Drugs / prilocaine
last change 3 days ago re-read 2 minutes ago

prilocaine

Small molecule

Developed for
chronic pain syndrome · hemorrhoid · cervical incompetence · diabetes mellitus · female infertility · hernia, double inguinal · osteoarthritis, knee · premature ejaculation
+6 more · shoulder impingement syndrome · stroke disorder · thalassemia · coronary vasospasm · frozen shoulder · myofascial pain syndrome
Investigated by
Cairo University · Aalborg University · Assiut University · University of Campinas, Brazil · CAMC Health System · Centre Hospitalier Universitaire Saint Pierre
+53 more · São Paulo Research Foundation · ASST Gaetano Pini-CTO · Academic Medical Center - University of Amsterdam · Ain Shams University · Ankara University · Assistance Publique - Hôpitaux de Paris · Bagcilar Training and Research Hospital · Centre Hospitalier le Mans · Colorado Clinical & Translational Sciences Institute · Dentsply International · Diskapi Teaching and Research Hospital · Dow University of Health Sciences · Dr. Pere Roura-Poch · Enrique Velasco Serna · Erasmus Medical Center · Franciscan University Center · Gustavo Adolfo Sarriá · Guy's and St Thomas' NHS Foundation Trust · Helwan University · Hippocration General Hospital · Hopital Saint Roch · Hospital General Universitario Gregorio Marañon · Indonesia Endowment Fund for Education · Indonesia University · Institue of Microengineering and Nanoelectronics (IMEN), Universiti Kebangsaan Malaysia · Loma Linda University · Lund University Hospital · Marmara University · Miguel Delicado Miralles · National Institute on Aging (NIA) · National Science and Technology Council, Taiwan · National Taiwan University Hospital · National University Hospital, Singapore · Netherlands Institute for Pigment Disorders · Obstetric Anaesthetists' Association United Kingdom · Oregon Health and Science University · Patricia Beltra Lopez · Plethora Solutions Ltd · Pontificia Universidad Catolica de Chile · Regionshospitalet Horsens · St. Mary's Research Center, Canada · Stanford University · Sultan Abdulhamid Han Training and Research Hospital, Istanbul, Turkey · Tanta University · Technical University of Munich · Universitas Sebelas Maret · Universiti Kebangsaan Malaysia Medical Centre · Universiti Kebangsaan Malaysia Medical Molecular Biology Institute (UMBI) · University Hospital Waterford · University Hospital, Angers · University Hospital, Montpellier · University of Aarhus · University of Colorado, Denver

Regulatory milestones approvals, filings & regulatory actions · 2 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved EU (EMA) Fortacin 2013-11-15 europa.eu
Approved US (FDA) CITANEST PLAIN 1965-11-18 fda.gov

