Drugs / Aflibercept
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Aflibercept

Protein / enzyme biologic targets VEGFA via inhibition

Developed for
diabetic macular edema · wet macular degeneration · colorectal cancer · age-related macular degeneration · choroidal neovascularization · macular retinal edema · retinal vein occlusion · diabetic retinopathy
+101 more · cancer · macular degeneration · metastatic malignant neoplasm · proliferative diabetic retinopathy · central retinal vein occlusion with macular edema · occlusion of tributary of retinal vein · perifoveal exudative vascular anomalous complex · retinal vascular disorder · central retinal vein occlusion · neovascular glaucoma · rectal cancer · retinal detachment · neoplasm · ovarian cancer · retinopathy of prematurity · anaplastic astrocytoma · anaplastic oligodendroglioma · cancer of unknown primary site · central serous chorioretinopathy · colon mucinous adenocarcinoma · colon signet ring cell adenocarcinoma · corneal neovascularization · cutaneous melanoma · cystoid macular edema · fallopian tube cancer · giant cell glioblastoma · glaucoma · gliosarcoma · histoplasmosis retinitis · lymphoma · metastatic melanoma · non-small cell lung carcinoma · ovarian carcinoma · rectal signet ring cell adenocarcinoma · rectum mucinous adenocarcinoma · uveal melanoma · adult glioblastoma · atypical chronic myeloid leukemia, BCR-ABL1 negative · biliary tract cancer · bladder adenocarcinoma · bladder squamous cell carcinoma · bladder transitional cell carcinoma · breast cancer · breast carcinoma · carcinoid tumor · childhood malignant neoplasm · chronic myelomonocytic leukemia · colorectal carcinoma · colorectal neoplasm · degenerative myopia · endometrial carcinoma · esophageal cancer · euthyroid Graves orbitopathy · fibrolamellar hepatocellular carcinoma · gastric cancer · hemangioma of retina · iris melanoma · leiomyosarcoma · leukemia · lung neoplasm · macular telangiectasia type 1 · malignant epithelial tumor of ovary · medium/large size posterior uveal melanoma · metastasis from malignant tumor of colon · myelodysplastic syndrome · non-Hodgkin lymphoma · ocular melanoma with extraocular extension · ocular vascular disorder · optic choroid disorder · optic nerve disorder · ovarian carcinosarcoma · ovarian sarcoma · pancreatic endocrine carcinoma · pancreatic neoplasm · pancreatic neuroendocrine tumor · patterned macular dystrophy · peritoneum cancer · plasma cell myeloma · proliferative vitreoretinopathy · prostate cancer · pseudoxanthoma elasticum (inherited or acquired) · pterygium · rectosigmoid carcinoma · renal cell adenocarcinoma · renal cell carcinoma · renal pelvis/ureter urothelial carcinoma · retinal disorder · retinitis pigmentosa · rubeosis iridis · sarcoma · severe nonproliferative diabetic retinopathy · small cell lung carcinoma · thyroid gland follicular carcinoma · thyroid gland papillary carcinoma · urethra cancer · uterine carcinosarcoma · uterine corpus sarcoma · uveal disorder · age related macular degeneration 7 · partial retinal vein occlusion · radiation-induced disorder
Investigated by
Regeneron Pharmaceuticals · Bayer · Sanofi · National Cancer Institute (NCI) · Kim's Eye Hospital · Unity Health Toronto
+195 more · Greater Houston Retina Research · Jaeb Center for Health Research · Vitreous -Retina- Macula Consultants of New York · Adverum Biotechnologies, Inc. · Hospices Civils de Lyon · National Eye Institute (NEI) · Novartis Pharmaceuticals · Tennessee Retina · Duke University · Federation Francophone de Cancerologie Digestive · Fortrea · Hadassah Medical Organization · Instituto de Olhos de Goiania · Moorfields Eye Hospital NHS Foundation Trust · NSABP Foundation Inc · National Institutes of Health (NIH) · Northern California Retina Vitreous Associates · Ocular Therapeutix, Inc. · Poitiers University Hospital · Pusan National University Hospital · Qilu Pharmaceutical Co., Ltd. · Rafic Hariri University Hospital · Retina Research Institute, LLC · Rishi Singh · Singapore National Eye Centre · Southeast Retina Center, Georgia · Tanta University · University of Brescia · University of California, Los Angeles · University of California, San Diego · Valley Retina Institute · Yeungnam University College of Medicine · Zhongshan Ophthalmic Center, Sun Yat-sen University · AIO-Studien-gGmbH · Affiliated Traditional Chinese Medicine Hospital of Xinjiang Medical University · Ahmad Zeeshan Jamil · Al Hadi Hospital · Al-Azhar University · Al-Mustansiriyah University · Alcon Research · Alvotech Swiss AG · Amgen · Amin El Sayed Nawar · Amy C Schefler, MD · Asan Medical Center · Assign Data Management and Biostatistics GmbH · Augenabteilung Allgemeines Krankenhaus Linz · Azienda Ospedaliera Universitaria Policlinico Paolo Giaccone Palermo · Azienda USL Toscana Centro · Baghdad Medical City · Balamurali Ambati · Barcelona Macula Foundation · Barts & The London NHS Trust · Brown University · CMH Multan Institute of Medical Sciences · CR-CSSS Champlain-Charles-Le Moyne · Careggi University Hospital · Centre Hospitalier Intercommunal Creteil · Centre Hospitalier Universitaire Dijon · Centre Oscar Lambret · Chang Gung Memorial Hospital · Charles C Wykoff, PhD, MD · City of Hope Medical Center · Clearside Biomedical, Inc. · Clinical Trials Resource Group, LLC · Dana-Farber Cancer Institute · David M. Brown, M.D. · Department of Medical Services Ministry of Public Health of Thailand · Dongguan Guangming Ophthalmic Hospital · Edward Wood, MD · Emory University · European Organisation for Research and Treatment of Cancer - EORTC · Eye Associates of New Mexico · Federal University of São Paulo · all 201 on the full record

Regulatory milestones approvals, filings & regulatory actions · 12 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansions (2) US (FDA) EYLEA HD 2025-11-19 – 2026-04-02 fda.gov
Label expansions (7) US (FDA) EYLEA 2012-09-21 – 2023-02-08 fda.gov
Label expansion US (FDA) ZALTRAP 2015-09-17 fda.gov
Approved EU (EMA) Eylea 2012-11-21 europa.eu
Approved US (FDA) EYLEA 2011-11-18 fda.gov

