Drugs / Ledipasvir
last change Dec 2023 re-read 2 minutes ago

Ledipasvir

Small molecule

Developed for
chronic hepatitis C virus infection · hepatitis C virus infection · COVID-19 · hepatocellular carcinoma · indolent B-cell non-Hodgkin lymphoma · acute hepatitis C virus infection · cirrhosis of liver · hepatitis
+2 more · hepatitis B virus infection · porphyria cutanea tarda
Investigated by
Gilead Sciences · National Institute of Allergy and Infectious Diseases (NIAID) · ANRS, Emerging Infectious Diseases · National Taiwan University Hospital · University of Maryland, Baltimore · Advancing Clinical Therapeutics Globally for HIV/AIDS and Other Infections
+55 more · Ain Shams University · Alexandria University · Almaza Military Fever Hospital · Assiut University · Bakhtar Bioshimi Co · Baqiyatallah Research Center for Gastroenterology and Liver Diseases · Beijing 302 Hospital · Cairo University · Catherine Chappell · Chang Gung Memorial Hospital · Chi Mei Medical Hospital · Chiayi Christian Hospital · China Medical University Hospital · City of Hope National Medical Center · Clément Sophie · Directorate of Health and Family Welfare, Punjab · Duke University · Emory University · Fondazione Italiana Linfomi - ETS · Gastaldi Giacomo · Genuine Research Center, Egypt · Hannover Medical School · Helwan University · HepNet Study House, German Liverfoundation · Humanity and Health Research Centre · Iran Hepatitis Network · Janssen Sciences Ireland UC · Kaiser Permanente · Kaohsiung Medical University Chung-Ho Memorial Hospital · Mansoura University Children Hospital · Marqués de Valdecilla Research Institute (IDIVAL) · MinaPharm Pharmaceuticals · National Cheng-Kung University Hospital · National Hepatology & Tropical Medicine Research Institute · National Institute of Diabetes and Digestive and Kidney Diseases (NIDDK) · National Institutes of Health (NIH) · National Institutes of Health Clinical Center (CC) · National Liver Institute, Egypt · Peter J. Ruane, M.D., Inc. · Post Graduate Institute of Medical Education and Research, Chandigarh · Ram Manohar Lohia Institute of Medical Sciences, Lucknow · Sanjay Gandhi Postgraduate Institute of Medical Sciences · Stanford University · Taipei Veterans General Hospital, Taiwan · Tanta University · Tanta University · Tehran University of Medical Sciences · Tri-Service General Hospital (TSGH) · University Health Network, Toronto · University Hospital, Geneva · University of Colorado, Denver · University of Nebraska · University of Wuerzburg · Wake Forest University Health Sciences · Yassin Abdelghaffar Charity Center for Liver Disease and Research

Regulatory milestones approvals, filings & regulatory actions · 2 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved EU (EMA) Harvoni 2014-11-17 europa.eu
Approved US (FDA) HARVONI 2014-10-10 fda.gov

