Drugs / procarbazine
last change May 2026 re-read 2 minutes ago

procarbazine

Small molecule

Developed for
lymphoma · Hodgkins lymphoma · central nervous system neoplasm · glioblastoma · primary central nervous system lymphoma · central nervous system cancer · brain neoplasm · classic Hodgkin lymphoma
+7 more · diffuse large B-cell lymphoma · large-cell immunoblastic lymphoma · malignant glioma · non-Hodgkin lymphoma · precursor lymphoblastic lymphoma/leukemia · anaplastic astrocytoma · oligodendroglioma
Investigated by
National Cancer Institute (NCI) · European Organisation for Research and Treatment of Cancer - EORTC · Alliance for Clinical Trials in Oncology · Case Comprehensive Cancer Center · Memorial Sloan Kettering Cancer Center · University of Cologne
+69 more · Children's Cancer and Leukaemia Group · Eastern Cooperative Oncology Group · Lymphoma Study Association · SWOG Cancer Research Network · Children's Oncology Group · M.D. Anderson Cancer Center · Medical Research Council · NCIC Clinical Trials Group · North Central Cancer Treatment Group · Radiation Therapy Oncology Group · University College, London · AIDS Malignancy Consortium · Australasian Leukaemia and Lymphoma Group · Beijing Tiantan Hospital · Canadian Cancer Trials Group · Cancer Institute WIA · Cancer Research UK · Cancer Research UK & UCL Cancer Trials Centre · Children's Cancer Group · Children's Hospital of Philadelphia · Christine Mauz-Körholz · Columbia University · Consorzio Mario Negri Sud · Cordgenics, LLC · Deutsche AIDS Gesellschaft e.V. · ECOG-ACRIN Cancer Research Group · Fondazione Italiana Linfomi - ETS · Fondazione Michelangelo · GITIL (GRUPPO ITALIANO TERAPIE INNOVATIVE NEI LINFOMI) · Grup per l'Estudi dels Limfomes de Catalunya i Balears · Harlachinger Krebshilfe e.V. · Hebei Yanda Hospital · Incheon St.Mary's Hospital · Indiana University · Institute of Cancer Research, United Kingdom · International Extranodal Lymphoma Study Group (IELSG) · Kentuckiana Cancer Institute · Lee's Pharmaceutical Limited · Ludwig-Maximilians - University of Munich · Lymphoma Trials Office · Merck KGaA, Darmstadt, Germany · Merck Sharp & Dohme LLC · NRG Oncology · National Cancer Center, Korea · National Research Center for Hematology, Russia · New Approaches to Brain Tumor Therapy Consortium · Nordic Lymphoma Group · Northern Sydney and Central Coast Area Health Service · Northwestern Memorial Hospital · Northwestern University · OHSU Knight Cancer Institute · Ospedale Santa Croce-Carle Cuneo · Pfizer · Pharmacyclics LLC. · Polish Lymphoma Research Group · St. Jude Children's Research Hospital · Technical University Dresden · The Emmes Company, LLC · UNICANCER · University Hospital Carl Gustav Carus · University Hospital Cologne · University Hospital Freiburg · University Hospital Heidelberg · University Hospital Ulm · University of Arkansas · University of Vermont · University of Virginia · Wake Forest University Health Sciences · Weill Medical College of Cornell University

Regulatory milestones approvals, filings & regulatory actions · 1 recorded

MilestoneJurisdictionBrandIndicationDateSentence it was read from
Approved US (FDA) MATULANE 1969-07-22 fda.gov