Trials 274 · started per year

today
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EU approved 2012
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200220032004200520062007200820092010201120122013201420152016201720182019202020212022202320242025202620272028
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 03 trials
Phase 0 NCT06879301 Oct → Nov 2025 overdue choroidal neovascularization, diabetic macular edema, retinal vein occlusion Tanta University Not yet recruiting No outcome recorded
Phase 0 NCT06205979 Dec 2023 → Jun 2024 diabetic macular edema Sohag University Unknown No outcome recorded
Phase 0 NCT03766425 Jun 2017 → Jul 2019 glaucoma, optic nerve disorder Medical University of Lublin Completed No outcome recorded
Phase 128 trials
Phase 1 NCT03396861 Feb → Aug 2019 Tufts Medical Center Terminated No outcome recorded
Phase 1 NCT02403128 May 2015 → Feb 2020 macular retinal edema, retinal vascular disorder Kamal Kishore, MD Unknown No outcome recorded
Phase 1 NCT02298959 Apr 2015 → May 2025 overdue colorectal carcinoma, cutaneous melanoma, metastatic malignant neoplasm, metastatic melanoma +3 National Cancer Institute (NCI) Active not recruiting No outcome recorded
Phase 1 NCT02192541 Dec 2014 → Feb 2016 neoplasm National Cancer Institute (NCI) Terminated No outcome recorded
Phase 1 NCT02204683 Sep 2014 → Dec 2016 wet macular degeneration University of Nebraska Completed No outcome recorded
Phase 1 NCT02159989 Jun 2014 → Jun 2021 fibrolamellar hepatocellular carcinoma, metastatic malignant neoplasm, ovarian carcinoma, pancreatic neuroendocrine tumor National Cancer Institute (NCI) Completed No outcome recorded
Phase 1 NCT02173873 Jun 2014 → Sep 2016 age-related macular degeneration, central retinal vein occlusion Rafic Hariri University Hospital Unknown No outcome recorded
Phase 1 NCT01930552 Sep 2013 → Dec 2014 cancer Sanofi Completed No outcome recorded
Phase 1 NCT01843725 Sep 2013 → Oct 2016 biliary tract cancer, breast cancer, colorectal cancer, esophageal cancer +1 Jules Bordet Institute Completed No outcome recorded
Phase 1 NCT01868360 Jun 2013 → Oct 2015 corneal neovascularization Balamurali Ambati Terminated No outcome recorded
Phase 1/211 trials
Phase 1/2 NCT05769153 Dec 2023 → May 2027 expected wet macular degeneration Alcon Research Active not recruiting No outcome recorded
Phase 1/2 NCT04290195 Jun → Dec 2019 central retinal vein occlusion with macular edema Amin El Sayed Nawar Completed No outcome recorded
Phase 1/2 NCT03594461 Sep 2018 → Mar 2020 age-related macular degeneration Vitreous -Retina- Macula Consultants of New York Unknown No outcome recorded
Phase 1/2 NCT02797704 Mar 2017 → Sep 2019 corneal neovascularization Rabin Medical Center Terminated No outcome recorded
Phase 1/2 NCT02949024 Nov 2016 → Oct 2017 diabetic macular edema Clearside Biomedical, Inc. Completed No outcome recorded
Phase 1/2 NCT01955629 Dec 2013 → Mar 2015 colorectal cancer Sanofi Terminated No outcome recorded
Phase 1/2 NCT01790893 Mar 2013 → Aug 2014 histoplasmosis retinitis John Kitchens, MD Unknown No outcome recorded
Phase 1/2 NCT01724554 Nov 2012 → Oct 2014 central retinal vein occlusion, proliferative diabetic retinopathy Ophthalmic Consultants of Boston Completed No outcome recorded
Phase 1/2 NCT01661972 Aug 2012 → Jun 2016 colorectal cancer John Strickler, M.D. Completed No outcome recorded
Phase 1/2 NCT00794417 Nov 2008 → Jun 2011 non-small cell lung carcinoma Regeneron Pharmaceuticals Terminated No outcome recorded
Phase 278 trials
Phase 2 NCT06121180 Nov 2024 → Oct 2030 expected uveal melanoma H. Lee Moffitt Cancer Center and Research Institute Recruiting No outcome recorded
Phase 2 NCT06011798 Aug 2023 → Jan 2025 diabetes mellitus, diabetic macular edema, macular retinal edema Unity Biotechnology, Inc. Completed No outcome recorded
Phase 2 NCT04588948 Dec 2020 → Jun 2021 diabetic macular edema Stanford University Withdrawn No outcome recorded
Phase 2 NCT04311606 Nov 2020 → Dec 2024 euthyroid Graves orbitopathy Massachusetts Eye and Ear Infirmary Completed No outcome recorded
Phase 2 NCT04580147 Oct 2020 → Sep 2023 proliferative vitreoretinopathy, rhegmatogenous retinal detachment M. Ali Khan, MD Unknown No outcome recorded
Phase 2 NCT04418427 May 2020 → Nov 2022 diabetic macular edema Adverum Biotechnologies, Inc. Completed No outcome recorded
Phase 2 NCT03920878 May → Jun 2020 cataract, diabetic macular edema Emory University Withdrawn No outcome recorded
Phase 2 NCT04200248 Dec 2019 → Nov 2021 wet macular degeneration Ribomic USA Inc Completed No outcome recorded
Phase 2 NCT04126317 Nov 2019 → May 2021 wet macular degeneration Regeneron Pharmaceuticals Completed No outcome recorded
Phase 2 NCT03629210 Sep 2019 → Feb 2021 diabetic macular edema Pradeepa Yoganathan Withdrawn No outcome recorded
Phase 2/35 trials
Phase 2/3 NCT03143192 Mar 2017 → May 2019 diabetic macular edema Keyvan Koushan Completed No outcome recorded
Phase 2/3 NCT02772497 Jan → May 2016 diabetic macular edema Marashi Eye Clinic Completed No outcome recorded
Phase 2/3 NCT01813773 Mar 2013 → Apr 2016 proliferative diabetic retinopathy Ophthalmic Consultants of Long Island Completed No outcome recorded
Phase 2/3 NCT01646554 Dec 2012 → Dec 2015 metastasis from malignant tumor of colon European Organisation for Research and Treatment of Cancer - EORTC Withdrawn No outcome recorded
Phase 2/3 NCT00327444 Jul 2006 → Oct 2009 ovarian cancer Sanofi Completed No outcome recorded
Phase 353 trials
Phase 3 NCT07389980 Dec 2026 → Nov 2028 expected perifoveal exudative vascular anomalous complex Yeungnam University College of Medicine Recruiting No outcome recorded
Phase 3 NCT07482176 Mar 2026 → Nov 2027 expected wet macular degeneration Adverum Biotechnologies, Inc. Recruiting No outcome recorded
Phase 3 NCT06856577 Feb 2025 → Dec 2026 expected wet macular degeneration Adverum Biotechnologies, Inc. Active not recruiting No outcome recorded
Phase 3 NCT06495918 Nov 2024 → Jan 2027 expected wet macular degeneration Ocular Therapeutix, Inc. Active not recruiting No outcome recorded
Phase 3 NCT06491914 Jul 2024 → Aug 2025 overdue diabetic macular edema, wet macular degeneration Regeneron Pharmaceuticals Active not recruiting No outcome recorded
Phase 3 NCT06422507 May 2024 → Dec 2025 diabetic macular edema Bayer Completed No outcome recorded
Phase 3 NCT05989126 Apr → May 2024 diabetic macular edema, wet macular degeneration Regeneron Pharmaceuticals Completed No outcome recorded
Phase 3 NCT06223958 Jan 2024 → Apr 2026 overdue wet macular degeneration Ocular Therapeutix, Inc. Active not recruiting No outcome recorded
Phase 3 NCT05850520 May 2023 → Nov 2024 retinal vein occlusion Bayer Completed No outcome recorded
Phase 3 NCT05704725 Jan → Feb 2023 retinal vascular disorder Amgen Completed No outcome recorded
Phase 478 trials
Phase 4 NCT07612904 Jun 2026 → Jun 2028 expected diabetic macular edema The Third Peoples Hospital of Dalian Not yet recruiting No outcome recorded
Phase 4 NCT07438119 Mar 2026 → Sep 2027 expected diabetic macular edema Kun Liu Not yet recruiting No outcome recorded
Phase 4 NCT07365371 Jan 2026 → Dec 2027 expected perifoveal exudative vascular anomalous complex, wet macular degeneration Shanghai General Hospital, Shanghai Jiao Tong University School of Medicine Not yet recruiting No outcome recorded
Phase 4 NCT07301775 Jan → Jun 2026 overdue cataract, diabetic macular edema Ahmad Zeeshan Jamil Not yet recruiting No outcome recorded
Phase 4 NCT07118670 Dec 2025 → Feb 2028 expected proliferative diabetic retinopathy Edward Wood, MD Active not recruiting No outcome recorded
