Drugs / Megestrol Acetate
last change Aug 2026 re-read 2 minutes ago

Megestrol Acetate

Other / unclassified

Developed for
atypical endometrial hyperplasia · endometrial cancer · eating disorder · HIV wasting syndrome · hypoproteinemia, hypercatabolic · endometrial carcinoma · breast cancer · non-small cell lung carcinoma
+30 more · endometrial endometrioid adenocarcinoma · small cell lung carcinoma · cancer · chemotherapy-induced toxicity · endometrium adenocarcinoma · head and neck cancer · HIV infectious disease · nutritional disorder · adrenal cortex carcinoma · anorexia nervosa · breast neoplasm · cancer-related condition · chronic obstructive pulmonary disease · dementia · endometrioid adenocarcinoma · esophageal squamous cell carcinoma · gastric carcinoma · gastroesophageal cancer · head and neck squamous cell carcinoma · idiopathic central precocious puberty · intraepithelial neoplasia · liver cancer · malignant mesothelioma · paraneoplastic gastrointestinal syndrome · squamous cell intraepithelial neoplasia · stage I endometrioid carcinoma · uterine cancer · uterine corpus cancer · uterus carcinoma in situ · endometrial disorder
Investigated by
National Cancer Institute (NCI) · Changchun GeneScience Pharmaceutical Co., Ltd. · Fudan University · Bristol-Myers Squibb · Henan Cancer Hospital · Xiaojun Chen
+99 more · Northwestern University · Peking University People's Hospital · Asan Medical Center · Beijing Chao Yang Hospital · Guangzhou Institute of Respiratory Disease · Gynecologic Oncology Group · Hunan Province Tumor Hospital · LG Life Sciences · NRG Oncology · National Institute of Allergy and Infectious Diseases (NIAID) · Peking Union Medical College Hospital · Peking University Third Hospital · Rottapharm Spain · Shengjing Hospital · The First Affiliated Hospital of Henan University of Science and Technology · Tongji Hospital · Wake Forest University Health Sciences · Aiping Zhou · Alliance for Clinical Trials in Oncology · Anticancer Fund, Belgium · AstraZeneca · Azienda Socio Sanitaria Territoriale degli Spedali Civili di Brescia · Brazilian National Cancer Institute · Cambridge University Hospitals NHS Foundation Trust · Canadian Clinical Trials Group (sponsor POLEmut-BLUE trial) · Canadian Institutes of Health Research (CIHR) · Cancer Research UK & UCL Cancer Trials Centre · Cancer Research UK Cambridge Institute · Chang Gung Memorial Hospital · Children's Hospital of Fudan University · City of Hope Medical Center · Comprehensive Cancer Centre The Netherlands · Covance · Daewon Pharmaceutical Co., Ltd. · Dutch Cancer Society · Dutch Gynaecological Oncology Group · Endo USA Inc., a Keenova Therapeutics Company · Gamma Project - ACTU · Guang'anmen Hospital of China Academy of Chinese Medical Sciences · Hospital Universitari de Bellvitge · Huashan Hospital · Huazhong University of Science and Technology · Institute Gustave Roussy (sponsor p53abn-RED trial) · KK Women's and Children's Hospital · Leiden University Medical Center · Leiden University Medical center (sponsor MMRd-GREEN trial) · Mayo Clinic · Merck Sharp & Dohme LLC · Milton S. Hershey Medical Center · NCIC Clinical Trials Group · NYU Langone Health · Nanfang Hospital, Southern Medical University · National Cancer Institute, France · National Center for Research Resources (NCRR) · National Medical Research Council (NMRC), Singapore · Ontario Institute for Cancer Research · Par Pharmaceutical, Inc. · Peking University · Qilu Hospital of Shandong University · Qingdao Central Hospital · Quintiles, Inc. · Roxane Laboratories · SFBC Anapharm · Second Xiangya Hospital of Central South University · Severance Hospital · Shaanxi Provincial Cancer Hospital · Shandong Cancer Hospital and Institute · Shandong University · Shanghai 6th People's Hospital · Shanghai Changning Maternity & Infant Health Hospital · Shanxi Bethune Hospital · Shenzhen Fifth People's Hospital · Sixth Affiliated Hospital, Sun Yat-sen University · St. Vincent Medical Center - Los Angeles · all 105 on the full record

