Drugs / Iloprost
last change 3 days ago re-read 2 minutes ago

Iloprost

Other / unclassified targets PTGIR via activation

Developed for
pulmonary hypertension · pulmonary arterial hypertension · chronic obstructive pulmonary disease · lung cancer · acute respiratory distress syndrome · infectious disease with sepsis · congenital heart disease · COVID-19
+26 more · lung carcinoma · type 2 diabetes mellitus · acute lung injury · acute respiratory failure · asthma · cardiac arrest · diastolic heart failure · Eisenmenger syndrome · idiopathic pulmonary fibrosis · left ventricular failure · multiple organ dysfunction syndrome · myocardial infarction · peripheral arterial disease · peripheral arterial occlusive disease 1 · pneumonia · precancerous condition · pulmonary hypertension owing to lung disease and/or hypoxia · Raynaud disease · respiratory failure · respiratory system disorder · sarcoidosis · sickle cell disease · systemic sclerosis · adult acute respiratory distress syndrome · chronic ulcer of skin · hypertensive disorder
Investigated by
Actelion · Bayer · Yonsei University · Pär Johansson · National Cancer Institute (NCI) · Duke University
+50 more · Heidelberg University · Rigshospitalet, Denmark · Shanghai Jiao Tong University School of Medicine · Thrombologic ApS · University of Oklahoma · University of Sao Paulo General Hospital · Aalborg University Hospital · Aarhus University Hospital · Air Force Military Medical University, China · Algora · Amsterdam UMC, location VUmc · Anders Perner · Assistance Publique - Hôpitaux de Paris · Cardiothoracic Surgical Group of Chinese Society of Pediatric Surgery · Carmel Medical Center · Charite University, Berlin, Germany · Fadoi Foundation, Italy · Hamad Medical Corporation · Independent Research Fund Denmark · Innovation Fund Denmark · Interstitial Lung Disease Study Group, Korea · Jakob Stensballe, MD, PhD · Lene Holmvang · Loma Linda University · Louisiana State University Health Sciences Center in New Orleans · Ludwig-Maximilians - University of Munich · Lund University Hospital · National Center for Research Resources (NCRR) · National Taiwan University Hospital · Novotech (Australia) Pty Limited · Odense University Hospital · Onassis Cardiac Surgery Centre · Oslo University Hospital · Pharmosa Biopharm Inc. · Prim PD Dr Afshin Assadian · Seattle Children's Hospital · Seoul St. Mary's Hospital · Sisse R. Ostrowski, MD PhD DMSc · The Catholic University of Korea · University Hospital, Grenoble · University Hospital, Rouen · University of California, Los Angeles · University of Chicago · University of Cincinnati · University of Colorado, Denver · University of Giessen · University of Pittsburgh · VA Loma Linda Health Care System · Vanderbilt University · Wilhelminenspital Vienna

Regulatory milestones approvals, filings & regulatory actions · 3 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansion US (FDA) VENTAVIS 2005-08-24 fda.gov
Approved US (FDA) VENTAVIS 2004-12-29 fda.gov
Approved EU (EMA) Ventavis 2003-09-15 europa.eu