Trials 50 · a red edge is where a trial was stopped

PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT03702218 Jul 2019 hepatitis C virus infection University of Maryland, Baltimore Withdrawn No outcome recorded
Phase 13 trials
Phase 1 NCT04039958 Apr → May 2017 Genuine Research Center, Egypt Completed No outcome recorded
Phase 1 NCT02683005 Sep 2016 → Feb 2020 chronic hepatitis C virus infection, pregnancy disorder Catherine Chappell Completed No outcome recorded
Phase 1 NCT02128217 May 2014 → Feb 2017 HIV infectious disease, hepatitis Advancing Clinical Therapeutics Globally for HIV/AIDS and Other Infections Completed No outcome recorded
Phase 217 trials
Phase 2 NCT03312023 Feb 2018 → Aug 2020 hepatitis B virus infection University of Maryland, Baltimore Completed No outcome recorded
Phase 2 NCT03118674 Sep 2017 → Mar 2022 hepatitis C virus infection, porphyria cutanea tarda Wake Forest University Health Sciences Completed No outcome recorded
Phase 2 NCT03261349 Sep 2017 → Dec 2020 indolent B-cell non-Hodgkin lymphoma National Taiwan University Hospital Unknown No outcome recorded
Phase 2 NCT02836925 Mar 2016 → Feb 2020 hepatitis C virus infection, indolent B-cell non-Hodgkin lymphoma Fondazione Italiana Linfomi - ETS Completed No outcome recorded
Phase 2 NCT02405013 Oct 2015 → Jul 2017 HIV infectious disease, hepatitis C virus infection ANRS, Emerging Infectious Diseases Completed No outcome recorded
Phase 2 NCT02421211 May → Nov 2015 chronic hepatitis C virus infection Janssen Sciences Ireland UC Completed No outcome recorded
Phase 2 NCT02470858 Jan → Dec 2015 chronic hepatitis C virus infection Humanity and Health Research Centre Completed No outcome recorded
Phase 2 NCT02249182 Nov 2014 → Jun 2018 hepatitis C virus infection Gilead Sciences Completed No outcome recorded
Phase 2 NCT02309918 Nov 2014 → Aug 2016 acute hepatitis C virus infection HepNet Study House, German Liverfoundation Completed No outcome recorded
Phase 2 NCT02125500 Aug 2014 → Dec 2015 HIV infectious disease, hepatitis C virus infection ANRS, Emerging Infectious Diseases Completed No outcome recorded
Phase 310 trials
Phase 3 NCT04530422 Apr → Jul 2020 COVID-19 Almaza Military Fever Hospital Completed No outcome recorded
Phase 3 NCT04353986 Jun 2018 → Apr 2023 beta-thalassemia major, hepatitis C virus infection Ain Shams University Unknown No outcome recorded
Phase 3 NCT03061032 Mar 2017 → Dec 2018 hepatitis C virus infection Iran Hepatitis Network Unknown No outcome recorded
Phase 3 NCT02705534 Sep 2016 → Sep 2017 cirrhosis of liver, hepatitis C virus infection Tehran University of Medical Sciences Completed No outcome recorded
Phase 3 NCT02707601 Apr 2016 → Sep 2017 HIV infectious disease, hepatitis C virus infection Gilead Sciences Completed No outcome recorded
Phase 3 NCT02771405 Mar 2016 → Dec 2017 chronic hepatitis C virus infection, hepatocellular carcinoma National Hepatology & Tropical Medicine Research Institute Completed No outcome recorded
Phase 3 NCT02478229 Jun 2015 → Apr 2016 hepatitis C virus infection University Health Network, Toronto Terminated No outcome recorded
Phase 3 NCT02073656 Feb → Nov 2014 HIV infectious disease, chronic hepatitis C virus infection Gilead Sciences Completed No outcome recorded
Phase 3 NCT02021656 Dec 2013 → Jul 2017 chronic hepatitis C virus infection Gilead Sciences Completed No outcome recorded
Phase 3 NCT01975675 Oct 2013 → Jun 2014 chronic hepatitis C virus infection Gilead Sciences Completed No outcome recorded
Phase 414 trials
Phase 4 NCT04498936 Jul → Oct 2020 COVID-19 Assiut University Completed No outcome recorded
Phase 4 NCT03743727 Aug 2018 → Mar 2019 Yassin Abdelghaffar Charity Center for Liver Disease and Research Unknown No outcome recorded