Phase 4 NCT06662994 Jul 2025 → Aug 2026 overdue diabetic macular edema Retina Consultants of Orange County Recruiting No outcome recorded
Phase 4 NCT06850571 Feb → Dec 2025 overdue diabetic retinopathy Al-Mustansiriyah University Recruiting No outcome recorded
Phase 4 NCT06683950 Oct 2024 → Jul 2026 age-related macular degeneration Kim's Eye Hospital Completed No outcome recorded
Phase 4 NCT06708637 Sep → Oct 2024 age-related macular degeneration, central retinal vein occlusion with macular edema, diabetic macular edema, occlusion of tributary of retinal vein Formycon AG Completed No outcome recorded
Phase 4 NCT06591598 Sep 2024 → Oct 2025 diabetic macular edema, wet macular degeneration Bayer Completed No outcome recorded
Phase not applicable17 trials
NCT07338097 Sep 2025 → Feb 2026 overdue diabetic macular edema CMH Multan Institute of Medical Sciences Enrolling by invitation No outcome recorded
NCT06610747 Oct 2024 → Apr 2027 expected diabetic macular edema Zhongshan Ophthalmic Center, Sun Yat-sen University Recruiting No outcome recorded
NCT04856397 May → Aug 2021 diabetic macular edema Uptown Eye Specialists Unknown No outcome recorded
NCT06391411 Mar 2021 → Mar 2022 age-related macular degeneration Careggi University Hospital Completed No outcome recorded
NCT06146309 Dec 2020 → Jul 2022 occlusion of tributary of retinal vein Al-Azhar University Completed No outcome recorded
NCT04970251 Nov 2018 → Mar 2021 neovascular glaucoma, ocular hypertension, perifoveal exudative vascular anomalous complex Siriraj Hospital Completed No outcome recorded
NCT02645266 May 2018 → Sep 2025 overdue diabetic macular edema McMaster University Active not recruiting No outcome recorded
NCT04075188 Sep 2017 → Jun 2018 choroidal neovascularization, optic choroid disorder Azienda Ospedaliera Universitaria Policlinico Paolo Giaccone Palermo Completed No outcome recorded
NCT03974425 Apr 2016 → Apr 2017 diabetic macular edema University of Alexandria Completed No outcome recorded
NCT03712670 Jan → Dec 2016 retinal disorder University of Brescia Completed No outcome recorded
Phase not stated1 trial
NCT01714115 hemangioma of retina Vitreous -Retina- Macula Consultants of New York No longer available No outcome recorded
Also used as a comparator or background therapy in 168 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT02457975 Background Jun 2015 → Aug 2019 diabetic retinopathy Medical College of Wisconsin Completed No outcome recorded
Phase 112 trials
Phase 1 NCT06817343 Background Sep 2024 → Feb 2029 expected wet macular degeneration Exegenesis Bio Active not recruiting No outcome recorded
Phase 1 NCT06132035 Comparator Dec 2023 → May 2025 overdue wet macular degeneration Caregen Co. Ltd. Recruiting No outcome recorded
Phase 1 NCT04919096 Comparator Apr → Sep 2022 wet macular degeneration Clover Biopharmaceuticals AUS Pty Withdrawn No outcome recorded
Phase 1 NCT04989699 Comparator Jul 2021 → Feb 2023 wet macular degeneration Ocular Therapeutix, Inc. Completed No outcome recorded
Phase 1 NCT05324592 Comparator Feb → Sep 2021 diabetic macular edema Mabwell (Shanghai) Bioscience Co., Ltd. Completed No outcome recorded
Phase 1/211 trials
Phase 1/2 NCT06672536 Comparator Nov 2024 → Sep 2026 expected wet macular degeneration Sinocelltech Ltd. Recruiting No outcome recorded
Phase 1/2 NCT06850922 Background Jun 2022 → May 2026 diabetic macular edema Genentech, Inc. Completed No outcome recorded
Phase 1/2 NCT05197270 Comparator Dec 2021 → Mar 2027 expected wet macular degeneration 4D Molecular Therapeutics Recruiting No outcome recorded
Phase 1/2 NCT05961007 Comparator Nov 2021 → Oct 2023 diabetic macular edema, wet macular degeneration Innovent Biologics (Suzhou) Co. Ltd. Suspended No outcome recorded
Phase 1/2 NCT04626128 Background Dec 2020 → Oct 2022 wet macular degeneration Clearside Biomedical, Inc. Completed No outcome recorded
Phase 240 trials
Phase 2 NCT07557121 Comparator Jul 2026 → Jun 2027 expected wet macular degeneration AiViva BioPharma, Inc. Not yet recruiting No outcome recorded
Phase 2 NCT07213570 Comparator Oct 2025 → Oct 2026 expected colorectal cancer National Cancer Institute, Naples Recruiting No outcome recorded
Phase 2 NCT07205887 Background Sep 2025 → Jun 2028 expected age-related macular degeneration, occlusion of tributary of retinal vein EyeBiotech Ltd. Recruiting No outcome recorded
Phase 2 NCT06942520 Comparator Mar 2025 → Dec 2027 expected diabetic macular edema Sierra Eye Associates Recruiting No outcome recorded
Phase 2 NCT06839339 Comparator Feb 2025 → Sep 2026 expected wet macular degeneration Beijing Anlong Biopharmaceutical Co., Ltd. Not yet recruiting No outcome recorded
Phase 2/38 trials
Phase 2/3 NCT07520318 Comparator Apr 2026 → Feb 2029 expected wet macular degeneration Shenzhen Oculgen Biomedical Technology Co., Ltd. Not yet recruiting No outcome recorded
Phase 2/3 NCT07496567 Comparator Apr 2026 → Jul 2028 expected choroidal neovascularization, wet macular degeneration EyeBiotech Ltd. Recruiting No outcome recorded
Phase 2/3 NCT07440225 Comparator Mar 2026 → Jun 2028 expected choroidal neovascularization, wet macular degeneration EyeBiotech Ltd. Recruiting No outcome recorded
Phase 2/3 NCT04429503 Comparator Jun 2020 → May 2022 diabetic macular edema, type 1 diabetes mellitus, type 2 diabetes mellitus Regeneron Pharmaceuticals Completed No outcome recorded
Phase 2/3 NCT04049266 Comparator Oct 2019 → Nov 2021 wet macular degeneration Kodiak Sciences Inc Terminated No outcome recorded
Phase 360 trials
Phase 3 NCT07705607 Comparator Sep 2026 → Nov 2028 expected diabetic macular edema Merck Sharp & Dohme LLC Not yet recruiting No outcome recorded
Phase 3 NCT07705555 Comparator Aug 2026 → Oct 2028 expected diabetic retinopathy, macular retinal edema Merck Sharp & Dohme LLC Not yet recruiting No outcome recorded
Phase 3 NCT07614776 Comparator May 2026 → Jul 2027 expected wet macular degeneration Amgen Recruiting No outcome recorded
Phase 3 NCT07489131 Comparator Apr 2026 → Jul 2027 expected diabetic macular edema Alvotech Swiss AG Recruiting No outcome recorded
Phase 3 NCT07489586 Comparator Mar → Dec 2026 expected wet macular degeneration Qilu Pharmaceutical Co., Ltd. Not yet recruiting No outcome recorded
Phase 424 trials
Phase 4 NCT05990829 Comparator Oct 2023 → Oct 2024 diabetic macular edema Tianjin Medical University Eye Hospital Unknown No outcome recorded
Phase 4 NCT05941715 Comparator Jul 2023 → Sep 2024 wet macular degeneration Medical University of Graz Completed No outcome recorded
Phase 4 NCT05710471 Comparator Jul 2022 → Jul 2023 age-related macular degeneration The University of Hong Kong Completed No outcome recorded
Phase 4 NCT05282420 Comparator Feb 2021 → Apr 2022 central retinal vein occlusion with macular edema South Valley University Unknown No outcome recorded
Phase 4 NCT04698850 Comparator Jan 2021 → Jan 2023 wet macular degeneration Faculty Hospital Kralovske Vinohrady Withdrawn No outcome recorded
Phase not applicable12 trials
NCT06929507 Comparator Mar 2025 → Mar 2026 overdue diabetic macular edema, impaired renal function disease, wet macular degeneration University Hospital, Alexandroupolis Recruiting No outcome recorded
NCT07096713 Comparator Jan → Jun 2024 Benha University Completed No outcome recorded
NCT04932980 Comparator May 2022 → Jun 2027 expected wet macular degeneration Berner Augenklinik Active not recruiting No outcome recorded
NCT04793100 Background Mar 2021 → Mar 2025 central retinal vein occlusion Fondation Ophtalmologique Adolphe de Rothschild Completed No outcome recorded
NCT03941587 Comparator Feb 2021 → Jun 2024 perifoveal exudative vascular anomalous complex Singapore National Eye Centre Completed No outcome recorded

