Drugs / Mesalamine
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Mesalamine

Small molecule

Developed for
ulcerative colitis · irritable bowel syndrome · Crohn disease · diverticulitis · diarrheal disease · proctitis · colitis · colorectal cancer
+16 more · HIV infectious disease · chronic beryllium disease · collagenous colitis · colonic neoplasm · colorectal adenoma · eosinophilic esophagitis · large intestine disorder · lymphocytic colitis · Lynch syndrome · microscopic colitis · protein-energy malnutrition · ulcer of anus and rectum · ulcerative stomatitis · colonic disorder · inflammatory bowel disease · solitary rectal ulcer syndrome
Investigated by
Shire · Dr. Falk Pharma GmbH · Ferring Pharmaceuticals · Warner Chilcott · Tillotts Pharma AG · Bausch Health Americas, Inc.
+68 more · Procter and Gamble · Holy Stone Healthcare Co., Ltd · National Institute of Allergy and Infectious Diseases (NIAID) · National Institute of Diabetes and Digestive and Kidney Diseases (NIDDK) · SOFAR S.p.A. · AHS Cancer Control Alberta · AIDS Healthcare Foundation · AbbVie · Alimenta AB · Ann-Sofie Backman · Ann-Sofie Backman, MD PhD, Sweden · Annette Langseder · Azienda Policlinico Umberto I · California HIV/AIDS Research Program · Cardiff and Vale University Health Board · Christoph Gasche · Connecticut Children's Medical Center · Edward V. Loftus MD · Endeavor Health · Faes Farma, S.A. · Food and Drug Administration (FDA) · Forest Laboratories · Grupo Espanol de Trabajo en Enfermedad de Crohn y Colitis Ulcerosa · HIV Immunotherapeutics Institute · Hans Törnblom · Haukeland University Hospital · Imperial College London · Innlandet Hospital Trust · James Lewis · Karolinska Institutet · Karolinska University Hospital · Kelsey Jones · Mayo Clinic · National Institute for Health Research, United Kingdom · National Jewish Health · Oslo University Hospital · Otsuka Pharmaceutical Development & Commercialization, Inc. · Paul E. Evans MD · Prof. Dr. Gabriela Möslein, Germany · Prof. Dr. Hans Vasen, The Netherlands · Prof. Dr. med. Jan Lubinski, Poland · Prof. Dr. med. Yaron Niv, Israel · Sahlgrenska University Hospital · Sandoz · Shiraz University of Medical Sciences · Shire Human Genetic Therapies, Inc. · Sixth Affiliated Hospital, Sun Yat-sen University · Smerud Medical Research International AS · Tehran University of Medical Sciences · Teva Pharmaceuticals USA · The Second Hospital of Nanjing Medical University · The Swedish Research Council · Thomas C. Smryk MD · UMC Utrecht · Univ. Prof. Dr. Judith Karner-Hanusch, Austria · University Hospital of Saint-Etienne · University of California, San Francisco · University of Chicago · University of Michigan · University of Nottingham · University of Utah · Willaim Tremaine MD · William J. Sandborn MD · Wolfson Medical Center · Xijing Hospital of Digestive Diseases · Zeria Pharmaceutical · Zhu Weiming · inVentiv Health Clinical

Regulatory milestones approvals, filings & regulatory actions · 10 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Label expansions (2) US (FDA) LIALDA 2011-07-14 – 2020-06-26 fda.gov
Label expansions (2) US (FDA) CANASA 2004-11-05 – 2016-09-02 fda.gov
Label expansions (2) US (FDA) DELZICOL 2014-04-28 – 2015-09-09 fda.gov
Label expansions (3) US (FDA) ASACOL 1997-08-19 – 2015-05-27 fda.gov
Approved US (FDA) ROWASA 1987-12-24 fda.gov