Trials 64 · started per year

today
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PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 01 trial
Phase 0 NCT00734773 Nov 2008 → ? central nervous system neoplasm, lymphoma Northwestern University Withdrawn No outcome recorded
Phase 11 trial
Phase 1 NCT00005796 Feb 2000 → Jun 2003 bone marrow disorder, central nervous system neoplasm, chemotherapy-induced toxicity Indiana University Completed No outcome recorded
Phase 1/21 trial
Phase 1/2 NCT00004004 Jul 1999 → Aug 2003 central nervous system neoplasm New Approaches to Brain Tumor Therapy Consortium Completed No outcome recorded
Phase 231 trials
Phase 2 NCT05008224 Oct 2021 → Oct 2023 classic Hodgkin lymphoma Merck Sharp & Dohme LLC Completed No outcome recorded
Phase 2 NCT05425654 May 2021 → May 2023 primary central nervous system lymphoma National Research Center for Hematology, Russia Unknown No outcome recorded
Phase 2 NCT03495960 Jun 2019 → Dec 2024 primary central nervous system lymphoma International Extranodal Lymphoma Study Group (IELSG) Completed No outcome recorded
Phase 2 NCT01775475 Sep 2016 → Apr 2021 diffuse large B-cell lymphoma, large-cell immunoblastic lymphoma, precursor lymphoblastic lymphoma/leukemia AIDS Malignancy Consortium Completed No outcome recorded
Phase 2 NCT01390584 May 2013 → Apr 2015 lymphoma ECOG-ACRIN Cancer Research Group Terminated No outcome recorded
Phase 2 NCT01737346 Oct 2012 → Sep 2013 glioblastoma Incheon St.Mary's Hospital Unknown No outcome recorded
Phase 2 NCT01118026 Sep 2010 → Sep 2020 lymphoma Alliance for Clinical Trials in Oncology Completed No outcome recorded
Phase 2 NCT01132807 May 2010 → Feb 2016 lymphoma Alliance for Clinical Trials in Oncology Completed No outcome recorded
Phase 2 NCT01124240 Nov 2009 → Nov 2012 glioblastoma Northern Sydney and Central Coast Area Health Service Unknown No outcome recorded
Phase 2 NCT00989352 Sep 2009 → Jun 2011 primary central nervous system lymphoma University Hospital Freiburg Unknown No outcome recorded
Phase 2/31 trial
Phase 2/3 NCT00003375 Oct 1998 → Aug 2005 central nervous system neoplasm Radiation Therapy Oncology Group Completed No outcome recorded
Phase 321 trials
Phase 3 NCT05675410 May 2023 → Apr 2031 expected Hodgkins lymphoma National Cancer Institute (NCI) Recruiting No outcome recorded
Phase 3 NCT03632135 May 2018 → Jun 2022 glioblastoma Cordgenics, LLC Completed No outcome recorded
Phase 3 NCT01652261 May 2013 → Oct 2014 Hodgkins lymphoma European Organisation for Research and Treatment of Cancer - EORTC Withdrawn No outcome recorded
Phase 3 NCT00887146 Sep 2009 → Oct 2029 expected central nervous system neoplasm Alliance for Clinical Trials in Oncology Active not recruiting No outcome recorded
Phase 3 NCT00678327 Aug 2008 → Jan 2016 lymphoma University College, London Completed No outcome recorded
Phase 3 NCT00515554 May 2008 → Jul 2019 Hodgkins lymphoma University of Cologne Completed No outcome recorded
Phase 3 NCT00433433 Oct 2006 → Dec 2011 lymphoma European Organisation for Research and Treatment of Cancer - EORTC Unknown No outcome recorded
Phase 3 NCT00052455 Oct 2002 → Sep 2010 central nervous system cancer Institute of Cancer Research, United Kingdom Completed No outcome recorded