Trials 66 · started per year

today
EU approved 2003
US approved 2004
1
1
1
1
1
3
9
1
5
2
4
3
6
1
2
4
2
3
1
3
4
1
1
2
2
2
199619971998199920002001200220032004200520062007200820092010201120122013201420152016201720182019202020212022202320242025202620272028
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT01209533 Sep 2010 → Jul 2011 asthma Vanderbilt University Completed No outcome recorded
Phase 15 trials
Phase 1 NCT06429930 Apr 2025 → Jun 2026 overdue pulmonary arterial hypertension Pharmosa Biopharm Inc. Recruiting No outcome recorded
Phase 1 NCT02237183 Nov 2015 → Mar 2020 lung carcinoma National Cancer Institute (NCI) Completed No outcome recorded
Phase 1 NCT01274481 Mar 2011 → Jul 2012 acute lung injury, acute respiratory distress syndrome, pulmonary hypertension University of Oklahoma Completed No outcome recorded
Phase 1 NCT00708565 Jul → Oct 2008 pulmonary hypertension VA Loma Linda Health Care System Unknown No outcome recorded
Phase 1 NCT00724321 Jul → Nov 2008 Loma Linda University Withdrawn No outcome recorded
Phase 1/25 trials
Phase 1/2 NCT04543682 May 2022 → May 2024 Charite University, Berlin, Germany Unknown No outcome recorded
Phase 1/2 NCT02032836 Mar 2014 → Jan 2015 pulmonary arterial hypertension Bayer Completed No outcome recorded
Phase 1/2 NCT01179776 Sep 2010 → May 2011 myocardial infarction Thrombologic ApS Completed No outcome recorded
Phase 1/2 NCT01082484 Jan 2010 → Jan 2011 University Hospital, Grenoble Completed No outcome recorded
Phase 1/2 NCT00981591 Sep 2009 → Mar 2013 acute respiratory distress syndrome, congenital heart disease, neonatal respiratory failure, pulmonary hypertension, neonatal Seattle Children's Hospital Withdrawn No outcome recorded
Phase 218 trials
Phase 2 NCT05411107 Jun 2024 → Dec 2026 chronic obstructive pulmonary disease, lung carcinoma National Cancer Institute (NCI) Withdrawn No outcome recorded
Phase 2 NCT06319274 Apr 2024 → Sep 2027 expected acute respiratory failure, infectious disease Pär Johansson Recruiting No outcome recorded
Phase 2 NCT04420741 Jun 2020 → Feb 2021 COVID-19, respiratory failure Pär Johansson Completed No outcome recorded
Phase 2 NCT04445246 May 2020 → May 2021 COVID-19, acute respiratory distress syndrome Hamad Medical Corporation Completed No outcome recorded
Phase 2 NCT03903939 May 2019 → Nov 2021 multiple organ dysfunction syndrome Pär Johansson Completed No outcome recorded
Phase 2 NCT02685618 Feb → Aug 2016 cardiac arrest Pär Johansson Completed No outcome recorded
Phase 2 NCT02482402 Feb → Mar 2015 left ventricular failure, pulmonary hypertension Heidelberg University Withdrawn No outcome recorded
Phase 2 NCT02204852 Sep 2014 → Aug 2016 infectious disease with sepsis Sisse R. Ostrowski, MD PhD DMSc Completed No outcome recorded
Phase 2 NCT01941225 Sep 2013 → Nov 2016 chronic obstructive pulmonary disease Louisiana State University Health Sciences Center in New Orleans Completed No outcome recorded
Phase 2 NCT01774058 Oct 2012 → Jun 2019 arteriosclerosis disorder, peripheral arterial occlusive disease 1, peripheral neuropathy, type 2 diabetes mellitus Prim PD Dr Afshin Assadian Unknown No outcome recorded
Phase 2/34 trials
Phase 2/3 NCT04123444 Oct 2019 → Jun 2022 infectious disease with sepsis Jakob Stensballe, MD, PhD Completed No outcome recorded
Phase 2/3 NCT01310751 Jan 2011 → Dec 2013 pulmonary hypertension Shanghai Jiao Tong University School of Medicine Completed No outcome recorded
Phase 2/3 NCT00439543 Mar → Aug 2007 pulmonary fibrosis, pulmonary hypertension Interstitial Lung Disease Study Group, Korea Unknown No outcome recorded
Phase 2/3 NCT00345501 Nov 2005 → Jul 2007 chronic kidney disease Onassis Cardiac Surgery Centre Completed No outcome recorded
Phase 312 trials
Phase 3 NCT07498309 Sep 2026 → Mar 2030 expected sickle cell disease University Hospital, Rouen Not yet recruiting No outcome recorded
Phase 3 NCT03788837 Jul 2019 → Jan 2024 infectious disease with sepsis Assistance Publique - Hôpitaux de Paris Completed No outcome recorded
Phase 3 NCT01712997 Sep 2012 → Sep 2014 pulmonary arterial hypertension Air Force Military Medical University, China Unknown No outcome recorded
Phase 3 NCT01469169 Jun 2012 → Dec 2014 pulmonary arterial hypertension Bayer Completed No outcome recorded
