jan 2016 malignant pancreatic neoplasm Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 1 NCT02033148 Aug 2014 → Jun 2016 cancer of unknown primary site Roswell Park Cancer Institute Withdrawn No outcome recorded
Phase 1 NCT02066870 Jan 2014 → Sep 2015 non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 1 NCT02024633 Dec 2013 → Dec 2015 malignant pancreatic neoplasm Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT01534585 Feb 2012 → Feb 2013 nasopharyngeal carcinoma Taizhou Hospital Completed No outcome recorded
Phase 1/2 NCT01516983 Dec 2011 → Jun 2013 metastatic malignant neoplasm in the brain, non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Completed No outcome recorded
Phase 246 trials
Phase 2 NCT06517953 Jul 2024 → Jul 2026 overdue non-small cell lung carcinoma Sun Yat-sen University Recruiting No outcome recorded
Phase 2 NCT05536505 Sep 2022 → Oct 2025 overdue Guangdong Association of Clinical Trials Recruiting No outcome recorded
Phase 2 NCT05514314 Sep 2022 → Sep 2024 non-small cell lung carcinoma Wu Nan Unknown No outcome recorded
Phase 2 NCT05263947 Jan 2022 → Dec 2023 non-small cell lung carcinoma Tianjin Medical University Cancer Institute and Hospital Completed No outcome recorded
Phase 2 NCT05132985 Jan 2022 → Jul 2024 overdue non-small cell lung carcinoma Liaoning Cancer Hospital & Institute Not yet recruiting No outcome recorded
Phase 2 NCT05104788 Oct 2021 → Mar 2024 overdue non-small cell lung carcinoma Peking University Cancer Hospital & Institute Recruiting No outcome recorded
Phase 2 NCT05007938 Aug 2021 → Dec 2024 overdue non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Active not recruiting No outcome recorded
Phase 2 NCT04193007 Dec 2019 → Dec 2021 metastatic malignant neoplasm in the brain, non-small cell lung carcinoma Second Affiliated Hospital of Nanchang University Unknown No outcome recorded
Phase 2 NCT03736837 Dec 2018 → Jan 2021 non-small cell lung carcinoma Tianjin Medical University Cancer Institute and Hospital Completed No outcome recorded
Phase 2 NCT03749213 Dec 2018 → Feb 2022 non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 314 trials
Phase 3 NCT06955325 May 2025 → Dec 2030 expected non-small cell lung carcinoma The First Affiliated Hospital of Guangzhou Medical University Not yet recruiting No outcome recorded
Phase 3 NCT04797806 Mar 2021 → Apr 2022 non-small cell lung carcinoma Tianjin Medical University Cancer Institute and Hospital Unknown No outcome recorded
Phase 3 NCT03992885 Jul 2019 → Jul 2020 non-small cell lung carcinoma Tianjin Medical University Cancer Institute and Hospital Unknown No outcome recorded
Phase 3 NCT04058704 Jul 2018 → Dec 2022 metastatic malignant neoplasm in the brain, non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 3 NCT03008109 Feb → Nov 2017 cancer of unknown primary site, non-small cell lung carcinoma Zaiwen Fan Unknown No outcome recorded
Phase 3 NCT02883543 Jun 2016 → Jun 2018 non-small cell lung carcinoma Daping Hospital and the Research Institute of Surgery of the Third Military Medical University Unknown No outcome recorded
Phase 3 NCT02714010 Aug 2015 → Dec 2021 non-small cell lung carcinoma Sun Yat-sen University Unknown No outcome recorded
Phase 3 NCT02448797 Jun 2015 → Jun 2022 non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 3 NCT02125240 Sep 2014 → Dec 2018 adenocarcinoma, non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 3 NCT01996098 Jan 2014 → Dec 2021 lung cancer Sun Yat-sen University Terminated No outcome recorded