Trials 56 · a red edge is where a trial was stopped

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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT05060913 Nov 2021 → Mar 2022 Dow University of Health Sciences Completed No outcome recorded
Phase 15 trials
Phase 1 NCT05062356 Nov 2021 → Aug 2024 chronic pain syndrome St. Mary's Research Center, Canada Completed No outcome recorded
Phase 1 NCT05912335 Jun 2021 → Feb 2022 tooth disorder University of Campinas, Brazil Completed No outcome recorded
Phase 1 NCT01324843 Jun 2009 → May 2010 National Institute on Aging (NIA) Completed No outcome recorded
Phase 1 NCT01425840 Mar → Nov 2008 University of Campinas, Brazil Completed No outcome recorded
Phase 1 NCT01054547 Sep → Dec 2006 University of Campinas, Brazil Completed No outcome recorded
Phase 25 trials
Phase 2 NCT05078463 Sep 2021 → Aug 2022 thalassemia Universiti Kebangsaan Malaysia Medical Centre Completed No outcome recorded
Phase 2 NCT03578783 Dec 2018 → May 2021 premature ejaculation Plethora Solutions Ltd Completed No outcome recorded
Phase 2 NCT03433976 May 2018 → May 2020 University Hospital, Montpellier Unknown No outcome recorded
Phase 2 NCT03036384 Mar → Nov 2016 Centre Hospitalier Universitaire Saint Pierre Completed No outcome recorded
Phase 2 NCT03607916 Feb → Aug 2014 Centre Hospitalier Universitaire Saint Pierre Completed No outcome recorded
Phase 34 trials
Phase 3 NCT06769204 Feb → Aug 2025 overdue female infertility Cairo University Not yet recruiting No outcome recorded
Phase 3 NCT03508804 Dec 2020 → Dec 2022 Stanford University Withdrawn No outcome recorded
Phase 3 NCT02130830 May 2014 → May 2016 hemorrhoid Pontificia Universidad Catolica de Chile Completed No outcome recorded
Phase 3 NCT00959595 Nov 2008 → Jan 2010 diabetes mellitus Lund University Hospital Completed No outcome recorded
Phase 423 trials
Phase 4 NCT06767085 Feb → Jul 2025 overdue Cairo University Not yet recruiting No outcome recorded
Phase 4 NCT07329582 May 2024 → Dec 2025 overdue National University Hospital, Singapore Active not recruiting No outcome recorded
Phase 4 NCT06133881 Dec 2023 → Feb 2024 Cairo University Completed No outcome recorded
Phase 4 NCT05970354 Sep 2023 → Dec 2024 overdue CAMC Health System Enrolling by invitation No outcome recorded
Phase 4 NCT05834647 Aug → Nov 2023 local anesthetic poisoning Universitas Sebelas Maret Unknown No outcome recorded
Phase 4 NCT05984264 Jan → Sep 2023 Assiut University Unknown No outcome recorded
Phase 4 NCT05649020 Nov 2022 → Dec 2023 Hospital General Universitario Gregorio Marañon Unknown No outcome recorded
Phase 4 NCT05610007 Jan → Aug 2022 Indonesia University Unknown No outcome recorded
Phase 4 NCT04394533 Aug 2021 → Aug 2025 cervical incompetence Guy's and St Thomas' NHS Foundation Trust Completed No outcome recorded
Phase 4 NCT04355598 Apr → Aug 2020 Cairo University Unknown No outcome recorded
Phase not applicable18 trials
NCT07683182 Nov 2025 → Jun 2026 overdue Marmara University Active not recruiting No outcome recorded
NCT06891794 Aug 2025 → Apr 2026 overdue uterine inflammatory disease Oregon Health and Science University Recruiting No outcome recorded
NCT07034456 Jul 2025 → Jan 2026 overdue Patricia Beltra Lopez Not yet recruiting No outcome recorded
NCT06600048 Sep 2024 → Mar 2025 Tanta University Completed No outcome recorded
NCT07664618 Apr 2024 → May 2025 Helwan University Completed No outcome recorded
NCT05877690 Oct 2023 → Oct 2024 Assiut University Unknown No outcome recorded
NCT05926895 Jun 2023 → Aug 2024 shoulder impingement syndrome Sultan Abdulhamid Han Training and Research Hospital, Istanbul, Turkey Completed No outcome recorded
NCT06274905 Feb → Jul 2023 head and neck cancer, skin neoplasm University Hospital Waterford Completed No outcome recorded
NCT07156968 Jan 2022 → Feb 2023 Ain Shams University Completed No outcome recorded
NCT05195177 Nov 2021 → Dec 2023 Aalborg University Unknown No outcome recorded
Also used as a comparator or background therapy in 64 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 02 trials
Phase 0 NCT06680167 Comparator Oct 2024 → Nov 2025 Sohag University Completed No outcome recorded
Phase 0 NCT02427724 Comparator Apr 2015 → May 2024 lentigo Northwestern University Completed No outcome recorded
Phase 14 trials
Phase 1 NCT03313336 Comparator Oct → Nov 2017 AstraZeneca Completed No outcome recorded
Phase 1 NCT03441841 Comparator Feb → Mar 2016 Galeno Desenvolvimento de Pesquisas Clínicas Completed No outcome recorded
Phase 1 NCT03325803 Background Sep 2015 → Sep 2016 actinic keratosis Dong-A University Completed No outcome recorded
Phase 1 NCT01073371 Comparator Jul 2008 → Aug 2009 University of Campinas, Brazil Completed No outcome recorded
Phase 1/23 trials
Phase 1/2 NCT05694858 Comparator Feb 2025 → Dec 2026 expected cataract, glaucoma Universiti Kebangsaan Malaysia Medical Centre Recruiting No outcome recorded
Phase 1/2 NCT06382220 Comparator Apr → Jul 2024 Fayoum University Hospital Completed No outcome recorded
Phase 1/2 NCT05289804 Comparator Sep 2022 → Dec 2025 cognitive disorder, cognitive impairment with or without cerebellar ataxia University of Dublin, Trinity College Completed No outcome recorded
Phase 22 trials
Phase 2 NCT02658773 Comparator Jan → May 2016 Assiut University Completed No outcome recorded
Phase 2 NCT00916942 Background Jun 2009 postherpetic neuralgia NeurogesX Completed No outcome recorded
Phase 2/33 trials
Phase 2/3 NCT04523961 Comparator Jan 2021 → Feb 2025 local anesthetic poisoning Mayo Clinic Completed No outcome recorded
Phase 2/3 NCT00932542 Comparator Apr 2010 → Feb 2011 hemorrhoid Federal University of São Paulo Unknown No outcome recorded
Phase 2/3 NCT00556478 Comparator Oct 2007 → Oct 2009 premature ejaculation Plethora Solutions Ltd Completed No outcome recorded
Phase 36 trials
Phase 3 NCT06703580 Comparator Nov 2024 → Dec 2025 Cairo University Completed No outcome recorded
Phase 3 NCT06165679 Comparator Dec 2023 → Jun 2025 Cairo University Completed No outcome recorded
Phase 3 NCT05726968 Comparator Nov 2022 → Jun 2023 Cairo University Completed No outcome recorded
Phase 3 NCT02990364 Comparator Dec 2015 → Dec 2016 American University of Beirut Medical Center Completed No outcome recorded
Phase 3 NCT03366246 Comparator Jun → Jul 2014 Galeno Desenvolvimento de Pesquisas Clínicas Completed No outcome recorded
Phase 419 trials
Phase 4 NCT07564180 Comparator May 2026 → May 2027 expected Amr mohamed Not yet recruiting No outcome recorded
Phase 4 NCT07546370 Comparator Apr 2026 → Apr 2027 expected Monakshi Sawhney Not yet recruiting No outcome recorded
Phase 4 NCT07262398 Comparator Aug → Dec 2024 Theodor Bilharz Research Institute Completed No outcome recorded
Phase 4 NCT05609565 Comparator Nov 2022 → Sep 2024 Ain Shams University Completed No outcome recorded
Phase 4 NCT06540599 Comparator Sep → Oct 2022 Gaziosmanpasa Research and Education Hospital Completed No outcome recorded
Phase not applicable25 trials
NCT07383571 Comparator Oct 2025 → Apr 2026 Cairo University Completed No outcome recorded
NCT05668286 Comparator May → Nov 2024 frozen shoulder Kartal City Hospital Unknown No outcome recorded
NCT06290583 Comparator Apr → Dec 2024 South Valley University Completed No outcome recorded
NCT06416111 Comparator Oct 2023 → Sep 2024 chronic kidney disease Ankara City Hospital Bilkent Completed No outcome recorded
NCT07174167 Comparator Apr 2023 → Feb 2024 osteoarthritis, knee Haydarpasa Numune Training and Research Hospital Completed No outcome recorded