Press releases naming this drug 54 releases

DateIssuerRelease
2026-04-02 Regeneron Pharmaceuticals EYLEA HD® (aflibercept) Approved by FDA as First and Only Injectable Anti-VEGF with Dosing Intervals Up to 5 Months for Wet Age-related Macular Degeneration (wAMD) and Diabetic Macular Edema (DME) regeneron.com
2026-02-02 Regeneron Pharmaceuticals EYLEA HD® (aflibercept) Injection 8 mg Presentations at Angiogenesis 2026 Underscore Strength of its Clinical Profile for the Treatment of Serious Retinal Diseases regeneron.com
2025-11-19 Regeneron Pharmaceuticals EYLEA HD® (aflibercept) Injection 8 mg Approved by FDA for the Treatment of Macular Edema Following Retinal Vein Occlusion (RVO) and for Monthly Dosing Across Approved Indications regeneron.com
2025-08-20 Regeneron Pharmaceuticals EYLEA HD® (aflibercept) Injection 8 mg Applications for Expanded U.S. Label and Prefilled Syringe Receive FDA Review Period Extension regeneron.com
2025-04-28 Regeneron Pharmaceuticals EYLEA HD® (aflibercept) Injection 8 mg Presentations at ARVO Reinforce Continued Safety and Efficacy and Highlight Early Real-World Outcomes for Patients with Serious Retinal Disease regeneron.com
2025-04-18 Regeneron Pharmaceuticals Regeneron Provides Update on EYLEA HD® (aflibercept) Injection 8 mg Supplemental Biologics License Application regeneron.com
2025-04-17 Regeneron Pharmaceuticals EYLEA HD® (aflibercept) Injection 8 mg sBLA Accepted for FDA Priority Review for Both the Treatment of Macular Edema Following Retinal Vein Occlusion (RVO) and for Monthly Dosing in Approved Indications regeneron.com
2025-02-08 Regeneron Pharmaceuticals Three-Year Results for EYLEA HD® (aflibercept) Injection 8 mg in Patients with Wet Age-related Macular Degeneration Demonstrate Continued Durable Vision Gains and Anatomic Improvements with Extended Dosing Intervals regeneron.com
2025-02-08 Regeneron Pharmaceuticals EYLEA HD® (aflibercept) Injection 8 mg Positive Phase 3 Results in Patients with Macular Edema following Retinal Vein Occlusion Presented at Angiogenesis Meeting regeneron.com
2025-01-13 Teva Branded Pharmaceutical Products R&D, Inc. Teva Announces Collaboration to Commercialize Formycon’s Biosimilar Candidate to Eylea® (aflibercept) in major parts of Europe and in Israel tevapharm.com
2025-01-13 Teva Branded Pharmaceutical Products R&D, Inc. Teva Announces Collaboration to Commercialize Formycon’s Biosimilar Candidate to Eylea® (aflibercept) in major parts of Europe and in Israel tevapharm.com
2024-12-17 Regeneron Pharmaceuticals EYLEA HD® (aflibercept) Injection 8 mg Phase 3 Trial Meets Primary Endpoint Showing Improved Vision with Extended Dosing Intervals in Patients with Macular Edema following Retinal Vein Occlusion regeneron.com

Evidence & citations 26 cited values

Every value below carries the sentence it was read from. 449 sources stand behind the page.