Regulatory milestones approvals, filings & regulatory actions · 1 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved US (FDA) MEGACE 1971-08-18 fda.gov

Trials 89 · started per year

today
US approved 1971
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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 19 trials
Phase 1 NCT07338487 Apr → Dec 2026 expected cervical cancer, hypoproteinemia, hypercatabolic Second Xiangya Hospital of Central South University Recruiting No outcome recorded
Phase 1 NCT07130617 Sep 2025 → Jul 2026 overdue Changchun GeneScience Pharmaceutical Co., Ltd. Not yet recruiting No outcome recorded
Phase 1 NCT05332483 Jul 2022 → Oct 2023 endometrial cancer Sunnybrook Health Sciences Centre Terminated No outcome recorded
Phase 1 NCT06147908 Jul → Oct 2022 Daewon Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT01383330 Jul → Sep 2011 Asan Medical Center Unknown No outcome recorded
Phase 1 NCT01342055 Mar → May 2011 LG Life Sciences Completed No outcome recorded
Phase 1 NCT02446353 Apr → Jun 2010 LG Life Sciences Completed No outcome recorded
Phase 1 NCT00637403 May 2006 Par Pharmaceutical, Inc. Terminated No outcome recorded
Phase 1 NCT00000737 HIV wasting syndrome, hypoproteinemia, hypercatabolic National Institute of Allergy and Infectious Diseases (NIAID) Completed No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT05538897 Mar 2023 → Jan 2027 expected endometrial endometrioid adenocarcinoma National Cancer Institute (NCI) Active not recruiting No outcome recorded
Phase 1/2 NCT00002465 Dec 1987 → ? breast cancer, endometrial cancer, malignant mesothelioma St. Vincent Medical Center - Los Angeles Unknown No outcome recorded
Phase 234 trials
Phase 2 NCT07565415 Jun 2026 → Sep 2027 expected hepatocellular carcinoma, hypoproteinemia, hypercatabolic, nutritional disorder Nanfang Hospital, Southern Medical University Not yet recruiting No outcome recorded
Phase 2 NCT07391826 Feb → Dec 2026 expected gastric carcinoma The First Affiliated Hospital with Nanjing Medical University Not yet recruiting No outcome recorded
Phase 2 NCT07377734 Jan 2026 → Dec 2027 expected atypical endometrial hyperplasia, endometrial cancer Wang Jianliu Recruiting No outcome recorded
Phase 2 NCT07246070 Dec 2025 → Aug 2026 overdue chemotherapy-induced toxicity Aiping Zhou Not yet recruiting No outcome recorded
Phase 2 NCT07092137 Oct 2025 → Oct 2026 expected lung cancer Guangzhou Institute of Respiratory Disease Not yet recruiting No outcome recorded
Phase 2 NCT06979596 Aug 2025 → Nov 2027 expected cancer Merck Sharp & Dohme LLC Recruiting No outcome recorded
Phase 2 NCT06909383 Jun 2025 → Jun 2026 overdue paraneoplastic gastrointestinal syndrome, small cell lung carcinoma Guangzhou Institute of Respiratory Disease Not yet recruiting No outcome recorded
Phase 2 NCT06914297 Apr 2025 → Oct 2027 expected endometrial cancer Fudan University Recruiting No outcome recorded
Phase 2 NCT06793228 Jan 2025 → Jan 2027 expected small cell lung carcinoma Henan Cancer Hospital Not yet recruiting No outcome recorded
Phase 2 NCT05913427 Jun 2022 → Jun 2027 expected adrenal cortex carcinoma Azienda Socio Sanitaria Territoriale degli Spedali Civili di Brescia Recruiting No outcome recorded
Phase 2/39 trials
Phase 2/3 NCT07319429 Jan 2026 → Dec 2027 expected endometrial cancer, infertility disorder Fudan University Recruiting No outcome recorded
Phase 2/3 NCT05316493 Jun 2022 → Feb 2026 overdue atypical endometrial hyperplasia, infertility disorder Xiaojun Chen Recruiting No outcome recorded
Phase 2/3 NCT05316467 May 2022 → Feb 2026 endometrial carcinoma, female infertility, obesity disorder Xiaojun Chen Terminated No outcome recorded
Phase 2/3 NCT05255653 Nov 2021 → Jan 2030 expected endometrial cancer Leiden University Medical Center Recruiting No outcome recorded