Trials 88 · started per year

today
US approved 1987
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198719881989199019911992199319941995199619971998199920002001200220032004200520062007200820092010201120122013201420152016201720182019202020212022202320242025202620272028
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 115 trials
Phase 1 NCT03327558 May → Jun 2017 ulcerative colitis Bausch Health Americas, Inc. Completed No outcome recorded
Phase 1 NCT02196662 Jul 2014 → Apr 2015 Holy Stone Healthcare Co., Ltd Completed No outcome recorded
Phase 1 NCT02125292 Jun 2014 Shire Completed No outcome recorded
Phase 1 NCT02306785 Oct 2012 → Feb 2013 ulcerative colitis Tillotts Pharma AG Completed No outcome recorded
Phase 1 NCT02306772 Dec 2011 → Feb 2012 ulcerative colitis Tillotts Pharma AG Completed No outcome recorded
Phase 1 NCT01469637 Nov → Dec 2011 Shire Completed No outcome recorded
Phase 1 NCT01442688 Oct → Nov 2011 Shire Completed No outcome recorded
Phase 1 NCT01418365 Aug → Oct 2011 Shire Completed No outcome recorded
Phase 1 NCT01402947 Jul → Aug 2011 Shire Completed No outcome recorded
Phase 1 NCT01130844 Oct 2010 → Jun 2013 ulcerative colitis Shire Completed No outcome recorded
Phase 1/24 trials
Phase 1/2 NCT05091775 Jun → Aug 2020 diarrheal disease, ulcer of anus and rectum Shiraz University of Medical Sciences Completed No outcome recorded
Phase 1/2 NCT03399903 May 2017 → Mar 2019 HIV infectious disease, colitis AIDS Healthcare Foundation Completed No outcome recorded
Phase 1/2 NCT01841099 Jun 2013 → May 2014 protein-energy malnutrition Kelsey Jones Completed No outcome recorded
Phase 1/2 NCT01088243 Mar 2010 → Mar 2015 chronic beryllium disease National Jewish Health Completed No outcome recorded
Phase 214 trials
Phase 2 NCT05663775 Aug 2024 → Aug 2026 overdue diarrheal disease, melanoma, rectal carcinoma AHS Cancer Control Alberta Recruiting No outcome recorded
Phase 2 NCT05488405 Feb → Jun 2023 eosinophilic esophagitis Dr. Falk Pharma GmbH Completed No outcome recorded
Phase 2 NCT04920149 Mar 2022 → Sep 2032 expected Lynch syndrome, colonic neoplasm Ann-Sofie Backman Recruiting No outcome recorded
Phase 2 NCT03070574 Nov 2017 → Apr 2019 colorectal cancer Christoph Gasche Terminated No outcome recorded
Phase 2 NCT02493712 Jan 2016 → Jul 2018 ulcerative colitis Holy Stone Healthcare Co., Ltd Completed No outcome recorded
Phase 2 NCT01966783 Sep 2013 → Aug 2015 proctitis Dr. Falk Pharma GmbH Completed No outcome recorded
Phase 2 NCT04032652 Dec 2012 → Nov 2014 ulcerative colitis Endeavor Health Terminated No outcome recorded
Phase 2 NCT02077777 Oct 2012 → Jun 2016 colorectal cancer SOFAR S.p.A. Completed No outcome recorded
Phase 2 NCT01894685 Jul 2012 → Jun 2015 colorectal adenoma UMC Utrecht Completed No outcome recorded
Phase 2 NCT01699438 Apr 2012 → Dec 2016 irritable bowel syndrome Hans Törnblom Completed No outcome recorded
Phase 2/32 trials
Phase 2/3 NCT02044952 Jan 2014 → May 2016 Crohn disease Zhu Weiming Unknown No outcome recorded
Phase 2/3 NCT00952952 Feb → Nov 2007 diarrheal disease, microscopic colitis Mayo Clinic Completed No outcome recorded
Phase 339 trials
Phase 3 NCT05316220 Sep 2025 → Jul 2026 ulcerative colitis AbbVie Withdrawn No outcome recorded
Phase 3 NCT06176560 Mar 2024 → Aug 2025 ulcerative colitis Faes Farma, S.A. Unknown No outcome recorded
Phase 3 NCT02665845 Jun 2016 → May 2021 ulcerative colitis University Hospital of Saint-Etienne Completed No outcome recorded
Phase 3 NCT02769494 Mar → Dec 2016 Crohn disease, ulcerative stomatitis Xijing Hospital of Digestive Diseases Withdrawn No outcome recorded
Phase 3 NCT02522780 Feb 2016 → Sep 2018 ulcerative colitis Ferring Pharmaceuticals Completed No outcome recorded
Phase 3 NCT02522767 Oct 2015 → Feb 2018 ulcerative colitis Ferring Pharmaceuticals Completed No outcome recorded
Phase 3 NCT02368717 Mar 2015 → Jan 2017 ulcerative colitis Ferring Pharmaceuticals Completed No outcome recorded
Phase 3 NCT02093663 Dec 2014 → Nov 2018 ulcerative colitis Shire Completed No outcome recorded
Phase 3 NCT01745770 Jan 2013 → Mar 2015 ulcerative colitis Dr. Falk Pharma GmbH Completed No outcome recorded
Phase 3 NCT01257399 Nov 2010 → Jan 2013 ulcerative colitis Tillotts Pharma AG Completed No outcome recorded
Phase 411 trials
Phase 4 NCT07248644 May → Sep 2026 expected ulcerative colitis Grupo Espanol de Trabajo en Enfermedad de Crohn y Colitis Ulcerosa Not yet recruiting No outcome recorded
Phase 4 NCT05205603 Jan 2022 → Jan 2024 ulcerative colitis Sixth Affiliated Hospital, Sun Yat-sen University Completed No outcome recorded
Phase 4 NCT02190526 Sep 2014 → Dec 2015 irritable bowel syndrome Tehran University of Medical Sciences Withdrawn No outcome recorded
Phase 4 NCT01536535 Jul 2012 → Apr 2018 ulcerative colitis Connecticut Children's Medical Center Completed No outcome recorded
Phase 4 NCT01316718 Mar 2011 → Sep 2013 irritable bowel syndrome University of Nottingham Completed No outcome recorded
Phase 4 NCT01201122 Sep 2010 → Dec 2015 ulcerative colitis Wolfson Medical Center Completed No outcome recorded
