Drugs / Pralatrexate
last change May 2026 re-read 2 minutes ago

Pralatrexate

Other / unclassified targets DHFR via inhibition

Developed for
peripheral T-cell lymphoma, not otherwise specified · T-cell non-Hodgkin lymphoma · anaplastic large cell lymphoma · angioimmunoblastic T-cell lymphoma · cancer of unknown primary site · hepatosplenic T-cell lymphoma · enteropathy-associated T-cell lymphoma · esophageal adenocarcinoma
+36 more · gastroesophageal junction adenocarcinoma · Hodgkins lymphoma · monomorphic epitheliotropic intestinal T-cell lymphoma · mycosis fungoides · Nodal T-follicular helper cell lymphoma, follicular type · plasma cell myeloma · primary cutaneous T-cell lymphoma · subcutaneous panniculitis-like T-cell lymphoma · acute leukemia of ambiguous lineage · acute lymphoblastic leukemia · B-cell non-Hodgkin lymphoma · breast carcinoma · cancer · esophageal squamous cell carcinoma · fallopian tube cancer · follicular lymphoma · gastric adenocarcinoma · gastric squamous cell carcinoma · head and neck cancer · hematopoietic and lymphoid cell neoplasm · lung cancer · lymphoma · non-Hodgkin lymphoma · non-small cell lung carcinoma · ovarian cancer · peritoneum cancer · primary cutaneous aggressive epidermotropic CD8+ T-cell lymphoma · primary cutaneous anaplastic large cell lymphoma · primary cutaneous gamma-delta t-cell lymphoma · Sezary syndrome · transitional cell carcinoma · undifferentiated carcinoma of esophagus · undifferentiated carcinoma of stomach · urinary bladder cancer · Waldenstrom macroglobulinemia · adult T-cell leukemia/lymphoma
Investigated by
National Cancer Institute (NCI) · Acrotech Biopharma Inc. · Spectrum Pharmaceuticals, Inc · National Comprehensive Cancer Network · Memorial Sloan Kettering Cancer Center · City of Hope Medical Center
+21 more · Jennifer Amengual · University of Nebraska · University of Virginia · Axis Clinicals Limited · Brigham and Women's Hospital · Columbia University · Dana-Farber Cancer Institute · Fred Hutchinson Cancer Center · M.D. Anderson Cancer Center · Massachusetts General Hospital · Merck Sharp & Dohme LLC · Mundipharma (China) Pharmaceutical Co. Ltd · Mundipharma K.K. · NYU Langone Health · New York University Cancer Institute · Ohio State University Comprehensive Cancer Center · Otsuka Pharmaceutical Development & Commercialization, Inc. · Roswell Park Cancer Institute · Stanford University · Taiwan Mundipharma Pharmaceuticals Ltd. · University of Washington

Regulatory milestones approvals, filings & regulatory actions · 2 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Refused (EMA) EU (EMA) Folotyn 2012-06-21 europa.eu
Approved US (FDA) FOLOTYN 2009-09-24 fda.gov