Phase 411 trials
Phase 4 NCT02744664 Apr 2016 → Aug 2017 lung neoplasm Fuda Cancer Hospital, Guangzhou Completed No outcome recorded
Phase 4 NCT02778893 Mar 2016 → Mar 2017 non-small cell lung carcinoma Henan Provincial People's Hospital Unknown No outcome recorded
Phase 4 NCT02404675 Apr 2015 → Dec 2017 non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 4 NCT02283424 Oct 2014 → Oct 2017 neoplastic disease or syndrome Chinese PLA General Hospital Unknown No outcome recorded
Phase 4 NCT02194556 Jul 2014 → Jul 2017 adenocarcinoma, non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 4 NCT02031601 Jan 2014 → Dec 2016 non-small cell lung carcinoma Qilu Hospital of Shandong University Unknown No outcome recorded
Phase 4 NCT01926171 Jun 2013 → Sep 2016 non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 4 NCT01720901 Feb 2013 → Dec 2015 non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Suspended No outcome recorded
Phase 4 NCT01665417 Aug 2012 → Jul 2017 adenocarcinoma, non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase 4 NCT01646450 Jul 2012 → Dec 2015 non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase not applicable4 trials
NCT03983811 Jul 2019 → Oct 2021 non-small cell lung carcinoma Nanfang Hospital, Southern Medical University Unknown No outcome recorded
NCT03766490 Mar → Dec 2019 non-small cell lung carcinoma The First Affiliated Hospital of Soochow University Unknown No outcome recorded
NCT03634059 Aug 2018 → Aug 2019 non-small cell lung carcinoma Hebei Medical University Fourth Hospital Unknown No outcome recorded
NCT03258671 Oct 2017 → Dec 2020 non-small cell lung carcinoma LuBing Unknown No outcome recorded
Also used as a comparator or background therapy in 16 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 29 trials
Phase 2 NCT03402464 Background Jan 2018 → Jun 2019 lung adenocarcinoma Peking University Cancer Hospital & Institute Unknown No outcome recorded
Phase 2 NCT03123484 Background Apr 2017 → Apr 2019 non-small cell lung carcinoma China Medical University, China Unknown No outcome recorded
Phase 2 NCT03595644 Background Feb 2017 → Jun 2019 non-small cell lung carcinoma Tongji Hospital Completed No outcome recorded
Phase 2 NCT02788058 Background May 2016 → May 2021 lung adenocarcinoma First People's Hospital of Hangzhou Unknown No outcome recorded
Phase 2 NCT02787447 Background May 2016 → Dec 2017 lung adenocarcinoma First People's Hospital of Hangzhou Unknown No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT04206072 Comparator Dec 2019 → Jul 2022 non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Completed No outcome recorded
Phase 33 trials
Phase 3 NCT06041776 Comparator Mar 2023 → Apr 2028 expected non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Recruiting No outcome recorded
Phase 3 NCT02882984 Background Mar 2015 → Mar 2020 Sichuan Provincial People's Hospital Unknown No outcome recorded
Phase 3 NCT02889692 Background Mar 2013 → Dec 2016 cancer Shanghai University of Traditional Chinese Medicine Completed No outcome recorded
Phase 42 trials
Phase 4 NCT04401059 Comparator Nov 2020 → Sep 2025 adenocarcinoma, non-small cell lung carcinoma Tian Xie Unknown No outcome recorded
Phase 4 NCT02103257 Comparator Mar 2014 → Mar 2016 adenocarcinoma, non-small cell lung carcinoma Betta Pharmaceuticals Co., Ltd. Unknown No outcome recorded
Phase not applicable1 trial
NCT04007835 Background Jul 2019 → Jul 2021 non-small cell lung carcinoma Guangdong Association of Clinical Trials Unknown No outcome recorded