Phase 2/3 NCT04683237 Mar 2021 → Nov 2025 atypical endometrial hyperplasia, infertility disorder, obesity disorder Xiaojun Chen Withdrawn No outcome recorded
Phase 2/3 NCT04491682 Sep 2020 → Jun 2022 atypical endometrial hyperplasia Fudan University Completed No outcome recorded
Phase 2/3 NCT03241888 Jul 2017 → Jun 2020 atypical endometrial hyperplasia Fudan University Completed No outcome recorded
Phase 2/3 NCT03241914 Jul 2017 → Jun 2020 stage I endometrioid carcinoma Fudan University Completed No outcome recorded
Phase 2/3 NCT00503516 Jun 2007 → Dec 2009 dementia Rottapharm Spain Terminated No outcome recorded
Phase 317 trials
Phase 3 NCT07543536 May 2026 → Apr 2029 expected breast cancer Sun Yat-sen University Not yet recruiting No outcome recorded
Phase 3 NCT07477808 Apr 2026 → Apr 2028 expected non-small cell lung carcinoma Hunan Province Tumor Hospital Not yet recruiting No outcome recorded
Phase 3 NCT07356037 Jan 2026 → Jun 2027 expected HIV wasting syndrome, hepatocellular carcinoma Changchun GeneScience Pharmaceutical Co., Ltd. Not yet recruiting No outcome recorded
Phase 3 NCT06998758 Nov 2025 → May 2027 expected Sixth Affiliated Hospital, Sun Yat-sen University Recruiting No outcome recorded
Phase 3 NCT07150663 Aug 2025 → Jun 2027 expected non-small cell lung carcinoma Changchun GeneScience Pharmaceutical Co., Ltd. Recruiting No outcome recorded
Phase 3 NCT06961188 Jun 2025 → Jun 2027 expected non-small cell lung carcinoma Changchun GeneScience Pharmaceutical Co., Ltd. Not yet recruiting No outcome recorded
Phase 3 NCT06828757 May 2025 → Dec 2026 expected non-small cell lung carcinoma Hunan Province Tumor Hospital Not yet recruiting No outcome recorded
Phase 3 NCT06961201 May 2025 → Dec 2026 expected small cell lung carcinoma Changchun GeneScience Pharmaceutical Co., Ltd. Not yet recruiting No outcome recorded
Phase 3 NCT06772428 Jan 2025 → Jun 2027 expected head and neck squamous cell carcinoma Changchun GeneScience Pharmaceutical Co., Ltd. Not yet recruiting No outcome recorded
Phase 3 NCT06500234 Jun 2024 → May 2025 overdue cancer, nutritional disorder Qingdao Central Hospital Recruiting No outcome recorded
Phase 410 trials
Phase 4 NCT07462663 Jan 2027 → Apr 2031 expected atypical endometrial hyperplasia, endometrial cancer, intraepithelial neoplasia, morbid obesity Hospital Universitari de Bellvitge Not yet recruiting No outcome recorded
Phase 4 NCT07254416 Dec 2025 → Dec 2026 expected Tianjin Medical University Cancer Institute and Hospital Not yet recruiting No outcome recorded
Phase 4 NCT07243379 Sep 2025 → Dec 2026 expected Changchun GeneScience Pharmaceutical Co., Ltd. Recruiting No outcome recorded
Phase 4 NCT06963593 Jun 2025 → Jun 2027 expected gastroesophageal cancer Peking University Not yet recruiting No outcome recorded
Phase 4 NCT03963752 Aug 2019 → Aug 2022 idiopathic central precocious puberty Children's Hospital of Fudan University Completed No outcome recorded
Phase 4 NCT03815019 Aug 2019 → Mar 2025 eating disorder University of Kansas Medical Center Completed No outcome recorded
Phase 4 NCT03777930 Dec 2018 → Oct 2020 cancer-related condition Shenzhen Fifth People's Hospital Unknown No outcome recorded
Phase 4 NCT02595723 Jul 2015 → Nov 2016 cognitive impairment with or without cerebellar ataxia University of Texas Southwestern Medical Center Completed No outcome recorded
Phase 4 NCT00163072 Oct 2005 → Dec 2012 hypoproteinemia, hypercatabolic Milton S. Hershey Medical Center Withdrawn No outcome recorded
Phase 4 NCT00002345 HIV infectious disease, eating disorder, hypoproteinemia, hypercatabolic Bristol-Myers Squibb Completed No outcome recorded
Phase not applicable8 trials