Phase 3 NCT01598441 Jun 2012 → Nov 2016 pulmonary hypertension Shanghai Jiao Tong University School of Medicine Completed No outcome recorded
Phase 3 NCT00927654 Jun 2009 → Mar 2012 pulmonary hypertension Ludwig-Maximilians - University of Munich Completed No outcome recorded
Phase 3 NCT00709098 Sep 2008 → Jun 2010 pulmonary arterial hypertension Actelion Completed No outcome recorded
Phase 3 NCT00723554 Jul 2008 → Aug 2010 pulmonary arterial hypertension Actelion Terminated No outcome recorded
Phase 3 NCT00709956 Jul 2008 → Aug 2009 pulmonary arterial hypertension Actelion Completed No outcome recorded
Phase 3 NCT00302211 Feb 2006 → Dec 2007 pulmonary hypertension Actelion Terminated No outcome recorded
Phase 48 trials
Phase 4 NCT07713914 Jul 2026 → Jul 2028 expected pulmonary arterial hypertension University of Sao Paulo General Hospital Recruiting No outcome recorded
Phase 4 NCT03620526 Nov 2017 → Jan 2020 diastolic heart failure National Taiwan University Hospital Unknown No outcome recorded
Phase 4 NCT03044314 Jul 2017 → Jun 2019 pulmonary hypertension Duke University Terminated No outcome recorded
Phase 4 NCT01116063 May 2010 → Jan 2013 chronic obstructive pulmonary disease Carmel Medical Center Unknown No outcome recorded
Phase 4 NCT00409526 Dec 2006 → Dec 2007 pulmonary hypertension University of Chicago Terminated No outcome recorded
Phase 4 NCT01718288 Nov 2006 → Mar 2011 peripheral arterial disease Fadoi Foundation, Italy Completed No outcome recorded
Phase 4 NCT00403650 Nov 2006 → Jul 2008 pulmonary arterial hypertension, sarcoidosis University of Cincinnati Completed No outcome recorded
Phase 4 NCT02170519 Sep 2006 → Jan 2009 pulmonary hypertension Duke University Terminated No outcome recorded
Phase not applicable13 trials
NCT07263958 Dec 2025 → Jun 2026 overdue chronic obstructive pulmonary disease, pulmonary hypertension owing to lung disease and/or hypoxia University of Sao Paulo General Hospital Not yet recruiting No outcome recorded
NCT04927039 Jun 2021 → Jun 2023 Yonsei University Unknown No outcome recorded
NCT04598191 Nov 2020 → Dec 2022 coronary artery disorder Yonsei University Unknown No outcome recorded
NCT04583046 Nov 2020 → Sep 2025 lung cancer Yonsei University Completed No outcome recorded
NCT03936140 Jan → Oct 2018 lung cancer Seoul St. Mary's Hospital Completed No outcome recorded
NCT03365479 May 2017 → Aug 2018 pulmonary arterial hypertension University of Giessen Completed No outcome recorded
NCT03380325 May 2016 → Jun 2017 type 2 diabetes mellitus Amsterdam UMC, location VUmc Completed No outcome recorded
NCT02784899 Oct 2015 → Jun 2017 lung cancer Yonsei University Completed No outcome recorded
NCT02490657 Jul 2015 → May 2016 chronic obstructive pulmonary disease Yonsei University Completed No outcome recorded
NCT01319045 Jun 2011 → May 2013 Eisenmenger syndrome, congenital heart disease University of California, Los Angeles Terminated No outcome recorded
Also used as a comparator or background therapy in 8 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 24 trials
Phase 2 NCT03867097 Comparator Mar → Aug 2019 systemic sclerosis Civi Biopharma, Inc. Completed No outcome recorded
Phase 2 NCT02238535 Comparator Sep 2014 → Mar 2016 pulmonary hypertension Meshalkin Research Institute of Pathology of Circulation Unknown No outcome recorded
Phase 2 NCT01320878 Comparator Oct 2007 → Jul 2009 pulmonary hypertension Shanghai Jiao Tong University School of Medicine Completed No outcome recorded
Phase 2 NCT00622687 Comparator Sep 1997 → Dec 2003 systemic sclerosis Charite University, Berlin, Germany Terminated No outcome recorded
Phase 32 trials
Phase 3 NCT04040322 Comparator Oct 2019 → Jun 2021 Raynaud disease Civi Biopharma, Inc. Completed No outcome recorded
Phase 3 NCT03111212 Comparator Jun 2019 → May 2021 adult acute respiratory distress syndrome University Hospital Tuebingen Completed No outcome recorded
Phase 41 trial
Phase 4 NCT00120380 Comparator Sep 2004 → May 2006 hypertensive disorder Hannover Medical School Terminated No outcome recorded
Phase not applicable1 trial
NCT05204784 Comparator Feb 2022 → Dec 2023 Raynaud disease, chronic ulcer of skin, systemic sclerosis Peter Korsten Unknown No outcome recorded