Phase 4 NCT01124149 Jun 2010 → Dec 2012 ulcerative colitis Shire Completed No outcome recorded
Phase 4 NCT01090102 Jun 2010 → Dec 2012 AIDS University of California, San Francisco Completed No outcome recorded
Phase 4 NCT01789294 Nov 2008 → Feb 2013 Azienda Policlinico Umberto I Unknown No outcome recorded
Phase 4 NCT00652145 Sep 2008 → Jan 2013 ulcerative colitis James Lewis Completed No outcome recorded
Phase not applicable3 trials
NCT03917095 May → Jun 2019 ulcerative colitis The Second Hospital of Nanjing Medical University Unknown No outcome recorded
NCT01999400 Apr 2012 → Sep 2015 University of Michigan Completed No outcome recorded
NCT00349388 Jul 2006 → Jan 2011 ulcerative colitis Annette Langseder Terminated No outcome recorded
Also used as a comparator or background therapy in 62 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT06525974 Comparator Sep 2024 → Sep 2026 expected ulcerative colitis Tanta University Not yet recruiting No outcome recorded
Phase 12 trials
Phase 1 NCT05912712 Comparator Jul 2023 → Jun 2025 solitary rectal ulcer syndrome, ulcerative colitis Xijing Hospital of Digestive Diseases Unknown No outcome recorded
Phase 1 NCT01020708 Comparator Nov 2009 → Sep 2010 ulcerative colitis Altheus Therapeutics, Inc. Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT05119140 Background Jun 2022 → May 2025 overdue ulcerative colitis Icahn School of Medicine at Mount Sinai Active not recruiting No outcome recorded
Phase 1/2 NCT03441893 Comparator Jan 2015 → Jul 2025 helminthiasis, protozoa infectious disease, ulcerative colitis Research Institute of Epidemiology, Microbiology and Infectious Diseases, Uzbekistan Unknown No outcome recorded
Phase 214 trials
Phase 2 NCT07333716 Comparator Jan 2026 → Feb 2027 expected ulcerative colitis Tanta University Recruiting No outcome recorded
Phase 2 NCT07349472 Comparator Jan 2026 → Jan 2027 expected inflammatory bowel disease Ihab Elsayed Hassan Recruiting No outcome recorded
Phase 2 NCT07064707 Comparator Jul 2025 → Jul 2026 overdue ulcerative colitis Alexandria University Recruiting No outcome recorded
Phase 2 NCT06993974 Comparator May 2025 → Aug 2026 overdue ulcerative colitis Alexandria University Recruiting No outcome recorded
Phase 2 NCT06213857 Background Feb → May 2025 overdue ulcerative colitis Tanta University Recruiting No outcome recorded
Phase 2/35 trials
Phase 2/3 NCT05988528 Comparator Aug 2023 → Feb 2025 inflammatory bowel disease Mostafa Bahaa Completed No outcome recorded
Phase 2/3 NCT05986136 Comparator Aug 2023 → Aug 2027 expected inflammatory bowel disease Mostafa Bahaa Recruiting No outcome recorded
Phase 2/3 NCT05753267 Comparator Feb 2023 → Sep 2025 inflammatory bowel disease Tanta University Completed No outcome recorded
Phase 2/3 NCT03804931 Background Jan 2019 → Dec 2028 expected ulcerative colitis Guangzhou First People's Hospital Recruiting No outcome recorded
Phase 2/3 NCT00774007 Comparator Sep 2004 → Nov 2005 irritable bowel syndrome SOFAR S.p.A. Completed No outcome recorded
Phase 322 trials
Phase 3 NCT03716388 Comparator Dec 2018 → Dec 2019 ulcerative colitis Dayanand Medical College and Hospital Unknown No outcome recorded
Phase 3 NCT03412682 Comparator Mar 2018 → May 2020 ulcerative colitis Ferring Pharmaceuticals Completed No outcome recorded
Phase 3 NCT02910245 Comparator Nov 2016 → Apr 2022 ulcerative colitis Academic Medical Center - University of Amsterdam Unknown No outcome recorded
Phase 3 NCT02683733 Comparator Feb 2016 → Feb 2017 ulcerative colitis Asian Institute of Gastroenterology, India Unknown No outcome recorded
Phase 3 NCT02280629 Comparator Oct 2014 → Oct 2018 ulcerative colitis Dr. Falk Pharma GmbH Completed No outcome recorded
Phase 48 trials
Phase 4 NCT07546097 Comparator Mar 2026 → Mar 2027 expected ulcerative colitis Yongquan Shi Recruiting No outcome recorded
Phase 4 NCT06625450 Comparator Oct 2024 → Dec 2025 overdue ulcerative colitis Post Graduate Institute of Medical Education and Research, Chandigarh Not yet recruiting No outcome recorded
Phase 4 NCT04133194 Comparator Nov 2019 → Dec 2024 ulcerative colitis Flemming Bendtsen Unknown No outcome recorded
Phase 4 NCT03110198 Comparator May 2017 → Jan 2018 ulcerative colitis Xijing Hospital of Digestive Diseases Unknown No outcome recorded
Phase 4 NCT01941589 Comparator Sep 2013 → Apr 2021 ulcerative colitis Sheba Medical Center Completed No outcome recorded
Phase not applicable8 trials
NCT07389824 Background Feb 2026 → Sep 2027 expected ulcerative colitis Qin Yu Not yet recruiting No outcome recorded
NCT06067698 Comparator Oct 2023 → Apr 2025 overdue ulcerative colitis Tanta University Recruiting No outcome recorded
NCT05780723 Comparator Apr 2023 → Oct 2024 ulcerative colitis Beijing Hospital of Traditional Chinese Medicine Completed No outcome recorded
NCT05538026 Comparator Sep 2020 → Jan 2022 ulcerative colitis Bogomolets National Medical University Completed No outcome recorded
NCT03415711 Background Apr 2017 → Apr 2019 ulcerative colitis VSL Pharmaceuticals Terminated No outcome recorded