Evidence & citations 26 cited values

Every value below carries the sentence it was read from. 122 sources stand behind the page.

FieldValueCited text
Known as prilocaine “EMLA Cream (Eutectic Mixture of Local Anesthetics) is an FDA-approved topical anesthetic comprised of 2.5% each of lidocaine/prilocaine. EMLA Cream was applied in approximately...” NCT00444626
116

“transrectal ultrasound guided 10 ml prilocaine and serum physiologic blend (5ml %2 prilocaine and 5 ml serum physiologic) injected separetly 5ml right and 5ml left junction...” NCT02025361

“The EMLA group received EMLA cream which consisted of 2.5% lidocaine and 2.5 % prilocaine in 2 ml of water/oil emulsion and then they received tegaderm as the dressing for...” NCT03134391

“At the start of session 2, one area of the middle forearms of the participant will be located (4x4cm). On the area, local anesthetic cream (2.5% lidocain/2.5 prilocaine) will...” NCT05195177

“EMLA®, a topical anesthetic cream containing lidocaine and prilocaine, will be applied under occlusion prior to tape application during 30 minutes with the aim of anesthetize...” NCT07034456

“liposome-encapsulated 2% ropivacaine, liposome-encapsulated 1% ropivacaine, a eutectic mixture of 2.5% lidocaine and 2.5% prilocaine (EMLA), and liposomal placebo gel,...” PMID 21106282 Nov 2010

“100 mg of the following formulations: Liposome-encapsulated 2,5% and 5% lidocaine gel, liposome placebo gel and 2.5% lidocaine and 2.5% prilocaine cream were applied once...” NCT01425840

“The purpose of this study is to compare the effects of vapocoolant spray and topical lidocaine 2.5% + prilocaine 2.5% cream (EMLA) on reducing pain during needle electromyography.” NCT01606046