Phase 4 NCT03721627 Apr 2018 → Apr 2019 Gaucher disease, chronic hepatitis C virus infection Mansoura University Children Hospital Unknown No outcome recorded
Phase 4 NCT03126370 Jan 2018 → Jul 2019 coinfection, hepatitis C virus infection University of Colorado, Denver Completed No outcome recorded
Phase 4 NCT04457050 Oct 2017 → Nov 2019 chronic hepatitis C virus infection Alexandria University Completed No outcome recorded
Phase 4 NCT03961828 Oct 2017 → Dec 2018 beta thalassemia, hepatitis C virus infection Tanta University Completed No outcome recorded
Phase 4 NCT03279133 Sep 2017 → Feb 2018 disease related to hematopoietic stem cell transplant Kaiser Permanente Withdrawn No outcome recorded
Phase 4 NCT03402165 Jan 2017 → Dec 2022 hepatitis C virus infection Tanta University Unknown No outcome recorded
Phase 4 NCT02858180 Dec 2016 → Apr 2019 chronic hepatitis C virus infection, chronic obstructive pulmonary disease, heart failure, interstitial lung disease Duke University Completed No outcome recorded
Phase 4 NCT02959359 Nov 2016 → Jun 2022 hepatocellular carcinoma Taipei Veterans General Hospital, Taiwan Withdrawn No outcome recorded
Phase not applicable5 trials
NCT03764345 Dec 2018 → Jul 2019 chronic hepatitis C virus infection National Liver Institute, Egypt Completed No outcome recorded
NCT03483987 Feb 2018 → Apr 2022 chronic hepatitis C virus infection Sanjay Gandhi Postgraduate Institute of Medical Sciences Terminated No outcome recorded
NCT03488485 Jun 2016 → Dec 2020 chronic hepatitis C virus infection Post Graduate Institute of Medical Education and Research, Chandigarh Unknown No outcome recorded
NCT02760355 Mar 2016 → Jun 2018 University Hospital, Geneva Completed No outcome recorded
NCT02469012 Oct 2014 → Oct 2016 chronic hepatitis C virus infection University of Wuerzburg Unknown No outcome recorded
Also used as a comparator or background therapy in 13 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT03188276 Comparator Feb 2016 → May 2017 chronic hepatitis C virus infection Third Affiliated Hospital, Sun Yat-Sen University Completed No outcome recorded
Phase 12 trials
Phase 1 NCT03005210 Comparator Nov 2016 Genuine Research Center, Egypt Completed No outcome recorded
Phase 1 NCT01193478 Comparator Aug 2010 → Jan 2011 hepatitis C virus infection Gilead Sciences Completed No outcome recorded
Phase 24 trials
Phase 2 NCT01435226 Comparator Sep 2011 → Jan 2013 chronic hepatitis C virus infection Gilead Sciences Completed No outcome recorded
Phase 2 NCT01434498 Comparator Sep 2011 → Jan 2013 chronic hepatitis C virus infection Gilead Sciences Completed No outcome recorded
Phase 2 NCT01356160 Comparator Jul 2011 → Jun 2013 chronic hepatitis C virus infection Gilead Sciences Completed No outcome recorded
Phase 2 NCT01353248 Comparator May 2011 → Oct 2012 chronic hepatitis C virus infection Gilead Sciences Completed No outcome recorded
Phase 32 trials
Phase 3 NCT03343444 Comparator Apr 2017 → Nov 2018 chronic hepatitis C virus infection Egyptian Liver Hospital Unknown No outcome recorded
Phase 3 NCT02363517 Comparator Feb 2015 → Dec 2018 hepatitis C virus infection, substance abuse Macfarlane Burnet Institute for Medical Research and Public Health Ltd Unknown No outcome recorded
Phase 43 trials
Phase 4 NCT02347345 Comparator Nov 2016 hepatitis C virus infection Rockefeller University Completed No outcome recorded
Phase 4 NCT02992457 Comparator Jan 2015 → Dec 2018 hepatitis C virus infection Tanta University Completed No outcome recorded
Phase 4 NCT03133065 Comparator Sep 2014 → Dec 2016 Ain Shams University Completed No outcome recorded
Phase not applicable1 trial
NCT03481036 Comparator Jun 2016 → Dec 2020 chronic hepatitis C virus infection Post Graduate Institute of Medical Education and Research, Chandigarh Unknown No outcome recorded