FieldValueCited text
Known as aflibercept “Threeintravitreous VEGF inhibitors - aflibercept (Eylea, Regeneron Pharmaceuticals), bevacizumab (Avastin, Genentech), and ranibizumab (Lucentis, Genentech) - are commonly used...” NCT02457975
380

“PURPOSE: To determine the maximum tolerated dose or maximal administered dose and pharmacokinetic and safety profiles of s.c. administered vascular endothelial growth factor...” PMID 20028764 Dec 2009

“Vascular endothelial growth factor (VEGF) Trap (aflibercept) is an angiogenesis inhibitor comprising portions of the extracellular domains of human VEGF receptors 1 and 2 fused...” PMID 19949018 Nov 2009

“Randomised, double-masked trial to compare the efficacy, safety and immunogenicity of the biosimilar aflibercept FYB203 with reference aflibercept in patients with neovascular...” PMID 41494750 Jan 2026

“COLLIDE is a multi-center, open-label, 1:1 randomized study looking at the effects of aflibercept (AFL; 2.0mg) plus OZURDEX (DEX; 0.7mg) implant combination therapy versus DEX...” NCT03629210

“Efficacy of Intravitreal Aflibercept Monotherapy for Submacular Hemorrhage Secondary to Neovascular Age-Related Macular Degeneration: A Prospective Clinical Trial” NCT03169660

“Anti-VEGFs including ranibizumab and biosimilars, aflibercept, faricimab, and brolucizumab will be used, as per the standard of care at participating sites.” NCT06985706

“Objective: To compare efficacy and safety of MYL-1701P, an aflibercept biosimilar, with reference aflibercept (Eylea [Regeneron]) in DME.” PMID 39264599 Oct 2024

“Outcome of Brolucizumab-dbll and Aflibercept Intravitreal Injection in the Treatment of Age-related Macular Neovascular Degeneration” NCT04882956

“Participants received 2mg Intravitreal aflibercept injection (IAI) (EYLEA, VEGF Trap-Eye, BAY86-5321) every 4 weeks (2Q4).” NCT01331681

Aflibercept 2 mg (0.05 ml) will be administered by intravitreal injection every month for three consecutive months.” NCT06845163

“Combination treatment may include: 5FU/LFA, capecitabine, oxaliplatin, irinotecan, bevacizumab, afliberceptNCT07213570

Aflibercept has been found to improve visual acuity and reduce macular thickness in pivotal trials.” NCT06416241

“Intravitreal injections of anti-VEGF (Aflibercept 2 mg, 0.05 ml) at a fixed regimen for six months” NCT06391411

“intravitreal injection of Anti-VEGF Aflibercept (Eylea®; manufactured in the United States)” NCT05282420

Aflibercept may stop the growth of cancer cells by blocking blood flow to the cancer.” NCT00601991

“intravitreal aflibercept for the treatment of center-involved diabetic macular edema” PMID 35422607 Apr 2022

“Arm 4 active comparator, aflibercept (2mg) as per US FDA Label, 50μL volume.” NCT07520318

“All patients will receive 2.0 mg intravitreal aflibercept injection.” NCT01495221