Press releases naming this drug 9 releases

DateIssuerRelease
2021-04-23 Teva Branded Pharmaceutical Products R&D, Inc. Teva Announces Launch of its Generic Version of Canasa® (mesalamine) Suppositories To Treat Adults with Active Ulcerative Proctitis (ulcerative rectal colitis), in the United States tevapharm.com
2019-05-10 Teva Branded Pharmaceutical Products R&D, Inc. Teva Announces the Launch of a Generic Version of Delzicol® (mesalamine) Delayed-Release Capsules in the United States tevapharm.com
2018-03-26 Teva Branded Pharmaceutical Products R&D, Inc. Teva Announces the Launch of a Generic Version of Lialda® in the United States tevapharm.com
2016-10-05 Takeda Patent Trial and Appeal Board Upholds the Validity of LIALDA® Patent takeda.com
2016-09-16 Takeda District Court Issues Ruling in Hatch Waxman Case Regarding Shire’s LIALDA® takeda.com
2016-03-29 Takeda Shire Wins Patent Trial against Watson Concerning LIALDA® takeda.com
2015-04-06 Takeda Shire Comments on USPTO Petitions Related to LIALDA and GATTEX takeda.com
2013-05-09 Takeda Shire Wins Patent Trial Against Watson Concerning LIALDA® takeda.com
2004-10-01 Teva Branded Pharmaceutical Products R&D, Inc. Teva Announces Approval Of Mesalamine Rectal Suspension Usp tevapharm.com

Evidence & citations 33 cited values

Every value below carries the sentence it was read from. 166 sources stand behind the page.