Press releases naming this drug 15 releases

DateIssuerRelease
2018-12-04 Gilead Sciences China’s National Medical Products Administration Approves Harvoni® (Ledipasvir/Sofosbuvir) for Treatment of Chronic Hepatitis C Virus Genotype 1-6 gilead.com
2018-09-24 Gilead Sciences Gilead Subsidiary to Launch Authorized Generics of Epclusa® (Sofosbuvir/Velpatasvir) and Harvoni® (Ledipasvir/Sofosbuvir) for the Treatment of Chronic Hepatitis C gilead.com
2017-04-21 Gilead Sciences Gilead Announces Scientific Presentations Demonstrating Efficacy of Harvoni® (Ledipasvir/Sofosbuvir) in Special Patient Populations With HCV Infection gilead.com
2014-11-18 Gilead Sciences European Commission Grants Marketing Authorization for Gilead’s Harvoni®▼ (Ledipasvir/Sofosbuvir), the First Single Tablet Regimen to Treat the Majority of Chronic Hepatitis C Patients With Genotype 1 and 4 gilead.com
2014-10-16 Gilead Sciences Health Canada Issues Notice of Compliance for Gilead’s Harvoni™ (Ledipasvir/Sofosbuvir), the First Once-Daily Single Tablet Regimen for the Treatment of Genotype 1 Chronic Hepatitis C gilead.com
2014-10-10 Gilead Sciences U.S. Food and Drug Administration Approves Gilead’s Harvoni® (Ledipasvir/Sofosbuvir), the First Once-Daily Single Tablet Regimen for the Treatment of Genotype 1 Chronic Hepatitis C gilead.com
2014-09-26 Gilead Sciences European CHMP Adopts Positive Opinion for Gilead’s Harvoni® (Ledipasvir/Sofosbuvir) for the Treatment of Chronic Hepatitis C Infection in Adults gilead.com
2014-09-24 Gilead Sciences Gilead Submits New Drug Application to Japan’s Pharmaceutical and Medical Devices Agency for Fixed-Dose Combination of Ledipasvir/Sofosbuvir for Chronic Hepatitis C Genotype 1 Infection gilead.com
2014-06-15 Gilead Sciences Gilead Announces Phase 3 Data Showing That the Fixed-Dose Combination of Ledipasvir/Sofosbuvir Achieved 100 Percent Sustained Virologic Response (SVR12) Among Patients with Chronic Hepatitis C in Japan gilead.com
2014-04-07 Gilead Sciences Gilead Announces U.S. FDA Priority Review Designation for Ledipasvir/Sofosbuvir Fixed-Dose Combination Tablet for Chronic Hepatitis C Genotype 1 Infection gilead.com
2014-03-27 Gilead Sciences European Medicines Agency Validates Gilead’s Marketing Application for Ledipasvir/Sofosbuvir Fixed-Dose Combination Tablet for Genotype 1 Chronic Hepatitis C Infection gilead.com
2014-02-10 Gilead Sciences Gilead Files for U.S. Approval of Ledipasvir/Sofosbuvir Fixed-Dose Combination Tablet for Genotype 1 Hepatitis C gilead.com

Evidence & citations 10 cited values

Every value below carries the sentence it was read from. 69 sources stand behind the page.

FieldValueCited text
Known as Ledipasvir “This study will evaluate efficacy of ledipasvir/sofosbuvir (LDV/SOF) and safety and tolerability of switching to elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide...” NCT02707601
54

“This study is to evaluate the antiviral efficacy, safety, and tolerability of combination therapy with ledipasvir/sofosbuvir (LDV/SOF) fixed-dose combination (FDC) +...” NCT02226549

“Chinese patients with chronic HCV genotype 1b infection without cirrhosis were randomly allocated by a computer program to one of three treatment groups (sofosbuvir,...” PMID 27917405 Jul 2016

“After taking tenofovir alafenamide/emtricitabine for 12 weeks, participants will then start taking ledipasvir 90 mg/sofosbuvir 400 mg (Harvoni) in combination with the...” NCT03126370

“Study to Investigate the Efficacy and Safety of Ledipasvir/Sofosbuvir Fixed-Dose Combination for 12 Weeks in Subjects With Chronic Genotype 1 and 4 HCV Infection With Autoimmune Disease” NCT02691728

Ledipasvir/sofosbuvir is a two-drug, fixed-dose combination tablet approved in the USA, European Union, and Japan for chronic genotype 1 HCV infection.” PMID 27198664 May 2016

“For adolescents aged 12-17 years, the safety and efficacy of the fixed-dose combination sofosbuvir and ledipasvir for genotype 1 or 4 infection” NCT03764345

“One hundred patients aged 12-17 years received a combination tablet of 90 mg ledipasvir and 400 mg sofosbuvir once daily for 12 weeks.” PMID 27997679 Jun 2017

“Sofosbuvir/Ledipasvir 400mg/90mg (Harvoni®) in treatment-naïve patients infected with HCV genotype 1 or genotype 4 (12-week course)” NCT02405013

“Patients were given ledipasvir (90 mg) plus sofosbuvir (400 mg) as a fixed-dose combination tablet once daily for 6 weeks.” PMID 28029529 Oct 2016

“Eligible and consenting patients will be treated with sofosbuvir 400 mg daily and ledipasvir 90 mg daily for 8 weeks.” NCT02480166

“One capsule of Harvoni/ ledipasvir, 90 mg + sofosbuvir, 400 mg administered daily for 8, 12, or 24 weeks” NCT03118674

“the hepatitis C virus NS5A inhibitor ledipasvir and the NS5B nucleotide polymerase inhibitor sofosbuvir” PMID 25863559 Apr 2015

“Patients weighing 35 kg or more will receive the adult dose: ledipasvir (90 mg)/sofosbuvir (400 mg).” NCT03743727

“Fixed dose combination of sofosbuvir 400 mg plus ledipasvir 90 mg once daily plus ribavirin 1000 mg” NCT03483987