“This injection may be ranibizumab, bevacizumab, or aflibercept.” NCT02471651

“Eylea (Intravitreal Aflibercept, VEGF Trap-Eye, BAY86-5321)” NCT02581891

“Intravitreal Aflibercept Injection (EYLEA, VEGF Trap-Eye)” NCT00527423

“intravitreal ziv-aflibercept (aflibercept) injection” NCT03712904

“avastin,bevacizumab, eylea, aflibercept,” NCT02357342

“EYLEA (aflibercept) Injection” NCT01512966

“Eylea® (Aflibercept)” NCT04522167

“Eylea® (Aflibercept)” NCT05155293

“Eylea (Aflibercept)” NCT04450329

Aflibercept (Eylea)” NCT02348359

Aflibercept (Eylea)” NCT03585556

aflibercept (2mg)” NCT04626128

afliberceptNCT03630315

NCT02641457

NCT01909791

NCT07614776

NCT02307682

NCT02661711

NCT02129257

NCT02441907

NCT07612904

NCT02401945

NCT03006081

NCT03712670

NCT02403128

NCT07389980

NCT02645266

NCT01961414

NCT01521559

NCT02734407

NCT02540954

NCT00407654

NCT05324592

NCT02581995

NCT02441816

NCT02646670

NCT03630952

NCT04087746

NCT02624726

NCT02462889

NCT02418754

NCT01722656

NCT04592419

NCT03117634

NCT01926977

NCT06491914

NCT06929507

NCT02797704

NCT02045030

NCT06610747

NCT06850922

NCT02151695

NCT04004208

NCT04820452

NCT03085784

NCT01971190

NCT01882868

NCT05403749

NCT07205887

NCT00509795

NCT06330220

NCT02432547

NCT04810585

NCT02800642

NCT02559180

NCT06116890

NCT04079231

NCT02321267

NCT01958918

NCT01722045

NCT03804099

NCT06116916

NCT06099184

NCT02858076

NCT05324774

NCT04005352

NCT06879301

NCT03710564

NCT04153253

NCT01012973

NCT04200248

NCT04469595

NCT07557121

NCT02503540

NCT05885503

NCT04588948

NCT04126317

NCT07064759

NCT06683950

NCT04964089

NCT02130024

NCT02556229

NCT01578720

NCT06205979

NCT04411693

NCT02320474

NCT03999125

NCT04075188

NCT03802630

NCT03780361

NCT02204683

NCT04708145

NCT02258009

NCT04288232

NCT04989699

NCT04370379

NCT04707625

NCT03321513

NCT04707027

NCT04567550

NCT06856577

NCT02331927

NCT03709745

NCT04655482

NCT07317934

NCT00637377

NCT00644124

NCT05961007

NCT03043729

NCT03639675

NCT02309281

NCT01495208

NCT01543568

NCT06850571

NCT02181556

NCT04014556

NCT03386474

NCT04480463

NCT01724554

NCT02157077

NCT01657669

NCT03172299

NCT03405376

NCT04015180

NCT01988246

NCT01482910

NCT02092532

NCT05727397

NCT03468296

NCT01579760

NCT06011798

NCT01805297

NCT01652196

NCT01813773

NCT04757636

NCT06223958

NCT06683742

NCT00851084

NCT02949024

NCT02396316

NCT01969708

NCT03249740

NCT05662410

NCT03810313

NCT04527107

NCT03355638

NCT03845049

NCT03832179

NCT02788877

NCT06146309

NCT02303184

NCT00876044

NCT04331730

NCT02586727

NCT01148615

NCT01930552

NCT05251636

NCT02257632

NCT04603937

NCT03577899

NCT01940887

NCT04702048

NCT01746875

NCT03823300

NCT01363440

NCT04418427

NCT03823287

NCT01896284

NCT03126786

NCT01617148

NCT00532155

NCT01824225

NCT03264274

NCT01918878

NCT06132035

NCT02297204

NCT01627249

NCT00320788

NCT02495181

NCT02257502

NCT02630277

NCT06422507

NCT04919096

NCT05063734

NCT01646554

NCT03974425

NCT01783886

NCT00794417

NCT02033018

NCT02457026

NCT02863354

NCT01965041

NCT02860858

NCT07482176

NCT02120950

NCT01688960

NCT03056079

NCT01802684

NCT05710471

NCT03651011

NCT01773954

NCT04663750

NCT01669720

NCT00561470

NCT07365371

NCT05587062

NCT00964795

NCT03766425

NCT02392364

NCT03452527

NCT00545246

NCT04698850

NCT01857544

NCT00396591

NCT03453281

NCT02980874

NCT02072408

NCT05941715

NCT03481634

NCT03481660

NCT05126966

NCT02537054

NCT04423718

NCT04058067

NCT03186326

NCT01868360

NCT02689518

NCT06556368

NCT03866746

NCT04101721

NCT04932980

NCT02174211

NCT05275205

NCT04101877

NCT05972473

NCT01714115

NCT02681783

NCT05197270

NCT02976012

NCT00574275

NCT03917472

NCT06321302

NCT07338097

NCT07705555

NCT07705607

NCT02340949

NCT01796964

NCT04392479

NCT07449936

NCT02718326

NCT05407636

NCT02924987

NCT01749956

NCT01950741

NCT00921661

NCT07449923

NCT06668064

NCT00479076

NCT05990829

NCT06196840

NCT05704725

NCT02002377

NCT02633852

NCT03396861

NCT03397264

NCT01955629

NCT04580147

NCT00284141

NCT00437034

NCT03279289

NCT03953079

NCT02274259

NCT05345236

NCT05930561

NCT04113538

NCT02634333

NCT02173990

NCT04270747

NCT07489586

NCT02573038

NCT06662994

NCT06942520

NCT02651168

NCT07118670

NCT04049266

NCT03594461

NCT02118831

NCT01843725

NCT04611152

NCT05381948

NCT01571284

NCT06817343

NCT04740931

NCT05891548

NCT00327444

NCT05769153

NCT04740905

NCT02878681

NCT04047472

NCT03022292

NCT03767738

NCT00519285

NCT04311606

NCT00327171

NCT00789477

NCT04429503

NCT04970251

NCT03622580

NCT01870427

NCT02970916

NCT02299336

NCT06495918

NCT05473715

NCT02434328

NCT06591598

NCT02387957

NCT03941587

NCT05850520

NCT01711879

NCT06839339

NCT02296567

NCT04793100

NCT02384759

NCT02818998

NCT03622593

NCT07496567

NCT01871376

NCT02363621

NCT02713204

NCT02305238

NCT01670721

NCT07096713

NCT07301775

NCT03920878

NCT03059277

NCT02712008

NCT07440225

NCT01670162

NCT06864988

NCT05989126

NCT01661270

NCT03530267

NCT07438119

NCT02381730

NCT01790893

NCT02085005

NCT01997164

NCT05511038

NCT01710332

NCT04684394

NCT03531294

NCT03197480

Known as AFL “EYLEA® (AFL 2.0 mg intravitreal injections) is an anti-VEGF treatment.” NCT03629210
Known as AFLB “Aflibercept (AFLB) 2 mg IVT” NCT06864988
1

“Aflibercept (AFLB) 2 mg IVT” NCT07064759

Known as Aflibercept (Eylea) Aflibercept (Eylea)NCT06845163
2

Aflibercept (Eylea)NCT03585556

Aflibercept (Eylea)NCT02348359

Known as aflibercept HD “Eylea HD (aflibercept HD)” NCT07489131
Known as Alflibercept ClinicalTrials.gov intervention name — accepted as the source's own label NCT03340610
Known as AVE0005 “To determine the overall objective response rate (ORR) of AVE0005 (ziv-aflibercept, aflibercept, VEGF trap, ZALTRAP®) 4.0 mg/kg intravenously (IV) every 2 weeks in participants...” NCT00284141
15

“A Phase I Open-label Dose-escalation Study of Intravenous Aflibercept (AVE0005, VEGF Trap) in Combination With R-CHOP Administered Every 2 Weeks or Every 3 Weeks in Patients...” NCT00644124

“Drug: Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00532155

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00574275

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00327171

“aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00327444

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00396591

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00561470

“Drug: aflibercept (AVE0005)” NCT00545246

“aflibercept (AVE0005)” NCT00479076

AVE0005 (aflibercept)” NCT00921661

“aflibercept (AVE0005)” NCT00876044

“Aflibercept (AVE0005)” NCT01148615

“AFLIBERCEPT AVE0005NCT01571284

“Aflibercept AVE0005NCT01930552

“Aflibercept AVE0005NCT01955629

Known as BAY86-5321 “The study treatment Aflibercept (also called BAY 86-5321) is a drug that blocks a protein called vascular endothelial growth factor (VEGF) which causes abnormal growth and...” NCT06591598
25

“Participants received 2mg Intravitreal aflibercept injection (IAI) (EYLEA, VEGF Trap-Eye, BAY86-5321) every 4 weeks (2Q4).” NCT01331681

“The study treatment intravitreal aflibercept (also called BAY865321) is injected into the eye.” NCT05473715

“Intravitreal Aflibercept Injection (IAI; EYLEA®; BAY86-5321)” NCT01363440

“Eylea (Intravitreal Aflibercept, VEGF Trap-Eye, BAY86-5321)” NCT02581891

“Intravitreal Aflibercept Injection (IAI;EYLEA®;BAY86-5321)” NCT01521559

“Aflibercept, VEGF Trap-Eye(Eylea, BAY86-5321)_higher dose” NCT05850520

“Aflibercept Injection (EYLEA, VEGF Trap-Eye, BAY86-5321)” NCT00637377

“Aflibercept Injection (EYLEA, VEGF Trap-Eye, BAY86-5321)” NCT01012973

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02305238

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT05511038

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT01783886

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02818998

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT01482910

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02120950

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02540954

“Eylea (Aflibercept, VEGF Trap-Eye, BAY86-5321)” NCT02581995

“Aflibercept VEGF Trap-Eye (Eylea, BAY86-5321)” NCT04423718

“Aflibercept 8 mg (VEGF Trap-Eye, BAY86-5321)” NCT06662994

“2 mg aflibercept (EYLEA, BAY 86-5321)” NCT06422507

“Aflibercept (Eylea, BAY 86-5321)” NCT02396316

“Aflibercept (EYLEA, BAY86-5321)” NCT03639675

“Eylea (Aflibercept, BAY86-5321)” NCT04015180

“Aflibercept (Eylea, BAY86-5321)” NCT02800642

“Eylea (Aflibercept, BAY86-5321)” NCT04004208

“VEGF Trap-Eye (BAY86-5321)” NCT01249664

Known as Eylea “Threeintravitreous VEGF inhibitors - aflibercept (Eylea, Regeneron Pharmaceuticals), bevacizumab (Avastin, Genentech), and ranibizumab (Lucentis, Genentech) - are commonly used...” NCT02457975
87