Trials 33 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 110 trials
Phase 1 NCT07691450 Jan 2027 → Nov 2029 expected Nodal T-follicular helper cell lymphoma, follicular type, anaplastic large cell lymphoma, angioimmunoblastic T-cell lymphoma, enteropathy-associated T-cell lymphoma +6 City of Hope Medical Center Not yet recruiting No outcome recorded
Phase 1 NCT07036133 Dec 2022 → Feb 2027 expected cancer, hematopoietic and lymphoid cell neoplasm Acrotech Biopharma Inc. Recruiting No outcome recorded
Phase 1 NCT03240211 Feb 2022 → Jul 2025 overdue primary cutaneous T-cell lymphoma University of Virginia Active not recruiting No outcome recorded
Phase 1 NCT02594267 Nov 2015 → Apr 2017 peripheral T-cell lymphoma, not otherwise specified Acrotech Biopharma Inc. Completed No outcome recorded
Phase 1 NCT01532011 Mar 2012 → Jun 2016 cancer of unknown primary site M.D. Anderson Cancer Center Completed No outcome recorded
Phase 1 NCT01206465 Sep 2010 → Feb 2015 cancer of unknown primary site University of Nebraska Completed No outcome recorded
Phase 1 NCT01114282 Aug 2010 → Feb 2014 plasma cell myeloma Stanford University Completed No outcome recorded
Phase 1 NCT01134341 Mar 2010 → Aug 2015 Sezary syndrome, mycosis fungoides, primary cutaneous anaplastic large cell lymphoma Acrotech Biopharma Inc. Completed No outcome recorded
Phase 1 NCT00554827 Aug 2007 → Jan 2012 primary cutaneous T-cell lymphoma Acrotech Biopharma Inc. Completed No outcome recorded
Phase 1 NCT00024245 May 2001 → Apr 2003 cancer of unknown primary site Memorial Sloan Kettering Cancer Center Completed No outcome recorded
Phase 1/28 trials
Phase 1/2 NCT07225985 Apr 2026 → Sep 2030 expected T-cell non-Hodgkin lymphoma Fred Hutchinson Cancer Center Recruiting No outcome recorded
Phase 1/2 NCT03598998 Feb 2019 → May 2023 overdue Nodal T-follicular helper cell lymphoma, follicular type, anaplastic large cell lymphoma, angioimmunoblastic T-cell lymphoma, enteropathy-associated T-cell lymphoma +6 City of Hope Medical Center Active not recruiting No outcome recorded
Phase 1/2 NCT03161223 May 2018 → Feb 2023 overdue T-cell non-Hodgkin lymphoma University of Virginia Recruiting No outcome recorded
Phase 1/2 NCT02013362 Mar 2014 → Dec 2015 peripheral T-cell lymphoma, not otherwise specified Mundipharma K.K. Completed No outcome recorded
Phase 1/2 NCT01947140 Sep 2013 → Sep 2022 Hodgkins lymphoma, non-Hodgkin lymphoma, plasma cell myeloma Jennifer Amengual Completed No outcome recorded
Phase 1/2 NCT01188876 Aug 2010 → Jul 2016 fallopian tube cancer, ovarian cancer, peritoneum cancer Massachusetts General Hospital Completed No outcome recorded
Phase 1/2 NCT00481871 May 2007 → May 2011 Hodgkins lymphoma, T-cell non-Hodgkin lymphoma, Waldenstrom macroglobulinemia Acrotech Biopharma Inc. Completed No outcome recorded
Phase 1/2 NCT00052442 Aug 2002 → Mar 2009 lymphoma Spectrum Pharmaceuticals, Inc Completed No outcome recorded
Phase 210 trials
Phase 2 NCT01336933 Jul 2011 → Dec 2016 anaplastic large cell lymphoma, angioimmunoblastic T-cell lymphoma, hepatosplenic T-cell lymphoma, peripheral T-cell lymphoma, not otherwise specified University of Nebraska Completed No outcome recorded
Phase 2 NCT01178944 Sep 2010 → Jan 2015 esophageal adenocarcinoma, gastric adenocarcinoma, gastric squamous cell carcinoma, gastroesophageal junction adenocarcinoma +2 Roswell Park Cancer Institute Completed No outcome recorded
Phase 2 NCT01183065 Aug 2010 → Apr 2014 head and neck cancer Memorial Sloan Kettering Cancer Center Completed No outcome recorded
Phase 2 NCT01129206 Jul 2010 → Sep 2012 esophageal adenocarcinoma, esophageal squamous cell carcinoma, gastroesophageal junction adenocarcinoma Ohio State University Comprehensive Cancer Center Completed No outcome recorded
Phase 2 NCT01118624 Mar 2010 → Apr 2012 breast carcinoma Acrotech Biopharma Inc. Completed No outcome recorded
Phase 2 NCT00998946 Sep 2009 → Aug 2012 B-cell non-Hodgkin lymphoma Spectrum Pharmaceuticals, Inc Completed No outcome recorded
Phase 2 NCT00722553 Jul 2008 → Apr 2011 transitional cell carcinoma, urinary bladder cancer Acrotech Biopharma Inc. Completed No outcome recorded
Phase 2 NCT00606502 Jan 2008 → Jun 2010 non-small cell lung carcinoma Spectrum Pharmaceuticals, Inc Completed No outcome recorded
Phase 2 NCT00364923 Aug 2006 → Jan 2009 peripheral T-cell lymphoma, not otherwise specified Acrotech Biopharma Inc. Completed No outcome recorded
Phase 2 NCT00004238 Jul 1999 → Jun 2002 lung cancer Memorial Sloan Kettering Cancer Center Completed No outcome recorded
Phase 33 trials
Phase 3 NCT03355768 Sep → Nov 2018 peripheral T-cell lymphoma, not otherwise specified Jennifer Amengual Withdrawn No outcome recorded
Phase 3 NCT03349333 Sep 2015 → Jul 2017 T-cell non-Hodgkin lymphoma, peripheral T-cell lymphoma, not otherwise specified Mundipharma (China) Pharmaceutical Co. Ltd Completed No outcome recorded
Phase 3 NCT01420679 Aug 2011 → Dec 2017 peripheral T-cell lymphoma, not otherwise specified Spectrum Pharmaceuticals, Inc Terminated No outcome recorded
Phase 41 trial
Phase 4 NCT03150602 Aug 2016 → Dec 2020 lymphoid system deterioration, progressive, peripheral T-cell lymphoma, not otherwise specified Taiwan Mundipharma Pharmaceuticals Ltd. Unknown No outcome recorded
Phase not applicable1 trial
NCT02551718 Sep 2015 → Jun 2020 acute leukemia of ambiguous lineage, acute lymphoblastic leukemia University of Washington Completed No outcome recorded
Also used as a comparator or background therapy in 8 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 12 trials
Phase 1 NCT01820091 Background Apr 2013 → Apr 2015 non-small cell lung carcinoma Acrotech Biopharma Inc. Withdrawn No outcome recorded
Phase 1 NCT01789723 Background Mar 2013 → Mar 2015 non-Hodgkin lymphoma Acrotech Biopharma Inc. Withdrawn No outcome recorded
Phase 23 trials
Phase 2 NCT04747236 Comparator Feb 2021 → Jun 2028 expected University of Virginia Recruiting No outcome recorded
Phase 2 NCT02106650 Background Jul 2014 → Oct 2018 peripheral T-cell lymphoma, not otherwise specified Acrotech Biopharma Inc. Completed No outcome recorded
Phase 2 NCT01626664 Comparator Jun 2012 → Aug 2015 adult T-cell leukemia/lymphoma Kyowa Kirin, Inc. Completed No outcome recorded
Phase 33 trials
Phase 3 NCT06561048 Comparator Oct 2024 → Nov 2027 expected Nodal T-follicular helper cell lymphoma, follicular type, anaplastic large cell lymphoma, angioimmunoblastic T-cell lymphoma, peripheral T-cell lymphoma, not otherwise specified Corvus Pharmaceuticals, Inc. Recruiting No outcome recorded
Phase 3 NCT06072131 Comparator Oct 2023 → Jul 2030 expected peripheral T-cell lymphoma, not otherwise specified Acrotech Biopharma Inc. Recruiting No outcome recorded
Phase 3 NCT01482962 Comparator Jun 2012 → Jun 2015 peripheral T-cell lymphoma, not otherwise specified Millennium Pharmaceuticals, Inc. Completed No outcome recorded