“sofosbuvir (SOF) + ledipasvir (LDV) or SOF + daclatasvir (DCV) ± ribavirin (RBV)” NCT03488485

“Test drug (Soviredia)1 tablet contains 400 mg Sofosbuvir and 90 mg LedipasvirNCT04039958

“2 recipient are treated with sofosbuvir 400mg + ledipasvir 90mg for 24 weeks” NCT03133065

“Harvoni (ledipasvir/sofosbuvir) + Ribavirin - Genotypes 1, 4, 5, 6; GFR\>30” NCT03702218

“Sofosbuvir, Ledipasvir, Ribavirin for Hepatitis C Cirrhotics, Genotype 1” NCT02705534

Ledipasvir and Sofosbuvir for HCV in Patients Coinfected with HIV-1.” PMID 26196665 Jul 2015

“1 tablet contains 400 mg Sofosbuvir and 90 mg LedipasvirNCT03005210

Ledipasvir (LDV) tablets administered orally once daily” NCT01260350

“Sofosbuvir and Ledipasvir with weight based Ribavirin” NCT03481036

“combination of sofosbuvir plus ledipasvir (SOF + LDP)” NCT02363517

“Sofosbuvir + LedipasvirNCT02469012

NCT02125500

NCT02347345

NCT02478229

NCT03721627

NCT02081079

NCT02959359

NCT02128217

NCT03343444

NCT02771405

NCT04353986

NCT02339038

NCT03312023

NCT02858180

NCT02768961

NCT04498936

NCT04457050

NCT03279133

NCT03961828

NCT04530422

NCT02421211

NCT02683005

NCT03061032

NCT02992457

NCT01805882

NCT03261349

NCT03402165

NCT02760355

NCT02836925

NCT03188276

Known as GS-5885 “a fixed dose combination of GS-7977 and GS-5885 in HIV/HCV Genotype 1 (GT-1) subjects” NCT01878799
8

“Ledipasvir is also known as GS-5885.” NCT02125500

NCT01353248

NCT01371578

NCT01384383

NCT01356160

NCT01435226

NCT01434498

NCT01193478

Known as LDP “combination of sofosbuvir plus ledipasvir (SOF + LDP)” NCT02363517
Known as LDV “This study is to evaluate the antiviral efficacy, safety, and tolerability of combination therapy with ledipasvir/sofosbuvir (LDV/SOF) fixed-dose combination (FDC) +...” NCT02226549
10

“containing the NS5B polymerase inhibitor sofosbuvir (SOF) 90 mg and the NS5A inhibitor ledipasvir (LDV) 400mg, marked a new era of IFN and ribavirin free, directly acting...” NCT02683005

“In India, four DAAs are available (sofosbuvir [SOF], daclatasvir [DCV], ledipasvir [LDV] and velpatasvir [VEL]).” NCT03483987

“Ledipasvir/Sofosbuvir fixed dose combination (FDC) tablet (LDV 90 mg/SOF 400 mg) once daily” NCT02309918

“combined therapy ledipasvir (LDV) and sofosbuvir (SOF) for treating HCV Genotype 4” NCT03743727

“G1, 4, 5, and 6 patients were treated with SOF+ledipasvir (LDV)+RBV for 12 weeks” PMID 30211847 Jan 2019

“sofosbuvir (SOF) + ledipasvir (LDV) or SOF + daclatasvir (DCV) ± ribavirin (RBV)” NCT03488485

“Includes 400 mg sofosbuvir (SOF) and 90 mg ledipasvir (LDV)” NCT02858180

“Ledipasvir (LDV) tablets administered orally once daily” NCT01260350

“sofosbuvir (SOF)/ledipasvir (LDV)” NCT01975675

“Ledipasvir (LDV)” NCT02421211

Known as Ledipasvir (GS-5885) Ledipasvir (GS-5885)NCT01805882
Known as Ledipasvir acetonate ChEMBL registry synonym — accepted as the source's own label CHEMBL2374220
Known as Ledipasvir component of harvoni ChEMBL registry synonym — accepted as the source's own label CHEMBL2374220
Action Inhibit “GS-5885 is a novel hepatitis C virus (HCV) NS5A inhibitor.” PMID 23877691 Jul 2013
Modality Small molecule “NS5A inhibitor ledipasvir” PMID 24262278 Nov 2013
Route Oral “tablet, oral, 3 mg once daily for 3 days” NCT01193478