“A 24 Month Phase 2A Open Label Safety Study of Fovista® (Anti-PDGF-BB Pegylated Aptamer) Regiment Administered in Combination With Avastin®, Eylea®, or Lucentis®) During the...” NCT02214628

“InCNV is treated at the moment with off-label anti-VEGF (Vascular Endothelial Growth Factor) therapy and could also benefit from aflibercept (EYLEA), a new anti-VEGF currently...” NCT02556229

“Each eye will receive three to five q4week loading anti-VEGF injections of aflibercept (2-mg, EYLEA®) after enrollment to complete the initial loading phase of 5 doses.” NCT06610747

“The purpose of this study is to compare the safety and efficacy of intravitreal Eylea injections at a set interval, versus a variable dosing schedule” NCT02392364

“The included patients received 5 loading doses of intravitreal Aflibercept (2.0 mg/0.05 mL) (Eylea; Bayer, Berlin, Germany) given monthly.” NCT03974425

“Subjects will receive monthly intravitreous injections of Avacincaptad Pegol in combination with Lucentis, Avastin or Eylea.” NCT02397954

“Participants received 2mg Intravitreal aflibercept injection (IAI) (EYLEA, VEGF Trap-Eye, BAY86-5321) every 4 weeks (2Q4).” NCT01331681

“Effect of Aflibercept (Eylea®) in the Management of Bevacizumab (Avastin®) Resistant Diabetic Macular Edema” NCT02924987

“Biological: Aflibercept IVT * Commercially available Active Comparator * Other Names: EyleaNCT06942520

“intravitreal injection of Anti-VEGF Aflibercept (Eylea®; manufactured in the United States)” NCT05282420

“Aflibercept (trade name: Eylea®/EYLEA®) is an anti-VEGF drug developed by Regeneron/Bayer.” NCT05324774

“could also benefit from aflibercept (EYLEA), a new anti-VEGF currently indicated in AMD.” NCT02573038

“2mg intravitreal Aflibercept(Eylea) injection at baseline, at 1 month, and at 2 month” NCT01971190

“Patient will receiver Eylea® (Aflibercept) intravitreal injection once in a month” NCT06132035

“2.0 mg/0.05 mL of aflibercept (Eylea) is injected into the vitreous cavity” NCT03804099

“A comparator drug, Eylea® (aflibercept), will also be used in this study.” NCT07520318

“Efficacy of Aflibercept (Eylea®) on Choroidal Neovascularization (Type 3)” NCT02320474

EYLEA® (AFL 2.0 mg intravitreal injections) is an anti-VEGF treatment.” NCT03629210

“Intravitreal Aflibercept Injection (IAI; EYLEA®; BAY86-5321)” NCT01363440

“Intravitreal Aflibercept Injection (IAI;EYLEA®;BAY86-5321)” NCT01521559

“Aflibercept, VEGF Trap-Eye(Eylea, BAY86-5321)_higher dose” NCT05850520

“Intravitreal Aflibercept Injection (EYLEA, VEGF Trap-Eye)” NCT00527423

“Aflibercept Injection (EYLEA, VEGF Trap-Eye, BAY86-5321)” NCT00637377

“Aflibercept 2 mg/0.05 mL (Eylea; Bayer, Berlin, Germany)” NCT04014556

“Aflibercept Injection (EYLEA, VEGF Trap-Eye, BAY86-5321)” NCT01012973

Eylea® (Aflibercept, 114.3 mg/mL, 8 mg Per 70 μL)” NCT07489586

“administration of anti-VEGF Aflibercept (Eylea)” NCT04932980

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02818998

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02305238

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT01783886

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT05511038

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02120950

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT01482910

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02540954

Eylea (Aflibercept, VEGF Trap-Eye, BAY86-5321)” NCT02581995

“Aflibercept VEGF Trap-Eye (Eylea, BAY86-5321)” NCT04423718

“a drug called aflibercept (also called EYLEA)” NCT01773954

“intravitreal injection of aflibercept (EYLEA)” NCT02257502

EYLEA® (aflibercept) Injection 2 mg (0.05mL)” NCT06864988

EYLEA® (aflibercept) Injection 2 mg (0.05mL)” NCT05275205

EYLEA® (aflibercept) Injection 2 mg (0.05mL)” NCT07064759

EYLEA® (aflibercept) Injection 2 mg (0.05mL)” NCT07557121

EYLEA (Aflibercept) intravitreal injection” NCT01578720

“Drug: Aflibercept (BAY86-5321, Eylea)” NCT06591598

“2 mg aflibercept (EYLEA, BAY 86-5321)” NCT06422507

“Drug: Aflibercept Injection [Eylea]” NCT04288232

“Drug: Aflibercept Injection [Eylea]” NCT06330220

“Aflibercept (Eylea, BAY 86-5321)” NCT02396316

Eylea (Aflibercept, BAY86-5321)” NCT04015180

“Aflibercept (EYLEA, BAY86-5321)” NCT03639675

“Aflibercept (Eylea, BAY86-5321)” NCT02800642

Eylea (Aflibercept, BAY86-5321)” NCT04004208

“Aflibercept(BAY86-5321, Eylea)” NCT05473715

“Aflibercept (Eylea®) - US only” NCT06321302

EYLEA (aflibercept) Injection” NCT01512966

“Aflibercept Injection [Eylea]” NCT03453281

“Aflibercept Injection [Eylea]” NCT03197480

“Aflibercept Injection [Eylea]” NCT03355638

“Aflibercept Injection [Eylea]” NCT03651011

“Aflibercept Injection [Eylea]” NCT06205979

“Aflibercept Injection [Eylea]” NCT04153253

“Aflibercept Injection [Eylea]” NCT02645266

“Aflibercept Injection [Eylea]” NCT03845049

“Aflibercept (Eylea®)” NCT02646670

“Aflibercept (Eylea)” NCT07301775

“Aflibercept (EYLEA)” NCT01918878

Eylea®” NCT02418754

NCT02732899

NCT02581891

NCT01414153

NCT06672536

NCT06470373

NCT03610646

NCT05155293

NCT04856397

NCT04864834

NCT04450329

NCT05571267

NCT04572698

NCT04058535

NCT03374670

NCT02591914

NCT02228304

NCT02142296

NCT04522167

NCT04739306

NCT03984110

Known as EYLEA (aflibercept) Injection “EYLEA® (aflibercept) Injection” NCT02713204
2

“EYLEA® (aflibercept) Injection” NCT02712008

“EYLEA® (aflibercept) Injection” NCT02718326

Known as Eylea HD ClinicalTrials.gov intervention name — accepted as the source's own label NCT07489131
Known as Eylea is the brand name. Eylea is the brand name.NCT02142296
Known as FYB203 ClinicalTrials.gov intervention name — accepted as the source's own label NCT06708637
1

NCT04522167

Known as IAI “The purpose of this study is to evaluate the safety and efficacy of intravitreal aflibercept injection (IAI) in patients with neovascular polypoidal choroidal vasculopathy.” NCT02092532
3