NCT07408505 Jun 2026 → Dec 2027 expected pancreatic ductal adenocarcinoma Shandong Cancer Hospital and Institute Recruiting No outcome recorded
NCT06830018 Jan 2025 → Jan 2026 overdue Changchun GeneScience Pharmaceutical Co., Ltd. Recruiting No outcome recorded
NCT06549855 Oct 2024 → Jul 2029 expected endometrial cancer, endometrioid adenocarcinoma Peking University People's Hospital Not yet recruiting No outcome recorded
NCT06468215 Jul 2024 → Jul 2028 expected endometrial endometrioid adenocarcinoma Peking University People's Hospital Not yet recruiting No outcome recorded
NCT05945407 Aug 2016 → Dec 2023 overdue endometrial cancer, endometrial endometrioid adenocarcinoma Peking University People's Hospital Recruiting No outcome recorded
NCT00575029 Apr → Dec 2004 adrenocortical insufficiency University of Arkansas Completed No outcome recorded
NCT00004664 Jun 1995 → ? AIDS, HIV wasting syndrome National Center for Research Resources (NCRR) Completed No outcome recorded
NCT00002182 HIV infectious disease Gamma Project - ACTU Completed No outcome recorded
Also used as a comparator or background therapy in 27 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 14 trials
Phase 1 NCT01589562 Comparator Apr → Jun 2012 Daewon Pharmaceutical Co., Ltd. Completed No outcome recorded
Phase 1 NCT01456624 Comparator Sep 2011 → Jun 2012 Asan Medical Center Completed No outcome recorded
Phase 1 NCT01397214 Comparator Jul → Sep 2011 eating disorder, hypoproteinemia, hypercatabolic Boryung Pharmaceutical Co., Ltd Completed No outcome recorded
Phase 1 NCT00638079 Comparator Jun → Jul 2006 Endo USA Inc., a Keenova Therapeutics Company Completed No outcome recorded
Phase 211 trials
Phase 2 NCT07714070 Background Jul 2026 → Sep 2027 expected atypical endometrial hyperplasia, endometrial cancer, progesterone resistance Peking University People's Hospital Not yet recruiting No outcome recorded
Phase 2 NCT07436793 Comparator Jun 2026 → Jun 2030 expected endometrial disorder, endometrial endometrioid adenocarcinoma New Mexico Cancer Research Alliance Recruiting No outcome recorded
Phase 2 NCT05380479 Comparator Jun 2022 → Jan 2023 eating disorder Bangabandhu Sheikh Mujib Medical University, Dhaka, Bangladesh Unknown No outcome recorded
Phase 2 NCT05247268 Comparator Mar 2022 → Mar 2027 expected endometrial carcinoma Fudan University Recruiting No outcome recorded
Phase 2 NCT03283488 Comparator Mar 2019 → Feb 2022 eating disorder, hypoproteinemia, hypercatabolic University of Sao Paulo Completed No outcome recorded
Phase 2/33 trials
Phase 2/3 NCT04607252 Comparator Jan → Jun 2021 atypical endometrial hyperplasia Fudan University Terminated No outcome recorded
Phase 2/3 NCT04385667 Comparator May 2020 → Dec 2022 atypical endometrial hyperplasia Zagazig University Completed No outcome recorded
Phase 2/3 NCT02619266 Comparator Dec 2015 → Dec 2016 eating disorder Xinqiao Hospital of Chongqing Unknown No outcome recorded
Phase 38 trials
Phase 3 NCT06671548 Background Jan 2024 → Nov 2026 expected leiomyoma Qilu Pharmaceutical Co., Ltd. Recruiting No outcome recorded
Phase 3 NCT04897217 Comparator Jun 2023 → Oct 2024 atypical endometrial hyperplasia Wake Forest University Health Sciences Withdrawn No outcome recorded
Phase 3 NCT04939090 Comparator Jan 2022 → Apr 2027 expected cancer, hematopoietic and lymphoid cell neoplasm Alliance for Clinical Trials in Oncology Active not recruiting No outcome recorded
Phase 3 NCT00637806 Comparator Jun → Sep 2006 Par Pharmaceutical, Inc. Terminated No outcome recorded
Phase 3 NCT00637728 Comparator Jun → Sep 2006 eating disorder Par Pharmaceutical, Inc. Terminated No outcome recorded
Phase not applicable1 trial
NCT06417736 Background Dec 2023 → Jul 2025 overdue endometrial cancer Women's Hospital School Of Medicine Zhejiang University Recruiting No outcome recorded