“a local anaesthetic cream consisting of equal parts of lidocaine and prilocaine (1g contains 25 mg of lidocaine and 25 mg of prilocaine, AstraZeneca A/S, Albertslund, Denmark)” NCT04076865

“standard EMLA patch which is a eutectic emulsion mixture of lidocaine and prilocaine at 1:1 ratio (i.e. each gram of EMLA cream contains lidocaine and prilocaine, 25 mg each).” NCT05694858

“EMLA cream 5% 25g lidocaine, 25g prilocaine; Astra Zeneca. Topically applied followed by Tegaderm dressing to cover. Length of duration monitored and recorded as part of study” NCT06274905

“EMLA (eutectic mixture of local anesthetic) cream is the combination of lidocaine and prilocaine which have been effectively used in few studies to reduce needle prick pain.” NCT04050059

“EMLA® Test Patch containing the active ingredients lidocaine base 25 mg/g and prilocaine base 25 mg/g in an oil-in-water emulsion saturating the absorbent cellulose disc.” NCT03313336

“Effect of Local Anesthetic EMLA (Lidocaine 2.5% and Prilocaine 2.5%) Cream and Reduction in Dose, Pain and Intravenous Analgesic During Permanent Pacemaker Implantation” NCT02016976

“the prilocaine group underwent spinal anaesthesia with 60 mg intrathecal prilocaine; and the bupivacaine group received 12.5 mg intrathecal heavy bupivacaine.” PMID 33428221 Jan 2021

“PSD502 is a topical (applied to skin) anesthetic spray containing a mixture of two drugs called lidocaine and prilocaine that will be applied to the penis.” NCT03578783

“This research study uses Eutectic Mixture of Local Anesthetics (EMLA) Cream (lidocaine 2.5% and prilocaine 2.5%) as the topical anaesthetic agent.” NCT05078463

“In the Active Comparator arm, lidocaine 2.5% and prilocaine 2.5% cream placed over area where lumbar puncture will occur for at least 30 minutes.” NCT01628874

“EMLA cream is a eutectic mixture of 2.5% lidocaine and 2.5% prilocaine, used as a topical anaesthetic to diminish pain from cutaneous procedures.” NCT02990364

“hydrogels containing LAs - lidocaine and prilocaine (both at 2.5%) encapsulated in CLN (XAN-CLN) or not (XAN-CLN ), EMLA and placebo hydrogel” NCT05912335

“OBJECTIVE: To compare the anesthetic performances of 3% prilocaine and 4% articaine when used for the extraction of the maxillary teeth.” PMID 32934619 May 2020

“40 mg (low dose) intrathecal hyperbaric prilocaine 2% (Takipril, Sunny Medical group, Egypt under liscense from Sintetica, Switzerland)” NCT06382220

“EMLA cream with occluding dressing on the shoulder before surgery(5% of eutectic mixture with 2.5% lidocaine and 2.5% prilocaine)” NCT01845532

“EMLA anesthetic ointment (AO-Astra Zeneca) is an emulsion of lidocaine 2.5% and prilocaine 2.5% in a ratio of 1:1 by weight” NCT03501212

“Eutectic mixture of lidocaine 25 mg/g and prilocaine 25 mg/g cream (EMLA cream) will be applied at this test region at t1.” NCT02246179

“50 g of a local anesthetic agent containing 2.5% Lidocaine and 2.5% Prilocaine (EMLA®, AstraZeneca - Södertälje, Sweden)” NCT00959595

“Then one area will be pre-treated with cutaneous 2.5% lidocaine/2.5% prilocaine cream (EMLA cream) for 1 hour.” NCT04858360

“2 puffs of lidocaine-prilocaine spray into the cervix and cervical canal 5 minutes before the procedure” NCT06769204

“Group I received thoracic interlaminar epidural injections of 6 mL of 2% preservative-free prilocaine.” NCT06507995

“one cream will be an anesthetic (lidocaine and prilocaine) and the other will be a placebo lotion.” NCT01324843

“hyperbaric Prilocaine 2% in a reduced dose (30mg) in combination with Fentanyl (25µg)” NCT05726968

“a eutectic mixture containing 25 mg/g of lidocaine and 25 mg/g of prilocaine (EMLA®)” NCT01860235

“EMLA is a mixture of lidocaine (2.5%) and prilocaine (2.5%) in a cream base.” NCT04378283

“EMLA cream (lidocaine 2.5% and prilocaine 2.5% in a ratio of 1:1 by weight)” NCT03072394

“Eutectic Mixture of Local Anesthetics (Lidocaine 2.5% and Prilocaine 2.5%)” NCT05970354