FieldValueCited text
Known as Mesalamine “SPD476 (LIALDA in the US; MEZAVANT in the EU; otherwise known as MMX mesalamine; Shire Pharmaceuticals Inc., Wayne, PA, under license from Giuliani SpA, Milan, Italy) is a...” PMID 17241860 Oct 2006
83

“The objective of this study is to evaluate and compare the bioavailability of mesalamine and therefore to assess the bioequivalence of 375 mg APRISOTM extended-release capsule...” NCT03327558

“After the screening visits, eligible patients will be randomized to 1 of 3 study groups: (1) IBD98 M 0.8 g/day (mesalamine 0.8 g with sodium hyaluronate 92 mg), (2) IBD98 M 1.2...” NCT02493712

“A randomised, open-label, parallel-group study of mesalamine pharmacokinetics following Lialda 2 × 1.2 g once daily (QD) (dose A), Asacol 6 × 400 mg QD (dose B), or Asacol 2 ×...” PMID 32671846 Aug 2020

“compare the rate and extent of absorption of mesalamine-sodium hyaluronate 200 mg-28.75 mg delayed-release capsule (IBD98-M, Test) versus Delzicol 400 mg delayed-release...” NCT02196662

“Patients received corticosteroids alone or corticosteroid + mesalamine (4 g/day mesalamine) by a stratified randomization according to mesalamine use before admission.” PMID 35272029 Mar 2022

“MMX mesalazine/mesalamine (4.8 g) administered QD orally on Days 1-3, then a single oral dose of Amoxicillin (500 mg) + MMX mesalazine/mesalamine (4.8 g) on Day 4.” NCT01442688

“Patients were randomly assigned to groups that were given budesonide MMX (9 mg or 6 mg), mesalamine (2.4 g, as reference), or placebo for 8 weeks.” PMID 22892337 Aug 2012

“Similarly, 5-aminosalycilates (5-ASA) agents in the form of mesalamine/mesalzine are well established proven therapy in mild-moderate UC” NCT02665845

“Effect of once- or twice-daily MMX mesalamine (SPD476) for the induction of remission of mild to moderately active ulcerative colitis.” PMID 17234558 Jan 2007

“This study evaluated the pharmacokinetics of mesalamine and its major metabolite of mesalamine known as N-acetyl-mesalamine in plasma.” NCT01999400

“Mesalazine (also known as mesalamine or 5- amino salicylic acid, 5-ASA) has a well-established role in UC management.” NCT06201793

“Asacol®, Asacol® HD, Lialda®, Pentasa® (generic: mesalamine), minimum daily dose ≥2.4 grams (g)” NCT01532648

“Asacol 4.8 g/day (800 mg mesalamine tablet) versus Asacol 2.4 g/day (400 mg mesalamine tablet)” NCT00350415

“new mesalamine suppositories (MAX-002) as compared to placebo and active medicine” NCT01016262

“PENTASA Sachet 6 g/Day (Mesalazine, Mesalamine) With Placebo.” NCT00862121

mesalamine; 5-aminosalicylic acid; 5-ASA; mesalazine” NCT01004185

“standardised mesalazine (mesalamine) therapy” PMID 31373712 Aug 2019

“Mesalazine (Mesalamine)” NCT00245505

NCT01045018

NCT01841099

NCT03716388

NCT01469637

NCT02280629

NCT05753267

NCT03415711

NCT01120340

NCT01088243

NCT02910245

NCT01201122

NCT00254618

NCT06525974

NCT00952952

NCT02522780

NCT02522767

NCT00554099

NCT01586533

NCT00446849

NCT05781698

NCT05488405

NCT06993974

NCT00326209

NCT00652145

NCT05567068

NCT00073021

NCT01696942

NCT01627262

NCT00514982

NCT01020708

NCT07349472

NCT01789294

NCT00577473

NCT00744016

NCT01418365

NCT01130844

NCT05988528

NCT01327300

NCT01209208

NCT03070574

NCT06213857

NCT05986136

NCT01402947

NCT05119140

NCT01177410

NCT06625450

NCT00840203

NCT00622375

NCT07333716

NCT01124149

NCT00343850

NCT01172444

NCT00767728

NCT00505778

NCT05663775

NCT04920149

NCT07064707

NCT06067698

NCT05316220

NCT01412372

NCT00802451

NCT02125292

NCT00746447

NCT01090102

NCT02093663

Known as 5- amino salicylic acid “Mesalamine or 5-amino salicylic acid (5-ASA), plays a crucial role in the treatment of ulcerative colitis (UC). It is the first-line therapy for mild to moderate cases of UC...” NCT07064707
13