“Intravitreal Aflibercept Injection (IAI;EYLEA®;BAY86-5321)” NCT01521559

“Intravitreal Aflibercept Injection (IAI)” NCT02713204

“Intravitreal Aflibercept Injection (IAI)” NCT01722045

Known as IVT-AFL “The VEGA trial assessed the efficacy and safety of intravitreal aflibercept (IVT-AFL) in patients with neovascular glaucoma in a 13-week, randomized, double-masked,...” PMID 33330958 Dec 2020
1

“intravitreal aflibercept (IVT-AFL)” PMID 33556381 Feb 2021

Known as REGN3 “Co-formulation for intravitreal (IVT) injection consisting of REGN910 (nesvacumab) and REGN3 (aflibercept)” NCT02712008
1

“Intravitreal injection of REGN2176-3 (REGN2176 1 mg and REGN3 2 mg) every 4 weeks for 12 weeks.” NCT02418754

Known as vascular endothelial growth factor (VEGF) Trap “Aflibercept, also known as vascular endothelial growth factor (VEGF) Trap, is an angiogenesis inhibitor with a unique mechanism of action.” NCT02624726
Known as VEGF Trap “Vascular endothelial growth factor (VEGF) Trap (aflibercept) is an angiogenesis inhibitor comprising portions of the extracellular domains of human VEGF receptors 1 and 2 fused...” PMID 19949018 Nov 2009
5

“A Phase I Open-label Dose-escalation Study of Intravenous Aflibercept (AVE0005, VEGF Trap) in Combination With R-CHOP Administered Every 2 Weeks or Every 3 Weeks in Patients...” NCT00644124

“An Exploratory Study of the Safety, Tolerability and Biological Effect of a Single Intravitreal Administration of VEGF Trap in Patients With Diabetic Macular Edema” NCT00320814

“Aflibercept (VEGF Trap) Recombinant human protein, at 25 mg/ml Dose : 4 mg/Kg -Day 1, q2w Route of administration: Intravenous (60 min infusion)” NCT01802684

NCT00383370

NCT00320775

Known as VEGF Trap-Eye “Participants received 2mg Intravitreal aflibercept injection (IAI) (EYLEA, VEGF Trap-Eye, BAY86-5321) every 4 weeks (2Q4).” NCT01331681
21

“intravitreal aflibercept injection (VEGF Trap-Eye; Regeneron, Tarrytown, NY, and Bayer HealthCare, Berlin, Germany)” PMID 23084240 Oct 2012

“Eylea (Intravitreal Aflibercept, VEGF Trap-Eye, BAY86-5321)” NCT02581891

“Aflibercept, VEGF Trap-Eye(Eylea, BAY86-5321)_higher dose” NCT05850520

“Intravitreal Aflibercept Injection (EYLEA, VEGF Trap-Eye)” NCT00527423

“Aflibercept Injection (EYLEA, VEGF Trap-Eye, BAY86-5321)” NCT00637377

“Aflibercept Injection (EYLEA, VEGF Trap-Eye, BAY86-5321)” NCT01012973

VEGF Trap-Eye (Intravitreal Aflibercept Injection [IAI])” NCT01521559

VEGF Trap-Eye (Intravitreal Aflibercept Injection)” NCT01722045

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02305238

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02818998

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT05511038

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT01783886

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT01482910

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02120950

“Aflibercept (Eylea, VEGF Trap-Eye, BAY86-5321)” NCT02540954

“Eylea (Aflibercept, VEGF Trap-Eye, BAY86-5321)” NCT02581995

“Aflibercept VEGF Trap-Eye (Eylea, BAY86-5321)” NCT04423718

“Aflibercept 8 mg (VEGF Trap-Eye, BAY86-5321)” NCT06662994

NCT01249664

NCT00943072

NCT00320814

Known as ZALTRAP “To determine the overall objective response rate (ORR) of AVE0005 (ziv-aflibercept, aflibercept, VEGF trap, ZALTRAP®) 4.0 mg/kg intravenously (IV) every 2 weeks in participants...” NCT00284141
9

“Ziv-aflibercept (Zaltrap, Regeneron) is a recombinant fusion protein that acts as a soluble decoy receptor” NCT02590094

“aflibercept(Zaltrap): 4 mg/kg IV infusion for over 1hr (Do not administer as an IV push or bolus)” NCT04810585

“Drug: Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00532155

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00327171

“aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00327444

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00396591

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00561470

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00574275

“Drug: Ziv-Aflibercept 25 MG/ML [Zaltrap]” NCT03423823

Known as Zhuochuming “Aflibercept Intravitreal Injection (Zhuochuming®)” NCT07612904
Known as ziv-aflibercept “To determine the overall objective response rate (ORR) of AVE0005 (ziv-aflibercept, aflibercept, VEGF trap, ZALTRAP®) 4.0 mg/kg intravenously (IV) every 2 weeks in participants...” NCT00284141
48

“The MTD and RPTD were: capecitabine 850 mg/m2, P.O. bid, days 1-14, and ziv-aflibercept 6 mg/kg I.V., day 1, of each 21-day cycle.” PMID 31675952 Nov 2019

“* Ziv-aflibercept: will be administered 4 mg/kg IV on Day 1 of each cycle, repeating every 14 days.” NCT02079220

“Patients receive a higher dose of ziv-aflibercept (VEGF Trap) IV over 1 hour on day 1.” NCT00357760

“Drug: Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00532155

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00561470

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00574275

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00327171

“aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00327444

“Aflibercept (ziv-aflibercept, AVE0005, VEGF trap, ZALTRAP®)” NCT00396591

“In the US, the US proper name is "ziv-aflibercept".” NCT02085005

“aflibercept (ziv-aflibercept)” NCT01688960

“Intravitreal ziv-AfliberceptNCT03660345

NCT03712904

NCT02556723

NCT00369590

NCT02645734

NCT00462826

NCT00509249

NCT00650923

NCT00083213

NCT00045266

NCT00407485

NCT03423823

NCT04290195

NCT00390234

NCT01889680

NCT02235324

NCT00828139

NCT00082823

NCT01747551

NCT02101918

NCT01782443

NCT01941173

NCT01258855

NCT00036946

NCT00622414

NCT02192541

NCT02298959

NCT02159989

NCT02590094

NCT00369655

NCT00729157

NCT06121180

NCT02173873

NCT00436501

NCT00450255

NCT02486484

NCT02772497

Action Inhibit “Evaluate the ability of this drug to bind and inactivate circulating vascular endothelial growth factor (VEGF) in these patients.” NCT00036946
Modality Protein / enzyme biologic “comprising portions of the extracellular domains of human VEGF receptors 1 and 2 fused to the Fc portion of human immunoglobulin G” PMID 19949018 Nov 2009
Route Subcutaneous “aflibercept administered subcutaneously to patients with advanced solid tumors.” PMID 20028764 Dec 2009