Evidence & citations 9 cited values

Every value below carries the sentence it was read from. 42 sources stand behind the page.

FieldValueCited text
Known as pralatrexate “Ponatinib Pralatrexate Rapamycin” NCT02551718
38

Pralatrexate (Folotyn)” NCT02106650

NCT01188876

NCT01336933

NCT00364923

NCT00052442

NCT03355768

NCT03161223

NCT01532011

NCT01129206

NCT01206465

NCT06072131

NCT00998946

NCT00722553

NCT01420679

NCT03240211

NCT03598998

NCT00024245

NCT00481871

NCT03349333

NCT07225985

NCT01626664

NCT01178944

NCT01114282

NCT01183065

NCT06561048

NCT02594267

NCT03150602

NCT00606502

NCT04747236

NCT00554827

NCT07691450

NCT01482962

NCT02013362

NCT01118624

NCT01134341

NCT00004238

NCT01947140

NCT07036133

Known as Folotyn “Pralatrexate (Folotyn)” NCT02106650
2

NCT01820091

NCT01789723

Known as Folotyn - (Pralatrexate) Folotyn - (Pralatrexate)NCT01789723
Known as NSC-754230 ChEMBL registry synonym — accepted as the source's own label CHEMBL1201746
Known as Pralatrexato ChEMBL registry synonym — accepted as the source's own label CHEMBL1201746
Action Inhibit “Pralatrexate may stop the growth of tumor cells by blocking some of the enzymes needed for cell growth.” NCT01129206
Modality Other / unclassified “It is a type of dihydrofolate reductase (DHFR) inhibitor.” NCT07225985
Route Intravenous “Pralatrexate (PDX) 135 mg/m\^2 administered as an intravenous (IV) infusion over one hour” NCT00052442
Target DHFR “dihydrofolate reductase (DHFR) inhibitor” NCT07225985