“Mesalamine (5-ASA, 5-aminosalicylic acid), used safely in patients with ulcerative colitis, may reduce CRC risk in LS by decreasing microsatellite instability, a key driver of...” PMID 41213710 Nov 2025

“Despite mesalamine's or 5-amino salicylic acid's (5-ASA) established role in inducing and maintaining remission, some patients experience persistent symptoms and inflammatory activity.” PMID 41235106 Oct 2025

“Mesalazine (also known as mesalamine or 5- amino salicylic acid, 5-ASA) has a well-established role in UC management.” NCT06201793

“Mesalazine (also known as mesalamine or 5- amino salicylic acid, 5-ASA) has a well-established role in UC management.” NCT06525974

“Mesalamine (also known as mesalamine or 5- amino salicylic acid, 5-ASA) has a well-established role in UC management.” NCT05753267

“Limited data are available on mesalamine (5-aminosalicylic acid; 5-ASA) use in pediatric ulcerative colitis (UC).” PMID 26893546 Feb 2016

“Mesalamine or 5-amino salicylic acid (5-ASA), plays a crucial role in the treatment of ulcerative colitis (UC).” NCT06993974

“Mesalamine, also known as 5-aminosalicylic acid (5-ASA), is a medication used to treat ulcerative colitis.” NCT05986136

“Mesalamine (5-aminosalicylic acid, Apriso)” NCT01090102

NCT02683733

NCT00069498

NCT00984568

NCT01320436

Known as 5-aminosalicylic acid (5-ASA) “Mesalamine, also known as 5-aminosalicylic acid (5-ASA), is a medication used to treat ulcerative colitis.” NCT05988528
1

“Mesalamine, also known as 5-aminosalicylic acid (5-ASA)NCT05663775

Known as 5-ASA “Mesalamine or 5-amino salicylic acid (5-ASA), plays a crucial role in the treatment of ulcerative colitis (UC). It is the first-line therapy for mild to moderate cases of UC...” NCT07064707
11

“Despite mesalamine's or 5-amino salicylic acid's (5-ASA) established role in inducing and maintaining remission, some patients experience persistent symptoms and inflammatory activity.” PMID 41235106 Oct 2025

“Mesalamine (also known as mesalamine or 5- amino salicylic acid, 5-ASA) has a well-established role in UC management.” NCT05753267

“Mesalazine (also known as mesalamine or 5- amino salicylic acid, 5-ASA) has a well-established role in UC management.” NCT06525974

“Mesalazine (also known as mesalamine or 5- amino salicylic acid, 5-ASA) has a well-established role in UC management.” NCT06201793

“Limited data are available on mesalamine (5-aminosalicylic acid; 5-ASA) use in pediatric ulcerative colitis (UC).” PMID 26893546 Feb 2016

“Mesalamine or 5-amino salicylic acid (5-ASA), plays a crucial role in the treatment of ulcerative colitis (UC).” NCT06993974

“Mesalamine, also known as 5-aminosalicylic acid (5-ASA), is a medication used to treat ulcerative colitis.” NCT05986136

“the effect of the anti-inflammatory drug 5-aminosalicylic acid (5-ASA) on the gut mucosa” NCT00069498

“Zoenasa Rectal Gel (4.0g mesalamine \[5-ASA\], 1.0g N-acetylcysteine \[NAC\]; 60ml)” NCT01586533

“5-aminosalicylic compounds (5ASA) such as olsalazine and mesalamine” NCT01320436

“Several oral mesalazine (5-ASA) formulations exist” NCT04133194

Known as 5-ASA (5-Aminosalicylate) ClinicalTrials.gov intervention name — accepted as the source's own label NCT00603733
Known as Apriso “Three formulations of mesalamine, Pentasa, Apriso, and Lialda, were studied in the crossover phase” NCT01999400
1