Evidence & citations 14 cited values

Every value below carries the sentence it was read from. 75 sources stand behind the page.

FieldValueCited text
Known as Iloprost “Addition of a prostacyclin pathway agent (inhaled iloprost or oral selexipag) to ongoing dual therapy with an endothelin receptor antagonist and sildenafil as part of...” NCT07713914
70

“L608 is developed by Pharmosa Biopharm Inc. (PBI) as a new liposomal Iloprost formulation for inhalation use in the treatment of patients with WHO Group 1 PAH.” NCT06429930

“Standard of care treatment consists of intravenous iloprost infusions at a dose of 0.5-2 ng/kg/min administered over at least 6 hours as per local standard” NCT05204784

“3000 ng of iloprost (Ilomedin), diluted in 15ml saline solution, were injected into the common femoral artery.” NCT01774058

“20 µg/mL iloprost nebulizer solution, inhaled with FOX nebulizer” NCT02032836

NCT03867097

NCT02490657

NCT00709956

NCT00345501

NCT00235521

NCT00004786

NCT03788837

NCT01116063

NCT00439543

NCT00403650

NCT00302211

NCT02170519

NCT03620526

NCT00453414

NCT07263958

NCT03380325

NCT00185315

NCT02482402

NCT01320878

NCT01209533

NCT02204852

NCT03365479

NCT06319274

NCT00120380

NCT01712997

NCT03936140

NCT07498309

NCT00561223

NCT01598441

NCT00723554

NCT00981591

NCT04123444

NCT04040322

NCT00109681

NCT01437878

NCT04583046

NCT01319045

NCT03044314

NCT00709098

NCT02237183

NCT02685618

NCT02784899

NCT00409526

NCT04598191

NCT04543682

NCT01718288

NCT00724321

NCT00622687

NCT00084409

NCT05411107

NCT00414687

NCT01274481

NCT03111212

NCT01469169

NCT00467896

NCT04445246

NCT00708565

NCT04927039

NCT01082484

NCT00216931

NCT00086463

NCT01941225

NCT04420741

NCT03903939

NCT00927654

NCT01310751

Known as Aurlumyn ChEMBL registry synonym — accepted as the source's own label CHEMBL494
Known as BAYQ6252 “lloprost(Ventavis,BAYQ6252, 20 µg/mL)” NCT02032836
Known as BAYQ6256 “Iloprost (Ventavis inhaled, BAYQ6256)” NCT01469169
2

“Ventavis (Iloprost, BAYQ6256)” NCT00414687

“Ventavis (Iloprost, BAYQ6256)” NCT00185315

Known as Ciloprost ChEMBL registry synonym — accepted as the source's own label CHEMBL494
Known as Endoprost ChEMBL registry synonym — accepted as the source's own label CHEMBL494
Known as Ilomedin “3000 ng of iloprost (Ilomedin), diluted in 15ml saline solution, were injected into the common femoral artery.” NCT01774058
2

NCT01179776

NCT01532544

Known as Ventavis “Comparison of Nitric Oxide to Iloprost (Ventavis) for Treatment of Pulmonary Hypertension in Children After Cardiopulmonary Bypass Surgery” NCT00235521
14

Ventavis® is the commercial brand name for inhaled iloprost in Brazil.” NCT07263958

“2 inhalations per day of 2.5 µg Iloprost \[Ventavis®\] per inhalation” NCT02482402

“iloprost inhalation solution (Ventavis) (5 μg)” NCT00302211

“Iloprost 10μg of inhaled iloprost (Ventavis®)” NCT03936140

“20μg (2ml) of inhaled iloprost (Ventavis®)” NCT04927039

“20μg(2ml) of inhaled iloprost (Ventavis®)” NCT02784899

“BAYQ6256 (Iloprost; Ventavis) Inhalation” NCT02032836

“Iloprost Inhalation Solution (Ventavis)” NCT00453414

“Iloprost Inhalation Solution (Ventavis)” NCT00109681

“Iloprost (Ventavis inhaled, BAYQ6256)” NCT01469169

Ventavis (Iloprost, BAYQ6256)” NCT00414687

Ventavis (Iloprost, BAYQ6256)” NCT00185315

“Iloprost (Ventavis)” NCT00927654

NCT02238535

Known as ZK 00036374 ChEMBL registry synonym — accepted as the source's own label CHEMBL494
Known as ZK-36374 ChEMBL registry synonym — accepted as the source's own label CHEMBL494
Action Activate “trials of inhaled prostacyclin agonists such as iloprost for the treatment of asthma” NCT01209533
1

“Prostanoid IP receptor agonist” CHEMBL494

Modality Other / unclassified “oral iloprost, a prostacyclin analog” NCT00004786
Route Oral “Patients receive oral iloprost or placebo twice daily for 6 weeks.” NCT00004786
Target PTGIR “Prostanoid IP receptor agonist” CHEMBL494