Evidence & citations 10 cited values

Every value below carries the sentence it was read from. 102 sources stand behind the page.

FieldValueCited text
Known as Icotinib “Gefitinib(Iressa,YiRuiKe), Erlotinib(Tarceva), Icotinib(Kaimeina), Osimertinib(Tagrisso), Almonertinib, Furmonertinib, etc.” NCT04401059
97

“Standard EGFR-TKI(Gefitinib, erlotinib or icotinib) Gefitinib: 250mg po Qd Erlotinib: 150mg po Qd Icotinib: 125mg po tid” NCT03595644

Icotinib is administered 125 mg three times per day, until disease progression or untolerated toxicity.” NCT04007835

Icotinib is a new first-generation epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors.” PMID 26148750 Jul 2015

“apatinib 500mg qd po plus Erlotinib 150mg qd po / apatinib 500mg qd po plus Icotinib 125mg tid po” NCT03634059

“Gefitinib 250mg po qd or Erlotinib 150mg po qd or Icotinib 125mg po tid” NCT02788058

“Gefitinib 250mg po qd or Erlotinib 150mg po qd or Icotinib 125mg po tid” NCT02787447

“Gefitinib 250mg po qd or Tarceva 150mg po qd or Icotinib 125mg po tid” NCT02714010

“The MRD positive group would receive icotinib as adjuvant treatment.” NCT05536505

Icotinib: 125 mg is administered orally three times per day.” NCT01707329

Icotinib: 125mg, oral administration, three times per day.” NCT01665417

“EGFR-TKI icotinib:125mg Tid RH-endostatin:15mg/m2 ,d1-7” NCT03008109

icotinib will be administered 150mg/d ivgtt tid” NCT03258671

NCT01926171

NCT03349203

NCT01744925

NCT02820116

NCT01719536

NCT02272127

NCT05007938

NCT02125240

NCT04797806

NCT01465243

NCT07458919

NCT02044328

NCT02215356

NCT02882984

NCT02027090

NCT02574091

NCT01843647

NCT02404675

NCT03402464

NCT01929200

NCT01514877

NCT02066870

NCT05104788

NCT03992885

NCT01516983

NCT03720873

NCT02486354

NCT02033148

NCT02737774

NCT03766490

NCT03222622

NCT03346811

NCT02960607

NCT02934256

NCT02961270

NCT03983811

NCT02024633

NCT03151161

NCT02738983

NCT04058704

NCT03153358

NCT02726568

NCT02009605

NCT01720901

NCT03544814

NCT03736837

NCT01646450

NCT03123484

NCT02283424

NCT01040780

NCT02375581

NCT02375022

NCT02103257

NCT01855854

NCT05263947

NCT06517953

NCT04206072

NCT02264210

NCT01973725

NCT02194556

NCT03396185

NCT05132985

NCT02889692

NCT02430974

NCT06955325

NCT02278458

NCT02191059

NCT01724801

NCT01688713

NCT02883543

NCT01963195

NCT02328261

NCT05514314

NCT01996098

NCT03749213

NCT02407366

NCT02362230

NCT01690390

NCT01534585

NCT03754530

NCT02744664

NCT02031601

NCT02062515

NCT02448797

NCT06041776

Known as Bpi-2009 ChEMBL registry synonym — accepted as the source's own label CHEMBL2087361
Known as BPI-2009H “Icotinib (BPI-2009H), a novel EGFR tyrosine kinase inhibitor, displays potent efficacy in preclinical studies.” PMID 22112293 Nov 2011
Known as Conmana “The primary purposes of this study are to assess the safety and efficacy of using high doses of the drug Icotinib (Conmana) as a way to treat patients with non-small cell lung...” NCT01690390
3

“Erlotinib (trade name: Tarceva®) (150mg oral daily) or Icotinib (trade name: Conmana®) (125mg oral three times a day).” NCT02738983

“high dose of Icotinib (Conmana)” NCT01720901

NCT02778893

Known as ectinib “Intervention: Drug: Icotinib Ectinib 125mg/ tablet, one tablet at a time, three times a day, take orally” NCT03992885
Known as icotinib hydrochloride Icotinib Hydrochloride is an oral, small-molecule epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor, which has been approved for treating advanced non-small...” NCT03222622
3

“To determine the pharmacokinetic (PK) profiles of icotinib (icotinib hydrochloride) in patients with advanced cancers.” NCT02033148

Icotinib Hydrochloride is a small-molecule epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor” NCT02574091

NCT02801435

Action Inhibit “Icotinib, one of the leading compounds selected from our compound library, was found to be a potent and specific epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI)” PMID 22112293 Nov 2011
Modality Small molecule “Icotinib hydrochloride is a novel oral EGFR TKIs” NCT01534585
Route Oral “Icotinib was administered at 125 mg orally 3 times/day until tumor progression or unacceptable toxicity” PMID 26148750 Jul 2015
Target EGFR “Icotinib, one of the leading compounds selected from our compound library, was found to be a potent and specific epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI)” PMID 22112293 Nov 2011