Press releases naming this drug 1 release

DateIssuerRelease
2003-05-06 Teva Branded Pharmaceutical Products R&D, Inc. Teva Announces Approval of Megestrol Acetate Oral Suspension tevapharm.com

Evidence & citations 14 cited values

Every value below carries the sentence it was read from. 119 sources stand behind the page.

FieldValueCited text
Known as megestrol acetate “High-potency progestin given orally as background therapy in both groups: medroxyprogesterone acetate 250-500 mg/day or megestrol acetate 160-320 mg/day, with the specific...” NCT07714070
102

“OBJECTIVE: To compare the efficacy of the levonorgestrel intrauterine system (LNG-IUS) versus megestrol acetate (MA) in inducing complete regression among women with atypical...” PMID 38425141 Feb 2024

“Eligible patients will be enrolled into the study and administered sodium cridanimod (500 mg i.m./ twice a week) in combination with megestrol acetate (160 mg p.o./ day) or...” NCT02064725

Megestrol acetate (Megace®) is a progestin analog that is FDA approved for the palliative treatment of breast and endometrial carcinoma.” NCT00163072

“They will take oral high-dose progestin (Medroxyprogesterone Acetate 250mg-500mg/d or Megestrol Acetate 160mg-320mg/d) daily.” NCT07377734

“Tolerability and pharmacokinetics of two formulations of megestrol acetate under fed conditions in healthy volunteers.” PMID 25450470 Oct 2014

“all subjects determined to be PrR positive will receive progestin monotherapy, megestrol acetate, for up to 24 weeks.” NCT03077698

“Typical regimens include medroxyprogesterone acetate (400-600 mg/day) or megestrol acetate (160-320 mg/day).” NCT07462663

Megestrol acetate (Megace) is a synthetic derivative of the natural occurring steroid hormone, progesterone.” NCT05492487

“two orally administered megestrol acetate suspensions (625 mg/5 mL) in healthy Korean male subjects” PMID 38586120 Mar 2024

“Efficacy of megestrol acetate (MA) was evaluated in patients who did not respond to CH.” PMID 18989154 Nov 2008

“with oral medroxyprogesterone acetate (MPA) 500mg/d or megestrol acetate (MA) 320mg/d” NCT06468215

“Pharmacokinetics of a nanocrystal-containing megestrol acetate formulation” PMID 27191767 Sep 2016

megestrol acetate (MA, 160 mg qd po)/megestrol acetate (MPA, 500 mg qd po)” NCT06914297

megestrol acetate 40 mg orally 4 times daily for up to 5 years.” PMID 24724218 Mar 2014