“Mesalamine (5-aminosalicylic acid, Apriso)” NCT01090102

Known as Asacol “This study was conducted to determine the efficacy and safety of once-daily dosing of delayed-release mesalamine (Asacol 400-mg tablets) compared with twice-daily dosing for...” PMID 20064514 Jan 2010
13

Asacol® is mesalazine in a pH-dependent tablet (Eudragit S) that remains intact until reaching the terminal ileum.” NCT04032652

“To demonstrate that import Mesalazine (Asacol®) is non-inferior to the reference drug, marketed Mesalazine” NCT01257386

“Patients received mesalazine (mesalamine) 4.8 g/day (Asacol 800 mg MR) or 2.4 g/day (Asacol 400 mg MR).” PMID 21385195 Mar 2011

Asacol®, Asacol® HD, Lialda®, Pentasa® (generic: mesalamine), minimum daily dose ≥2.4 grams (g)” NCT01532648

Asacol® 2.4 g/Day (400 mg Mesalamine Tablet)” NCT00554099

“1600 mg Asacol [mesalazine]” NCT04133194

Asacol 800 mg (mesalamine)” NCT00073021

“mesalazine (Asacol®)” NCT00708656

Asacol (mesalamine)” NCT00343850

NCT00349388

NCT00194818

NCT00713310

NCT00092508

Known as Asacol HD “Asacol®, Asacol® HD, Lialda®, Pentasa® (generic: mesalamine), minimum daily dose ≥2.4 grams (g)” NCT01532648
Known as Canasa Canasa® Rectal Suppositories (1000 mg Mesalamine, USP)” NCT01172444
Known as Delzicol “compare the rate and extent of absorption of mesalamine-sodium hyaluronate 200 mg-28.75 mg delayed-release capsule (IBD98-M, Test) versus Delzicol 400 mg delayed-release...” NCT02196662
1

Delzicol 100 mg mesalamine x 1 with 245 mL water; single dose” NCT01999400

Known as eMG “To compare the maintenance of remission from mild to moderate ulcerative colitis as measured by rectal bleeding and endoscopic mucosal appearance after 6 months of treatment...” NCT00767728
1

“encapsulated mesalamine Granules (eMG) (formerly referred to as Mesalamine Pellets [MP])” NCT00326209

Known as IBD98-M “compare the rate and extent of absorption of mesalamine-sodium hyaluronate 200 mg-28.75 mg delayed-release capsule (IBD98-M, Test) versus Delzicol 400 mg delayed-release...” NCT02196662
Known as IBD98-M without HA IBD98-M without HA: Mesalamine 200mg X2” NCT02196662
Known as Lialda “Three formulations of mesalamine, Pentasa, Apriso, and Lialda, were studied in the crossover phase” NCT01999400
1

“Asacol®, Asacol® HD, Lialda®, Pentasa® (generic: mesalamine), minimum daily dose ≥2.4 grams (g)” NCT01532648

Known as MAX-002 “new mesalamine suppositories (MAX-002) as compared to placebo and active medicine” NCT01016262
Known as MES “1 g mesalamine suppositories (1 g MES;” PMID 29702300 Apr 2018
Known as Mesalamin ClinicalTrials.gov intervention name — accepted as the source's own label NCT01059344
Known as Mesalazine “A Phase 1, Randomized, Open-label, Crossover, Drug Interaction Study Evaluating the Pharmacokinetic Profiles of Ciprofloxacin XR Administered Alone and in Combination With MMX®...” NCT01402947
68

“An Open Label, Single-site Pharmaco-Scintigraphic Study in Healthy Subjects With Radio-labelled TP05-tablets (Mesalazine) to Evaluate the Gastrointestinal Transit and Release...” NCT02306772

Mesalazine (mesalamine) granules (MG) were shown to be effective for the maintenance of remission of ulcerative colitis (UC) in two double-blind placebo-controlled trials.” PMID 22617015 May 2012

Mesalazine Modified-Release Tablet in the Treatment of Ulcerative Colitis in the Remission Phase: A Chinese, Multicenter, Single-Blind, Randomized Controlled Study.” PMID 26905266 Feb 2016

Mesalazine is an experimental drug designed to gradually release 5-ASA into the areas of large bowel associated with ulcerative colitis.” NCT00151892

“Multi MatriX system (MMX®) formulation of mesalazine/mesalazine (Lialda®; Mesavancol®; Mezavant®) (MMX Mesalazine/mesalamine).” NCT01469637