“Patients using paracervical block with prilocaine for analgesia” NCT06540599

“topically applied lidocaine-prilocaine (EMLA) cream” NCT02549105

“Emla 5% cream (Lignocaine 2.5% / Prilocaine 2.5%)” NCT01847157

“EMLA cream (lidocaine 2.5% and prilocaine 2.5%)” NCT04003012

“lidocaine 25 mg/g + prilocaine 25 mg/g cream” NCT02548533

“2.5% prilocaine-2.5% lidocaine cream” NCT06891794

“2.5% Lidocaine and 2.5% PrilocaineNCT05060913

“spinal anesthesia with prilocaineNCT07156968

“EMLA cream (lidocaine+prilocaine)” NCT06885723

NCT03038958

NCT00408941

NCT04394533

NCT06703580

NCT05751148

NCT04784104

NCT03219086

NCT02883179

NCT00932542

NCT01425619

NCT05289804

NCT06899438

NCT05877690

NCT07564180

NCT06165679

NCT05834647

NCT07383571

NCT05649020

NCT05648708

NCT07546370

NCT03441841

NCT05609565

NCT03731988

NCT01303614

NCT06416111

NCT06680167

NCT04756050

NCT02726620

NCT05062356

NCT01880775

NCT02390310

NCT03366246

NCT07664618

NCT04355598

NCT03508804

NCT02427724

NCT03071601

NCT06290583

NCT00916942

NCT06133881

NCT02130830

NCT04523961

NCT00556478

NCT00309673

NCT05926895

NCT05688202

NCT02658773

NCT05610007

NCT05984264

NCT02820688

NCT02372786

NCT06600048

NCT07262398

NCT06767085

NCT07329582

NCT01643616

NCT02384915

NCT07174167

NCT07683182

NCT02336958

NCT01591616

NCT01402869

NCT03325803

NCT01921231

NCT05891132

NCT03607916

NCT01309360

NCT05042817

NCT01073371

NCT03264586

NCT03799484

NCT03220555

NCT03036384

Known as ASTRA 1512 ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as ASTRA-1515 ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as citanest ClinicalTrials.gov intervention name — accepted as the source's own label NCT01412632
Known as Citanest hydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as Citanest plain ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as Citanest plain dental ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as L-67 HYDROCHLORIDE ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as NSC-40027 ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as NSC-758432 ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as Priloc “Injection of 1 CC Betamethasone Dipropionate + Betamethasone Sodium Phosphate (Diprospan) and 4 cc 2% Prilocaine (Priloc)mixture into the subacromial space” NCT05926895
Known as Priloc %2 “Autologous Blood Injection group were administered 1ml of autologous venous blood mixed with 2ml of 2% prilocaine HCl(Priloc %2,Vem,Turkey) subcutaneously.” NCT06236178
Known as Priloc HCl %2 “20 ml of bupivacaine(Buvicaine HCl %0.5) and prilocaine(Priloc HCl %2) 1:1 mixture” NCT04756050
Known as Prilocaina ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as Prilocaine component of emla ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as Prilocaine component of fortacin ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as Prilocaine component of oraqix ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as Prilocaine HCl “Those in the AB group were administered 1 ml of autologous venous blood mixed with 2 ml of 2% prilocaine HCl.” PMID 38963583 Jul 2024
1

“EPINEPHrine 1:200,000 / Prilocaine HCl 4 % 1.8 ML Cartridge” NCT05062356

Known as prilocaine hydrochloride “prilocaine 2% (Takipril, prilocaine hydrochloride 20 mg/mL, hyperbar, Sintetica)” NCT05726968
2

“prilocaine 2% (Takipril, prilocaine hydrochloride 20 mg/mL, hyperbar, Sintetica)” NCT06133881

NCT05668286

Known as Propitocaine ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as Propitocaine hydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Known as Takipril “40 mg (low dose) intrathecal hyperbaric prilocaine 2% (Takipril, Sunny Medical group, Egypt under liscense from Sintetica, Switzerland)” NCT06382220
2

“prilocaine 2% (Takipril, prilocaine hydrochloride 20 mg/mL, hyperbar, Sintetica)” NCT06133881

“prilocaine 2% (Takipril, prilocaine hydrochloride 20 mg/mL, hyperbar, Sintetica)” NCT05726968

Known as Xylonest ChEMBL registry synonym — accepted as the source's own label CHEMBL1194
Action Inhibit “This lidocaine/prilocaine preparation blocks sodium channels in peripheral nerves in the skin” NCT05289804
Modality Small molecule CHEMBL1194