Phase 3 NCT00049595 Aug 2002 → Jan 2010 lymphoma European Organisation for Research and Treatment of Cancer - EORTC Completed No outcome recorded
Phase 3 NCT01251107 Mar 2000 → Nov 2009 Hodgkins lymphoma Fondazione Michelangelo Completed No outcome recorded
Phase 41 trial
Phase 4 NCT00188149 May 2000 → Dec 2007 Hodgkins lymphoma University Hospital Carl Gustav Carus Unknown No outcome recorded
Phase not applicable7 trials
NCT02800447 Jun 2016 → Dec 2018 Hodgkins lymphoma Lee's Pharmaceutical Limited Unknown No outcome recorded
NCT02333513 Feb 2015 → Dec 2017 malignant glioma Hebei Yanda Hospital Unknown No outcome recorded
NCT01304849 Jan 2011 → Sep 2013 Hodgkins lymphoma Cancer Institute WIA Completed No outcome recorded
NCT00187057 Sep 2002 → Aug 2006 ataxia telangiectasia St. Jude Children's Research Hospital Completed No outcome recorded
NCT00594815 Aug 2002 → Feb 2016 lymphoma Memorial Sloan Kettering Cancer Center Completed No outcome recorded
NCT00416377 lymphoma Children's Cancer and Leukaemia Group Unknown No outcome recorded
NCT00417014 lymphoma Children's Cancer and Leukaemia Group Unknown No outcome recorded
Also used as a comparator or background therapy in 20 trials
PhaseRegistry idDatesIndicationSponsorStatusOutcome
Phase 11 trial
Phase 1 NCT06541665 Background May 2024 → Apr 2028 expected primary central nervous system lymphoma Ono Pharmaceutical Co., Ltd. Active not recruiting No outcome recorded
Phase 1/22 trials
Phase 1/2 NCT03576378 Background Aug 2018 → Oct 2023 Hodgkins lymphoma Spanish Lymphoma Cooperative Group Unknown No outcome recorded
Phase 1/2 NCT02315326 Background Dec 2014 → Jan 2026 central nervous system non-hodgkin lymphoma Memorial Sloan Kettering Cancer Center Completed No outcome recorded
Phase 27 trials
Phase 2 NCT07015242 Background Nov 2025 → Jan 2028 expected lymphoma Juno Therapeutics, Inc., a Bristol-Myers Squibb Company Recruiting No outcome recorded
Phase 2 NCT02298283 Background Apr 2015 → Jul 2020 Hodgkins lymphoma The Lymphoma Academic Research Organisation Completed No outcome recorded
Phase 2 NCT01569204 Comparator Oct 2012 → Mar 2014 Hodgkins lymphoma University of Cologne Completed No outcome recorded
Phase 2 NCT01399372 Background Sep 2011 → Mar 2020 chemotherapy-induced toxicity, cognitive disorder, lymphoma, radiation-induced disorder Radiation Therapy Oncology Group Completed No outcome recorded
Phase 2 NCT00503594 Comparator Jul 2007 → Jul 2010 lymphoma Assistance Publique - Hôpitaux de Paris Unknown No outcome recorded
Phase 310 trials
Phase 3 NCT06830421 Comparator Aug 2023 → Aug 2029 expected primary central nervous system lymphoma University Hospital Freiburg Recruiting No outcome recorded
Phase 3 NCT04702581 Background Dec 2021 → Dec 2030 expected oligodendroglioma Hospices Civils de Lyon Recruiting No outcome recorded
Phase 3 NCT05331521 Comparator Apr 2021 → Mar 2033 expected oligodendroglioma University Hospital Heidelberg Recruiting No outcome recorded
Phase 3 NCT02661503 Comparator Jul 2016 → Dec 2022 classic Hodgkin lymphoma University of Cologne Unknown No outcome recorded
Phase 3 NCT02444000 Background Sep 2015 → Oct 2022 malignant glioma Assistance Publique - Hôpitaux de Paris Completed No outcome recorded