“Asacol is a delayed-release tablet formulation designed to deliver mesalamine (also known as mesalazine) at a pH ≥ 7.0.” NCT00254618

Mesalazine (also known as mesalamine or 5- amino salicylic acid, 5-ASA) has a well-established role in UC management.” NCT06525974

“Asacol® is mesalazine in a pH-dependent tablet (Eudragit S) that remains intact until reaching the terminal ileum.” NCT04032652

“Patients received mesalazine (mesalamine) 4.8 g/day (Asacol 800 mg MR) or 2.4 g/day (Asacol 400 mg MR).” PMID 21385195 Mar 2011

“replacing thiopurines with high-dose oral mesalazine (≥ 3 g/day) may preserve remission” NCT07248644

Mesalazine is used to treat and prevent mild to moderate acute fissure disease” NCT05091775

“Metronidazole Drug Interaction Study With MMX® Mesalazine/Mesalamine” NCT01418365

“PENTASA Sachet 6 g/Day (Mesalazine, Mesalamine) With Placebo.” NCT00862121

“using scintigraphic images and mesalazine plasma levels (PK)” NCT02306785

“with mesalazine 4 g/day as maintenance therapy.” NCT07546097

“4800 grams/day of Mesalazine (Asacol/Mezavant)” NCT01534312

“MMX Mesalamine/Mesalazine (Low Dose)” NCT02093663

Mesalazine and/or Prednisone” NCT03804931

“MMX mesalamine/ mesalazineNCT01124149

NCT01894685

NCT00450086

NCT01966783

NCT00626288

NCT01699438

NCT00708656

NCT02769494

NCT02190526

NCT05912712

NCT02335281

NCT05780723

NCT03104036

NCT00774007

NCT00737789

NCT04133194

NCT00976690

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NCT01257386

Known as Mesalazine, Pentasa (trade name) Mesalazine, Pentasa (trade name)NCT01841099
Known as mesalzine “Similarly, 5-aminosalycilates (5-ASA) agents in the form of mesalamine/mesalzine are well established proven therapy in mild-moderate UC” NCT02665845
Known as Mesavancol “Multi MatriX system (MMX®) formulation of mesalazine/mesalazine (Lialda®; Mesavancol®; Mezavant®) (MMX Mesalazine/mesalamine).” NCT01469637
Known as MEZAVANT “SPD476 (LIALDA in the US; MEZAVANT in the EU; otherwise known as MMX mesalamine; Shire Pharmaceuticals Inc., Wayne, PA, under license from Giuliani SpA, Milan, Italy) is a...” PMID 17241860 Oct 2006
1

“Multi MatriX system (MMX®) formulation of mesalazine/mesalazine (Lialda®; Mesavancol®; Mezavant®) (MMX Mesalazine/mesalamine).” NCT01469637

Known as MMX Mesalamine “SPD476 (LIALDA in the US; MEZAVANT in the EU; otherwise known as MMX mesalamine; Shire Pharmaceuticals Inc., Wayne, PA, under license from Giuliani SpA, Milan, Italy) is a...” PMID 17241860 Oct 2006
3

“MMX® mesalamine is a once daily oral 5-aminosalicylic acid formulation, effective in induction and maintenance of ulcerative colitis remission.” PMID 24868146 May 2014

“Effect of once- or twice-daily MMX mesalamine (SPD476) for the induction of remission of mild to moderately active ulcerative colitis.” PMID 17234558 Jan 2007

“30 mg/kg/day of MMX Mesalamine tablets, dosed once daily for 7 days.” NCT01130844

Known as MMX mesalazine “AIM: Maintenance treatment in ulcerative colitis should be as convenient as possible, to increase the chance of compliance. MMX mesalazine is a once-daily, high-strength (1.2...” PMID 18272546 Feb 2008
3

“SPD476 (MMX mesalazine), is a novel, once daily, high-strength mesalazine formulation (1.2 g/tablet) that utilizes Multi Matrix System (MMX) technology to delay and extend...” PMID 16984503 Oct 2006

“Metronidazole Drug Interaction Study With MMX® Mesalazine/Mesalamine” NCT01418365

“SPD476, MMX™ mesalazine, 1.2g extended release tablet” NCT00545103

Known as MMX Mesalazine/mesalamine “Multi MatriX system (MMX®) formulation of mesalazine/mesalazine (Lialda®; Mesavancol®; Mezavant®) (MMX Mesalazine/mesalamine).” NCT01469637