megestrol acetate (1 mg) administered orally once daily” NCT06671548

Megestrol acetate 800mg/20ml, Suspension, Single dose” NCT01589562

megestrol acetate ("YiLiZhi") 160-320mg/d orally” NCT05945407

Megestrol AcetateNCT05255653

NCT04897217

NCT00637572

NCT02269670

NCT03815019

NCT03306472

NCT00739830

NCT07565415

NCT06549855

NCT03241914

NCT05913427

NCT00638079

NCT04576104

NCT01501396

NCT00041275

NCT03671811

NCT07092137

NCT05316493

NCT07246070

NCT06417736

NCT05316467

NCT07319429

NCT00503581

NCT00503516

NCT07436793

NCT03024580

NCT05247268

NCT07543536

NCT07391826

NCT04683237

NCT01968317

NCT00910091

NCT05332483

NCT00004912

NCT07338487

NCT06500234

NCT05380479

NCT06772428

NCT06961201

NCT03963752

NCT06979596

NCT06998758

NCT00507949

NCT07356037

NCT07130617

NCT00637806

NCT00002345

NCT07408505

NCT00005975

NCT00002300

NCT00637403

NCT00070148

NCT00575029

NCT05538897

NCT06830018

NCT01200602

NCT00000737

NCT07243379

NCT00637728

NCT06963593

NCT04939090

NCT07254416

NCT00729586

NCT00002465

NCT06961188

NCT01237327

NCT06909383

NCT06793228

NCT01943058

NCT03777930

NCT00483327

NCT00031707

NCT04491682

NCT07150663

NCT02980653

NCT02619266

NCT00002182

NCT00001079

NCT04607252

NCT00031785

NCT07477808

NCT03241888

NCT00006799

NCT00002067

NCT04491643

Known as MA-ES “It is available in its original formulation, Megace (MAOS), and as a nanocrystal dispersion, Megace ES (MA-ES).” PMID 19774117 Sep 2009
Known as MAOS “It is available in its original formulation, Megace (MAOS), and as a nanocrystal dispersion, Megace ES (MA-ES).” PMID 19774117 Sep 2009
Known as Megace “Phase III Double-Blind, Placebo-Controlled Randomized Comparison of Megestrol Acetate (Megace) Versus an N-3 Fatty Acid (EPA) Enriched Nutritional Supplement Versus Both for...” NCT00031707
8

“Various progestins have been investigated including Megace (megesterol acetate) and Provera (medroxyprogesterone acetate) for the treatment of endometrial cancer.” NCT00584857

“Megestrol acetate (Megace®) is a progestin analog that is FDA approved for the palliative treatment of breast and endometrial carcinoma.” NCT00163072

“It is available in its original formulation, Megace (MAOS), and as a nanocrystal dispersion, Megace ES (MA-ES).” PMID 19774117 Sep 2009

“Megestrol acetate (Megace) is a synthetic derivative of the natural occurring steroid hormone, progesterone.” NCT05492487

“Megestrol Acetate (Megace)” NCT00070148

“Drug: megaceNCT01383330

NCT01383330

NCT01456624

Known as Megace acetate Megace acetate oral suspension” NCT01397214
Known as Megesterol Acetate ClinicalTrials.gov intervention name — accepted as the source's own label NCT00584857
Known as megestrol “Hormone therapy using megestrol may fight liver cancer by blocking the uptake of estrogen.” NCT00041275
12

“Tablets of 160mg megestrol will be used according to randomization.” NCT05380479

NCT00066248

NCT04430361

NCT02595723

NCT00004664

NCT00016341

NCT06828757

NCT00002680

NCT03283488

NCT00420563

NCT01206478

NCT02644408

Known as Megestrol acetate: Megace Megestrol acetate: MegaceNCT01968317
Known as MPA “megestrol acetate (MA, 160 mg qd po)/megestrol acetate (MPA, 500 mg qd po)” NCT06914297
Known as Nano-crystalline Megestrol Acetate Nano-crystalline megestrol acetate is administered as an oral suspension at a dose of 625 mg once daily (5 mL, 125 mg/mL) starting concurrently with first-line chemotherapy and...” NCT07408505
1

“The oral suspension of megestrol acetate adopts nano-crystal technology (referred to as nano-crystalline megestrol acetate)” NCT07092137

Known as YiLiZhi “megestrol acetate ("YiLiZhi") 160-320mg/d orally” NCT05945407
Action Inhibit “Hormone therapy using megestrol may fight cancer by reducing the production of these hormones.” NCT00002465
Modality Other / unclassified “Megestrol Acetate (MA) is a progesterone-like hormone” NCT00575029
Route Oral “Megace oral suspension daily” NCT00002345