Evidence & citations 19 cited values

Every value below carries the sentence it was read from. 85 sources stand behind the page.

FieldValueCited text
Known as procarbazine “Control chemotherapy treatment will be chosen from any of the following standard-of-care chemotherapy drugs or combinations: * Carboplatin; * Irinotecan; * Etoposide; *...” NCT03632135
75

“bleomycin 10 units/m\^2 IV on Day 8 etoposide 200 mg/m\^2 IV on Days 1, 2 and 3 doxorubicin 35 mg/m\^2 IV on Day 1 cyclophosphamide 1250 mg/m\^2 IV on Day 1 vincristine 1.4...” NCT01118026

“BACOPP-D regimen which includes cyclophosphamide, adriamycin, dacarbazine, procarbazine, prednisolone, bleomycin and vincristine” NCT00188149

“temozolomide: capsules, up to 200 mg/sqm/day, 5 days per cycle; PCV (procarbazine, CCNU, vincristine): standard regimen” NCT00431561

“bleomycin, etoposide, adriamycin, cyclophosphamide, vincristine, procarbazine, and prednisone (BEACOPPesc)” NCT01652261

Procarbazine100 mg/m2/b.m./die 1°- 7° Prednison40 mg/m2/b.m./die 1°-14°” NCT00795613

“cyclophosphamide, procarbazine, etoposide and prednisone (BEACOPP)” PMID 28601705 Jun 2017

“Days 8-21: Procarbazine 60 mg/m2 orally (capped at 100 mg).” NCT05331521

“plus Procarbazine 100mg/m2 by mouth (OR) on Day1 through 5” NCT03576378

“Prednisone, Cyclophosphamide, Etoposide, ProcarbazineNCT00151281

“Cap Procarbazine 100mg/m2 Day 1 to Day 7 PO” NCT01304849

“Days 8 to 21: procarbazine 60 mg/m2 orally” NCT02444000

“Days 8 to 21: Procarbazine 60 mg/m2 orally” NCT04702581

Procarbazine 100 mg/m2 orally day 1 to 7” NCT00433433

“100 mg/m2 oral procarbazine on days 1-7” PMID 30658935 Jan 2019

“daily procarbazine (PCB, 50 mg p.o.” NCT01124240

ProcarbazineNCT00592111

NCT00265031

NCT00005796

NCT00887146

NCT00049439

NCT00004010

NCT00574496

NCT01132807

NCT00002840

NCT06541665

NCT00049595

NCT00666484

NCT00003375

NCT00004004

NCT03495960

NCT06830421

NCT00003788

NCT01399372

NCT00577993

NCT00052455

NCT00074191

NCT02333513

NCT00433459

NCT00003564

NCT05425654

NCT00187057

NCT00335140

NCT00002463

NCT00002944

NCT00025064

NCT01390584

NCT00416377

NCT00079105

NCT00003293

NCT01569204

NCT00079092

NCT01356680

NCT00002462

NCT01737346

NCT05008224

NCT00417014

NCT00379041

NCT01251107

NCT00503594

NCT00989352

NCT00264953

NCT00594815

NCT02661503

NCT02298283

NCT02315326

NCT00002806

NCT07015242

NCT01468740

NCT00002569

NCT00003101

NCT00515554

NCT00416832

NCT00003114

NCT00678327

NCT00003421

Known as Ibenzmethyzine hydrochloride ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Known as Matulane ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Known as Natulan ClinicalTrials.gov intervention name — accepted as the source's own label NCT02800447
Known as NCI-C 01810 ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Known as NSC-77213 “Procarbazine, PCB, NSC-77213NCT00002462
Known as PCB “Procarbazine, PCB, NSC-77213” NCT00002462
Known as Procarbacine ClinicalTrials.gov intervention name — accepted as the source's own label NCT00284271
Known as Procarbazina ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Known as Procarbazine hcl ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Known as procarbazine hydrochloride “Drug: procarbazine hydrochlorideNCT00002569
13

“Drug: procarbazine hydrochlorideNCT00079105

“Drug: Procarbazine HydrochlorideNCT00002463

“Drug: procarbazine hydrochlorideNCT00003375

“Drug: procarbazine hydrochlorideNCT00049595

“Drug: procarbazine hydrochlorideNCT00678327

“Drug: procarbazine hydrochlorideNCT00666484

procarbazine hydrochlorideNCT00002840

NCT05675410

NCT00822120

NCT01775475

NCT00003929

NCT00734773

NCT00003113

Known as Procarbazini hydrochloridum ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Known as RO 4 6467/1 ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Known as RO 4-646711 ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Known as RO-4-6467 ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Known as RO-4-6467 FREE BASE ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Known as RO-4-6467 HYDROCHLORIDE ChEMBL registry synonym — accepted as the source's own label CHEMBL1321
Modality Small molecule CHEMBL1321
Route Oral oral procarbazine and oral prednisone on days 1-10” NCT00002463